DK1943242T3 - Piperidin-4-yl-pyridazin-3-ylamin-derivater som hurtigt opløsende antagonister af dopamin-2-receptorer - Google Patents

Piperidin-4-yl-pyridazin-3-ylamin-derivater som hurtigt opløsende antagonister af dopamin-2-receptorer

Info

Publication number: DK1943242T3
Authority: DK; Denmark
Prior art keywords: pyridazin; dopamine; piperidin; antagonists; receptors
Prior art date: 2005-10-26

Application number

DK06807495.4T

Other languages

English (en)

Inventor

Bruyn Marcel Frans Leopold De

Gregor James Macdonald

Ludo Edmond Josephine Kennis

Xavier Jean Michel Langlois

Den Keybus Frans Alfons Maria Van

Roosbroeck Yves Emiel Maria Van

Original Assignee

Janssen Pharmaceutica Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-10-26

Filing date

2006-10-24

Publication date

2011-04-26

2006-10-24 Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv

2011-04-26 Application granted granted Critical

2011-04-26 Publication of DK1943242T3 publication Critical patent/DK1943242T3/da

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/50—Pyridazines; Hydrogenated pyridazines
- A61K31/501—Pyridazines; Hydrogenated pyridazines not condensed and containing further heterocyclic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings

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Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Epidemiology (AREA)
Psychiatry (AREA)
Pain & Pain Management (AREA)
Hospice & Palliative Care (AREA)
Psychology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

DK06807495.4T 2005-10-26 2006-10-24 Piperidin-4-yl-pyridazin-3-ylamin-derivater som hurtigt opløsende antagonister af dopamin-2-receptorer DK1943242T3 (da)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
EP05110028		2005-10-26
EP06100209		2006-01-10
EP06101545		2006-02-10
PCT/EP2006/067696 WO2007048779A1 (en)	2005-10-26	2006-10-24	Piperidin-4-yl-pyridazin-3-ylamine derivatives as fast dissociating dopamine 2 receptor antagonists

Publications (1)

Publication Number	Publication Date
DK1943242T3 true DK1943242T3 (da)	2011-04-26

Family

ID=35734993

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK06807495.4T DK1943242T3 (da)	2005-10-26	2006-10-24	Piperidin-4-yl-pyridazin-3-ylamin-derivater som hurtigt opløsende antagonister af dopamin-2-receptorer

Country Status (34)

Country	Link
US (3)	US8940743B2 (da)
EP (1)	EP1943242B1 (da)
JP (1)	JP5140598B2 (da)
KR (1)	KR101351910B1 (da)
CN (1)	CN101291925B (da)
AP (1)	AP2607A (da)
AR (1)	AR058151A1 (da)
AT (1)	ATE495167T1 (da)
AU (1)	AU2006307930B2 (da)
BR (1)	BRPI0617787A2 (da)
CA (1)	CA2623160C (da)
CR (1)	CR10020A (da)
CY (1)	CY1111977T1 (da)
DE (1)	DE602006019624D1 (da)
DK (1)	DK1943242T3 (da)
EA (1)	EA015681B1 (da)
EC (1)	ECSP088396A (da)
ES (1)	ES2359020T3 (da)
GT (1)	GT200800033A (da)
HN (1)	HN2008000646A (da)
HR (1)	HRP20110226T1 (da)
IL (1)	IL191016A (da)
JO (1)	JO2769B1 (da)
MY (1)	MY145609A (da)
NO (1)	NO20082350L (da)
NZ (1)	NZ566785A (da)
PL (1)	PL1943242T3 (da)
PT (1)	PT1943242E (da)
RS (1)	RS51674B (da)
SI (1)	SI1943242T1 (da)
TW (1)	TWI399373B (da)
UA (1)	UA94058C2 (da)
WO (1)	WO2007048779A1 (da)
ZA (1)	ZA200803668B (da)

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WO2008128996A1 (en)	2007-04-23	2008-10-30	Janssen Pharmaceutica N.V.	Thia(dia)zoles as fast dissociating dopamine 2 receptor antagonists
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2006
- 2006-10-12 JO JO2006368A patent/JO2769B1/en active
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Also Published As

Publication number	Publication date
KR20080067658A (ko)	2008-07-21
GT200800033A (es)	2009-08-20
SI1943242T1 (sl)	2011-05-31
ES2359020T3 (es)	2011-05-17
ATE495167T1 (de)	2011-01-15
JO2769B1 (en)	2014-03-15
AP2008004441A0 (en)	2008-04-30
MY145609A (en)	2012-03-15
US9468640B2 (en)	2016-10-18
NO20082350L (no)	2008-07-01
EP1943242B1 (en)	2011-01-12
US20170022181A1 (en)	2017-01-26
AR058151A1 (es)	2008-01-23
US20080227791A1 (en)	2008-09-18
HRP20110226T1 (hr)	2011-05-31
NZ566785A (en)	2010-03-26
RS51674B (sr)	2011-10-31
AU2006307930B2 (en)	2011-10-06
DE602006019624D1 (de)	2011-02-24
CA2623160A1 (en)	2007-05-03
US9751860B2 (en)	2017-09-05
CN101291925A (zh)	2008-10-22
ZA200803668B (en)	2009-09-30
PL1943242T3 (pl)	2011-06-30
US8940743B2 (en)	2015-01-27
US20150141432A1 (en)	2015-05-21
PT1943242E (pt)	2011-04-06
TW200732321A (en)	2007-09-01
CA2623160C (en)	2013-10-15
HK1124317A1 (en)	2009-07-10
TWI399373B (zh)	2013-06-21
EA200801184A1 (ru)	2008-08-29
KR101351910B1 (ko)	2014-01-16
JP5140598B2 (ja)	2013-02-06
EP1943242A1 (en)	2008-07-16
EA015681B1 (ru)	2011-10-31
IL191016A (en)	2013-10-31
AP2607A (en)	2013-03-05
WO2007048779A1 (en)	2007-05-03
BRPI0617787A2 (pt)	2009-12-01
UA94058C2 (ru)	2011-04-11
JP2009514815A (ja)	2009-04-09
AU2006307930A1 (en)	2007-05-03
CY1111977T1 (el)	2015-11-04
ECSP088396A (es)	2008-05-30
HN2008000646A (es)	2011-02-16
CR10020A (es)	2009-01-16
CN101291925B (zh)	2013-04-10

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