DK200201957A - 10-substituted erythromycin ketolides and methods of making - Google Patents

10-substituted erythromycin ketolides and methods of making Download PDF

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Publication number
DK200201957A
DK200201957A DK200201957A DKPA200201957A DK200201957A DK 200201957 A DK200201957 A DK 200201957A DK 200201957 A DK200201957 A DK 200201957A DK PA200201957 A DKPA200201957 A DK PA200201957A DK 200201957 A DK200201957 A DK 200201957A
Authority
DK
Denmark
Prior art keywords
previously defined
optionally substituted
heteroaryl
substituted
aryl
Prior art date
Application number
DK200201957A
Other languages
Danish (da)
English (en)
Inventor
Gunnes Soelvi
Undheim Kjell
Original Assignee
Alpharma Aps
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Alpharma Aps filed Critical Alpharma Aps
Priority to DK200201957A priority Critical patent/DK200201957A/da
Publication of DK200201957A publication Critical patent/DK200201957A/da
Priority to CA2789415A priority patent/CA2789415C/fr
Priority to EP10010725.9A priority patent/EP2371833A3/fr
Priority to PCT/GB2003/005659 priority patent/WO2004056843A2/fr
Priority to EP10010724.2A priority patent/EP2354147A3/fr
Priority to US10/539,759 priority patent/US7608596B2/en
Priority to AU2003290339A priority patent/AU2003290339B8/en
Priority to CA2509419A priority patent/CA2509419C/fr
Priority to CNA2003801069659A priority patent/CN1729200A/zh
Priority to EP03782698A priority patent/EP1575970A2/fr
Priority to US12/569,926 priority patent/US8076301B2/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Communicable Diseases (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Oncology (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
DK200201957A 2002-12-20 2002-12-20 10-substituted erythromycin ketolides and methods of making DK200201957A (da)

Priority Applications (11)

Application Number Priority Date Filing Date Title
DK200201957A DK200201957A (da) 2002-12-20 2002-12-20 10-substituted erythromycin ketolides and methods of making
EP03782698A EP1575970A2 (fr) 2002-12-20 2003-12-22 Macrolides 10-substitues
EP10010724.2A EP2354147A3 (fr) 2002-12-20 2003-12-22 Antibiotiques à macrolide substituée 10
EP10010725.9A EP2371833A3 (fr) 2002-12-20 2003-12-22 Antibiotiques à macrolide substituée 10
PCT/GB2003/005659 WO2004056843A2 (fr) 2002-12-20 2003-12-22 Macrolides
CA2789415A CA2789415C (fr) 2002-12-20 2003-12-22 Macrolides
US10/539,759 US7608596B2 (en) 2002-12-20 2003-12-22 10-substituted macrolide antibiotics
AU2003290339A AU2003290339B8 (en) 2002-12-20 2003-12-22 10-Substituted macrolide antibiotics
CA2509419A CA2509419C (fr) 2002-12-20 2003-12-22 Macrolides
CNA2003801069659A CN1729200A (zh) 2002-12-20 2003-12-22 大环内酯类
US12/569,926 US8076301B2 (en) 2002-12-20 2009-09-30 10-substituted macrolide antibiotics

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DK200201957A DK200201957A (da) 2002-12-20 2002-12-20 10-substituted erythromycin ketolides and methods of making

Publications (1)

Publication Number Publication Date
DK200201957A true DK200201957A (da) 2003-01-20

Family

ID=8161253

Family Applications (1)

Application Number Title Priority Date Filing Date
DK200201957A DK200201957A (da) 2002-12-20 2002-12-20 10-substituted erythromycin ketolides and methods of making

Country Status (7)

