DK265577A - Fremgangsmade til fremstilling af 2-deoxystreptamin-aminoglycosider - Google Patents

Fremgangsmade til fremstilling af 2-deoxystreptamin-aminoglycosider

Info

Publication number: DK265577A
Authority: DK; Denmark
Prior art keywords: preparing; procedure; deoxystreptamine aminoglycosides; deoxystreptamine; aminoglycosides
Prior art date: 1976-06-16

Application number

DK265577A

Other languages

English (en)

Other versions

DK147942C (da

DK147942B (da

Inventor

R M Plews

K Richardson

J R Wright

Original Assignee

Pfizer

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1976-06-16

Filing date

1977-06-15

Publication date

1977-12-17

1976-06-16 Priority claimed from GB24989/76A external-priority patent/GB1530202A/en

1977-06-15 Application filed by Pfizer filed Critical Pfizer

1977-12-17 Publication of DK265577A publication Critical patent/DK265577A/da

1985-01-14 Publication of DK147942B publication Critical patent/DK147942B/da

1985-09-02 Application granted granted Critical

1985-09-02 Publication of DK147942C publication Critical patent/DK147942C/da

Links

DTFAJAKTSMLKAT-JDCCYXBGSA-N 2-deoxystreptamine Chemical compound N[C@H]1C[C@@H](N)[C@H](O)[C@@H](O)[C@@H]1O DTFAJAKTSMLKAT-JDCCYXBGSA-N 0.000 title 1
229940126575 aminoglycoside Drugs 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
- C07H15/20—Carbocyclic rings
- C07H15/22—Cyclohexane rings, substituted by nitrogen atoms
- C07H15/222—Cyclohexane rings substituted by at least two nitrogen atoms
- C07H15/226—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings
- C07H15/234—Cyclohexane rings substituted by at least two nitrogen atoms with at least two saccharide radicals directly attached to the cyclohexane rings attached to non-adjacent ring carbon atoms of the cyclohexane rings, e.g. kanamycins, tobramycin, nebramycin, gentamicin A2
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Engineering & Computer Science (AREA)
Biochemistry (AREA)
Molecular Biology (AREA)
Genetics & Genomics (AREA)
Biotechnology (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
Oncology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Communicable Diseases (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Saccharide Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DK265577A 1976-06-16 1977-06-15 Analogifremgangsmaade til fremstilling af kanamycin a- eller kanamycin b-derivater eller syreadditionssalte deraf DK147942C (da)

Applications Claiming Priority (6)

Application Number	Priority Date	Filing Date	Title
GB2498976		1976-06-16
GB24989/76A GB1530202A (en)	1976-06-16	1976-06-16	Aminoglycosides
GB4014576		1976-09-28
GB4014576		1976-09-28
GB5129476		1976-12-08
GB5129476		1976-12-08

Publications (3)

Publication Number	Publication Date
DK265577A true DK265577A (da)	1977-12-17
DK147942B DK147942B (da)	1985-01-14
DK147942C DK147942C (da)	1985-09-02

Family

ID=27258386

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK265577A DK147942C (da)	1976-06-16	1977-06-15	Analogifremgangsmaade til fremstilling af kanamycin a- eller kanamycin b-derivater eller syreadditionssalte deraf

Country Status (31)

Country	Link
US (1)	US4214074A (da)
JP (1)	JPS52153943A (da)
AR (1)	AR222781A1 (da)
AT (1)	AT350722B (da)
BG (1)	BG28071A3 (da)
CA (1)	CA1075235A (da)
CH (1)	CH606079A5 (da)
CS (1)	CS203157B2 (da)
DD (1)	DD131019A5 (da)
DE (1)	DE2726839C3 (da)
DK (1)	DK147942C (da)
EG (1)	EG12742A (da)
ES (1)	ES459832A1 (da)
FI (1)	FI771873A7 (da)
FR (1)	FR2355029A1 (da)
GR (1)	GR66411B (da)
HU (1)	HU179054B (da)
IE (1)	IE45389B1 (da)
IL (1)	IL52181A (da)
LU (1)	LU77557A1 (da)
MX (1)	MX4323E (da)
NL (1)	NL170736C (da)
NO (1)	NO144851C (da)
NZ (1)	NZ184213A (da)
PH (1)	PH14663A (da)
PL (1)	PL108094B1 (da)
PT (1)	PT66669B (da)
RO (1)	RO73516A (da)
SE (1)	SE7706944L (da)
SU (1)	SU865128A3 (da)
YU (1)	YU132577A (da)

