DK175986A - Substituerede 2-(n-alkynyl-n-phenylamino)imidazolin-derivater - Google Patents

Substituerede 2-(n-alkynyl-n-phenylamino)imidazolin-derivater Download PDF

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Publication number
DK175986A
DK175986A DK175986A DK175986A DK175986A DK 175986 A DK175986 A DK 175986A DK 175986 A DK175986 A DK 175986A DK 175986 A DK175986 A DK 175986A DK 175986 A DK175986 A DK 175986A
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DK
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Prior art keywords
phenylamino
substituted
alkynyl
imidazoline derivatives
imidazoline
Prior art date
Application number
DK175986A
Other languages
English (en)
Other versions
DK175986D0 (da
Inventor
Franz Esser
Helmut Staehle
Herbert Koeppe
Wolfgang Abele
Ludwig Pichler
Walter Kobinger
Dietrich Arndts
Original Assignee
Boehringer Ingelheim Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Kg filed Critical Boehringer Ingelheim Kg
Publication of DK175986D0 publication Critical patent/DK175986D0/da
Publication of DK175986A publication Critical patent/DK175986A/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/44—Nitrogen atoms not forming part of a nitro radical
    • C07D233/50—Nitrogen atoms not forming part of a nitro radical with carbocyclic radicals directly attached to said nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/08—Vasodilators for multiple indications
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Cardiology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Description

mindste med alkyl eller alkoxy, der igen kan være halogensubstitueret; n er 1, 2 eller 3; samt deres syreadditionssalte.
Forbindelserne fremstilles ved forskellige fremgangsmåder; de besidder værdifulde farmakologiske og terapeutiske egenskaber.
DK175986A 1985-04-20 1986-04-17 Substituerede 2-(n-alkynyl-n-phenylamino)imidazolin-derivater DK175986A (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE3514351A DE3514351A1 (de) 1985-04-20 1985-04-20 Neue substituierte 2-(n-alkinyl-n-phenyl)amino)-imidazolinderivate, deren saeureadditionssalze, diese enthaltende arzneimittel und verfahren zu deren herstellung
DE3514351 1985-04-20

Publications (2)

Publication Number Publication Date
DK175986D0 DK175986D0 (da) 1986-04-17
DK175986A true DK175986A (da) 1986-10-21

Family

ID=6268710

Family Applications (1)

Application Number Title Priority Date Filing Date
DK175986A DK175986A (da) 1985-04-20 1986-04-17 Substituerede 2-(n-alkynyl-n-phenylamino)imidazolin-derivater

Country Status (9)

Country Link
EP (1) EP0202461A1 (da)
JP (1) JPS61249970A (da)
AU (1) AU5637786A (da)
DE (1) DE3514351A1 (da)
DK (1) DK175986A (da)
ES (1) ES8704463A1 (da)
FI (1) FI861643L (da)
IL (1) IL78537A0 (da)
ZA (1) ZA862923B (da)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2592042B1 (fr) * 1985-12-19 1988-03-25 Ile De France Nouveaux ortho-anisamides, leur procede d'obtention, et leurs applications therapeutiques
US6703409B2 (en) 2002-01-31 2004-03-09 Boehringer Ingelheim Pharma Gmbh & Co Kg 2′-Halo-3′,5′-dialkoxyphen-1′-yl-imino-2-imidazolidine and the use thereof as a drug
EP1333028A1 (en) * 2002-01-31 2003-08-06 Boehringer Ingelheim Pharma GmbH & Co.KG 2'-Halo-3',5'-dialkoxyphen-1'-yl-imino-2-imidazolidine derivatives and the use thereof for the treatment of urinary incontinence

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2523103C3 (de) * 1975-05-24 1979-11-29 C.H. Boehringer Sohn, 6507 Ingelheim Substituierte 2-[N-Progargyl-N-(2-chlorphenyl)amino] -imidazoline-^), deren Säureadditionssalze, Verfahren zu ihrer Herstellung und deren Verwendung
DE2831671A1 (de) * 1978-07-19 1980-02-07 Boehringer Sohn Ingelheim Neue substituierte 2-phenylamino-imidazoline-(2), deren saeureadditionssalze, diese enthaltende arzneimittel und verfahren zur herstellung derselben
DE2947563A1 (de) * 1979-11-26 1981-06-04 C.H. Boehringer Sohn, 6507 Ingelheim Neue substituierte 2-phenylamino-imidazoline-(2), deren saeureadditionssalze, diese enthaltende arzneimittel und verfahren zur herstellung derselben

Also Published As

Publication number Publication date
ZA862923B (en) 1987-12-30
IL78537A0 (en) 1986-08-31
DK175986D0 (da) 1986-04-17
AU5637786A (en) 1986-10-23
FI861643A7 (fi) 1986-10-21
FI861643A0 (fi) 1986-04-18
ES8704463A1 (es) 1987-04-01
ES554133A0 (es) 1987-04-01
FI861643L (fi) 1986-10-21
EP0202461A1 (de) 1986-11-26
JPS61249970A (ja) 1986-11-07
DE3514351A1 (de) 1986-11-06

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