Country Link
US (2) US7608596B2 (fr)
EP (3) EP1575970A2 (fr)
CN (1) CN1729200A (fr)
AU (1) AU2003290339B8 (fr)
CA (2) CA2509419C (fr)
DK (1) DK200201957A (fr)
WO (1) WO2004056843A2 (fr)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB201217310D0 (en) 2012-09-27 2012-11-14 C10 Pharma As Compounds
WO2019046409A1 (fr) 2017-08-30 2019-03-07 Ecolab Usa Inc. Molécules présentant un groupe hydrophobe et deux groupes ioniques hydrophiles identiques et compositions correspondantes
US11084974B2 (en) 2018-08-29 2021-08-10 Championx Usa Inc. Use of multiple charged cationic compounds derived from polyamines for clay stabilization in oil and gas operations
CA3110686C (fr) 2018-08-29 2025-11-04 Ecolab Usa Inc. Composes ioniques a charges multiples derives de polyamines et compositions a base de ces composes et procedes de preparation associes
WO2020047181A1 (fr) 2018-08-29 2020-03-05 Ecolab Usa Inc. Utilisation de composés ioniques à charges multiples dérivés de polyamines pour clarification d'eaux usées
CN116082183A (zh) 2018-08-29 2023-05-09 埃科莱布美国股份有限公司 衍生自多胺的带多个电荷的离子化合物及其组合物和其作为反相破乳剂用于油气操作的用途
US11058111B2 (en) 2018-08-29 2021-07-13 Ecolab Usa Inc. Use of multiple charged cationic compounds derived from primary amines or polyamines for microbial fouling control in a water system
CN113365498B (zh) 2019-01-29 2022-10-25 埃科莱布美国股份有限公司 阳离子糖基化合物用于在水系统中进行微生物结垢控制的用途
CA3136427C (fr) 2019-04-16 2023-10-24 Ecolab Usa Inc. Utilisation de composes cationiques a charges multiples derives de polyamines et leurs compositions pour lutter contre la corrosion dans un reseau d'alimentation en eau
CN117624172B (zh) * 2023-11-29 2024-07-16 山东第一医科大学附属眼科研究所(山东省眼科研究所、山东第一医科大学附属青岛眼科医院) 一种有机分子笼、有机分子笼纳米酶滴眼液及其制备方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6060234A (en) * 1991-01-17 2000-05-09 Abbott Laboratories Polyketide derivatives and recombinant methods for making same
FR2692579B1 (fr) * 1992-06-19 1995-06-02 Roussel Uclaf Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments.
ES2244001T3 (es) * 1996-07-05 2005-12-01 Biotica Technology Limited Eritromicinas y procedimiento para su preparacion.
FR2757168B1 (fr) * 1996-12-12 1999-06-11 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
US6440942B1 (en) * 2000-12-22 2002-08-27 Enanta Pharmaceuticals, Inc. 14-membered macrolides derived from leucomycins
CA2451391A1 (fr) 2001-07-03 2003-01-16 Chiron Corporation Macrolides et cetolides d'erythromycine modifiee c12 a activite antibacterienne
ATE425984T1 (de) * 2002-04-30 2009-04-15 Abbott Lab Trizyklische antibakterielle makrolidderivate
US6992069B2 (en) 2002-04-30 2006-01-31 Yu-Gui Gu Tricyclic macrolide antibacterial compounds

Also Published As

Publication number Publication date
CN1729200A (zh) 2006-02-01
CA2509419C (fr) 2013-07-02
AU2003290339A1 (en) 2004-07-14
US20060241060A1 (en) 2006-10-26
WO2004056843A3 (fr) 2004-10-21
EP1575970A2 (fr) 2005-09-21
AU2003290339B2 (en) 2010-10-28
US20100137234A1 (en) 2010-06-03
EP2371833A3 (fr) 2013-07-03
CA2789415C (fr) 2014-09-09
EP2354147A2 (fr) 2011-08-10
AU2003290339B8 (en) 2011-02-24
EP2354147A3 (fr) 2013-07-03
US7608596B2 (en) 2009-10-27
US8076301B2 (en) 2011-12-13
CA2789415A1 (fr) 2004-07-08
EP2371833A2 (fr) 2011-10-05
WO2004056843A2 (fr) 2004-07-08
CA2509419A1 (fr) 2004-07-08

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