Families Citing this family (14)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DK308878A (da) *	1977-08-18	1979-02-19	Pfizer	Aminoglyosidderivater og fremgangsmaader til deres fremstilling
DE2832268A1 (de) *	1978-07-22	1980-01-31	Bayer Ag	Pseudotrisaccharide
DE2928183A1 (de) *	1979-07-12	1981-01-29	Bayer Ag	1-n-alkylsisomicin-derivate, verfahren zu ihrer herstellung und ihre verwendung als arzneimittel
JPS5931266A (ja) *	1982-08-11	1984-02-20	株式会社日立製作所	エレベ−タ−の制御装置
KR100450607B1 (ko) *	2002-07-11	2004-09-30	경동제약 주식회사	가라민 유도체의 제조방법
US7794713B2 (en)	2004-04-07	2010-09-14	Lpath, Inc.	Compositions and methods for the treatment and prevention of hyperproliferative diseases
US7862812B2 (en)	2006-05-31	2011-01-04	Lpath, Inc.	Methods for decreasing immune response and treating immune conditions
EA017824B1 (ru)	2007-11-21	2013-03-29	Эйкеоджен, Инк.	Антибактериальные аналоги аминогликозида
CA2761756A1 (en) *	2009-05-14	2010-11-18	Achaogen, Inc.	Treatment of urinary tract infections with antibacterial aminoglycoside compounds
WO2010132768A1 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial derivatives of sisomicin
WO2010132765A2 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial aminoglycoside analogs
WO2010132757A2 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial aminoglycoside analogs
WO2010132760A1 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial derivatives of tobramycin
WO2010132759A1 (en)	2009-05-15	2010-11-18	Achaogen, Inc.	Antibacterial derivatives of dibekacin

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1033394A (en) *	1962-04-03	1966-06-22	Rit Rech Ind Therapeut	New therapeutic agents
US4002742A (en) *	1974-03-19	1977-01-11	Schering Corporation	1-N-alkyl-4,6-di-(aminoglycosyl)-1,3-diaminocyclitols, methods for their manufacture, methods for their use as antibacterial agents, and compositions useful therefor
US4000261A (en) *	1974-11-29	1976-12-28	Schering Corporation	5-epi-4,6-di-o-(aminoglycosyl)-2-deoxystreptamines, methods for their manufacture and intermediates useful therein, methods for their use as antibacterial agents and compositions useful therefor
US4000262A (en) *	1974-11-29	1976-12-28	Schering Corporation	5-epi-amino and 5-epi-azido-4,6-di-o-(aminoglycosyl)-2,5-dideoxystreptamines 1-n-alkyl-5-epi-amino and 1-n-alkyl-5-epi-azido-4,6-di-o-(aminoglycosyl)-2,5-dideoxystreptamines
US4062947A (en) *	1975-11-04	1977-12-13	Schering Corporation	Di-N-alkylaminoglycosides, methods for their manufacture and novel intermediates useful therein, method for their use as antibacterial agents and pharmaceutical compositions useful therefor
US4085208A (en) *	1976-06-21	1978-04-18	Schering Corporation	Process for preparing 4,6-di-O-(aminoglycosyl)-1,3-diaminocyclitols and novel 1-epimers and 1-N-alkyl derivatives produced thereby; methods for the use of the 1-epimer derivatives as antibacterial agents and compositions useful therefor

1977
- 1977-05-26 NZ NZ184213A patent/NZ184213A/xx unknown
- 1977-05-27 IL IL52181A patent/IL52181A/xx unknown
- 1977-05-27 YU YU01325/77A patent/YU132577A/xx unknown
- 1977-05-30 EG EG329/77A patent/EG12742A/xx active
- 1977-05-31 PH PH19833A patent/PH14663A/en unknown
- 1977-06-02 MX MX775775U patent/MX4323E/es unknown
- 1977-06-03 AR AR267934A patent/AR222781A1/es active
- 1977-06-03 CA CA279,773A patent/CA1075235A/en not_active Expired
- 1977-06-08 CS CS773790A patent/CS203157B2/cs unknown
- 1977-06-13 AT AT414277A patent/AT350722B/de not_active IP Right Cessation
- 1977-06-13 BG BG036611A patent/BG28071A3/xx unknown
- 1977-06-14 NO NO772089A patent/NO144851C/no unknown
- 1977-06-14 NL NLAANVRAGE7706514,A patent/NL170736C/xx not_active IP Right Cessation
- 1977-06-14 DE DE2726839A patent/DE2726839C3/de not_active Expired
- 1977-06-14 GR GR53699A patent/GR66411B/el unknown
- 1977-06-14 FI FI771873A patent/FI771873A7/fi not_active Application Discontinuation
- 1977-06-14 PT PT66669A patent/PT66669B/pt unknown
- 1977-06-15 HU HU77PI580A patent/HU179054B/hu unknown
- 1977-06-15 DD DD7700199503A patent/DD131019A5/xx unknown
- 1977-06-15 PL PL1977198872A patent/PL108094B1/pl not_active IP Right Cessation
- 1977-06-15 RO RO7790693A patent/RO73516A/ro unknown
- 1977-06-15 CH CH737577A patent/CH606079A5/xx not_active IP Right Cessation
- 1977-06-15 SU SU772494017A patent/SU865128A3/ru active
- 1977-06-15 JP JP7094477A patent/JPS52153943A/ja active Granted
- 1977-06-15 SE SE7706944A patent/SE7706944L/xx not_active Application Discontinuation
- 1977-06-15 FR FR7718367A patent/FR2355029A1/fr active Granted
- 1977-06-15 IE IE1222/77A patent/IE45389B1/en unknown
- 1977-06-15 DK DK265577A patent/DK147942C/da not_active IP Right Cessation
- 1977-06-16 LU LU77557A patent/LU77557A1/xx unknown
- 1977-06-16 ES ES459832A patent/ES459832A1/es not_active Expired
1978
- 1978-11-07 US US05/958,409 patent/US4214074A/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
CH606079A5 (da)	1978-10-13
IL52181A0 (en)	1977-07-31
SE7706944L (sv)	1977-12-17
PL198872A1 (pl)	1978-03-13
RO73516A (ro)	1981-08-30
IE45389L (en)	1977-12-16
FR2355029A1 (fr)	1978-01-13
NO144851C (no)	1981-11-25
DK147942C (da)	1985-09-02
DE2726839A1 (de)	1978-03-09
NZ184213A (en)	1980-05-27
SU865128A3 (ru)	1981-09-15
NL7706514A (nl)	1977-12-20
FI771873A7 (da)	1977-12-17
AU2551177A (en)	1978-04-13
IL52181A (en)	1981-03-31
EG12742A (en)	1979-12-31
DE2726839B2 (de)	1979-08-30
PT66669B (en)	1978-11-13
IE45389B1 (en)	1982-08-11
PH14663A (en)	1981-10-20
NL170736C (nl)	1982-12-16
LU77557A1 (fr)	1979-03-26
MX4323E (es)	1982-03-24
DK147942B (da)	1985-01-14
AR222781A1 (es)	1981-06-30
ES459832A1 (es)	1978-12-16
BG28071A3 (bg)	1980-02-25
DE2726839C3 (de)	1980-05-14
NO772089L (no)	1977-12-19
JPS52153943A (en)	1977-12-21
FR2355029B1 (da)	1980-04-18
NO144851B (no)	1981-08-17
JPS5713556B2 (da)	1982-03-17
DD131019A5 (de)	1978-05-24
ATA414277A (de)	1978-11-15
PL108094B1 (pl)	1980-03-31
PT66669A (en)	1977-07-01
CS203157B2 (en)	1981-02-27
HU179054B (en)	1982-08-28
AT350722B (de)	1979-06-11
US4214074A (en)	1980-07-22
GR66411B (da)	1981-03-20
CA1075235A (en)	1980-04-08
YU132577A (en)	1982-06-30

Legal Events

Date	Code	Title	Description
1987-03-02	PBP	Patent lapsed

Publication	Publication Date	Title
DK13177A (da)	1977-07-15	Fremgangsmade til fremstilling af phthalaner
DK116177A (da)	1977-09-18	Fremgangsmade til fremstilling af hentriakontapeptider
DK155733C (da)	1989-09-25	Fremgangsmaade til fremstilling af 4-hydroxy-2-oxo-pyrrolidinderivater
DK349478A (da)	1979-02-10	Fremgangsmaade til fremstilling af oligoimider
DK155279C (da)	1989-07-24	Fremgangsmaade til fremstilling af 4-hydroxy-2-oxo-pyrrolidinderivater
DK147777A (da)	1977-10-03	Fremgangsmade til fremstilling af acylchromaner
DK566777A (da)	1978-06-21	Fremgangsmaade til fremstilling af nucleosider
DK364178A (da)	1979-02-19	Fremgangsmaade til fremstilling af antibiotikum
DK243176A (da)	1976-12-04	Fremgangsmade til fremstilling af polycliske forbindelser
DK265577A (da)	1977-12-17	Fremgangsmade til fremstilling af 2-deoxystreptamin-aminoglycosider
IT1076788B (it)	1985-04-27	Procedimento per preparare organopolisilossani
DK144177A (da)	1977-10-03	Fremgangsmade til fremstilling af acylayanider
DK324776A (da)	1977-01-29	Fremgangsmade til fremstilling af 3-cyanoimino-3-aminopropionitriler
DK117677A (da)	1977-09-19	Fremgangsmade til fremstilling af piperidinderivater
DK329577A (da)	1978-01-23	Fremgangsmade til fremstilling af derivater af phenoxyhydroxypropylamin
DK145877A (da)	1977-10-03	Fremgangsmade til immoblisering af glucoseisomerase
DK305876A (da)	1977-01-09	Fremgangsmade til fremstilling af l-pyroglutamyl-l-prolinamid
DK143137C (da)	1981-11-09	Fremgangsmaade til fremstilling af phosphitchlorider
DK143281C (da)	1981-12-07	Fremgangsmaade til fremstilling af phosphitchlorider
DK428377A (da)	1978-03-31	Fremgangsmaade til fremstilling af pyridobenzodiazepinoner
DK310777A (da)	1978-01-10	Fremgangsmade til fremstilling af guaiacol-p-isobutyl-hydratropat
DK385478A (da)	1979-03-20	Fremgangsmaade til fremstilling af dibenzocycloocteniminer
DK86177A (da)	1977-08-27	Fremgangsmade til fremstilling af et antibiotikum
DK156955C (da)	1990-02-26	Fremgangsmaade til fremstilling af cyanosubstituerede cyclopropanderivater
DK88677A (da)	1977-09-02	Fremgangsmade til fremstilling af substituerede puriner