DK265780A - Enkaphalinderivater deres fremstilling og anvendelse som analgetika og antipsychotika mellemprodukter hertil samt disses fremstilling - Google Patents

Enkaphalinderivater deres fremstilling og anvendelse som analgetika og antipsychotika mellemprodukter hertil samt disses fremstilling

Info

Publication number
DK265780A
DK265780A DK265780A DK265780A DK265780A DK 265780 A DK265780 A DK 265780A DK 265780 A DK265780 A DK 265780A DK 265780 A DK265780 A DK 265780A DK 265780 A DK265780 A DK 265780A
Authority
DK
Denmark
Prior art keywords
preparation
encaphalin
analgetics
antipsychotics
intermediates
Prior art date
Application number
DK265780A
Other languages
English (en)
Inventor
A A Carr
R A Farr
J M Kane
Original Assignee
Richardson Merrell Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Richardson Merrell Inc filed Critical Richardson Merrell Inc
Publication of DK265780A publication Critical patent/DK265780A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06—Dipeptides
    • C07K5/06139—Dipeptides with the first amino acid being heterocyclic
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D241/00—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings
    • C07D241/02—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings
    • C07D241/06—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members
    • C07D241/08—Heterocyclic compounds containing 1,4-diazine or hydrogenated 1,4-diazine rings not condensed with other rings having one or two double bonds between ring members or between ring members and non-ring members with oxygen atoms directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/10—Tetrapeptides
    • C07K5/1024—Tetrapeptides with the first amino acid being heterocyclic
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Biophysics (AREA)
  • General Health & Medical Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Molecular Biology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
DK265780A 1979-06-21 1980-06-20 Enkaphalinderivater deres fremstilling og anvendelse som analgetika og antipsychotika mellemprodukter hertil samt disses fremstilling DK265780A (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US5095079A 1979-06-21 1979-06-21
US06/130,431 US4341698A (en) 1979-06-21 1980-03-14 Enkaphalin derivatives
AU91877/82A AU559278B2 (en) 1979-06-21 1982-12-24 Piperazines

Publications (1)

Publication Number Publication Date
DK265780A true DK265780A (da) 1980-12-22

Family

ID=36764304

Family Applications (1)

Application Number Title Priority Date Filing Date
DK265780A DK265780A (da) 1979-06-21 1980-06-20 Enkaphalinderivater deres fremstilling og anvendelse som analgetika og antipsychotika mellemprodukter hertil samt disses fremstilling

Country Status (17)

Country Link
US (1) US4341698A (da)
AU (1) AU559278B2 (da)
CA (1) CA1161838A (da)
CH (2) CH645363A5 (da)
DE (1) DE3022401A1 (da)
DK (1) DK265780A (da)
ES (1) ES8105720A1 (da)
FR (2) FR2459236A1 (da)
GB (3) GB2051821B (da)
IE (1) IE49834B1 (da)
IL (1) IL60245A (da)
IT (1) IT1148277B (da)
NL (1) NL8003580A (da)
NO (1) NO801855L (da)
NZ (1) NZ193934A (da)
PH (1) PH19222A (da)
SE (3) SE447250B (da)

Families Citing this family (23)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6194435B1 (en) 1996-10-11 2001-02-27 Cor Therapeutics, Inc. Lactams as selective factor Xa inhibitors
US6262047B1 (en) 1996-10-11 2001-07-17 Cor Therapeutics, Inc. Selective factor Xa inhibitors
US6369080B2 (en) 1996-10-11 2002-04-09 Cor Therapeutics, Inc. Selective factor Xa inhibitors
US6063794A (en) 1996-10-11 2000-05-16 Cor Therapeutics Inc. Selective factor Xa inhibitors
AU6896398A (en) 1997-04-14 1998-11-11 Cor Therapeutics, Inc. Selective factor xa inhibitors
NZ500353A (en) 1997-04-14 2002-02-01 Cor Therapeutics Inc Cyclic diaza compounds that are selective inhibitors of factor Xa
AU741099B2 (en) * 1997-04-14 2001-11-22 Millennium Pharmaceuticals, Inc. Selective factor Xa inhibitors
US6218382B1 (en) 1997-08-11 2001-04-17 Cor Therapeutics, Inc Selective factor Xa inhibitors
US6333321B1 (en) 1997-08-11 2001-12-25 Cor Therapeutics, Inc. Selective factor Xa inhibitors
US6228854B1 (en) 1997-08-11 2001-05-08 Cor Therapeutics, Inc. Selective factor Xa inhibitors
EP1868434A4 (en) 2005-03-22 2011-10-26 Azevan Pharmaceuticals Inc BETA-LACTAMYL ALKANIC ACIDS FOR THE TREATMENT OF PREMIERSTRUELLEN FAULTS
TR201907381T4 (tr) 2005-07-19 2019-06-21 Azevan Pharmaceuticals Inc Beta-laktamil fenilalanin, sistein ve serin vazopressin antagonisti.
MX2008012663A (es) * 2006-03-30 2008-10-13 Palatin Technologies Inc Constructos ciclicos de peptidos natriureticos.
US7964181B2 (en) * 2006-03-30 2011-06-21 Palatin Technologies, Inc. Amino acid surrogates for peptidic constructs
US8114844B2 (en) * 2006-03-30 2012-02-14 Palatin Technologies, Inc. Linear and cyclic melanocortin receptor-specific peptidomimetics
CA2647114C (en) * 2006-03-30 2016-10-11 Palatin Technologies, Inc. Amino acid surrogates for peptidic constructs
US8580746B2 (en) 2006-03-30 2013-11-12 Palatin Technologies, Inc. Amide linkage cyclic natriuretic peptide constructs
AU2007233123A1 (en) * 2006-03-30 2007-10-11 Palatin Technologies, Inc. Linear natriuretic peptide constructs
PL2354124T3 (pl) * 2006-12-19 2013-07-31 Hoffmann La Roche Pochodne heteroarylopirolidynylo- i piperydynyloketonów
AU2009259492A1 (en) * 2008-06-18 2009-12-23 F. Hoffmann-La Roche Ag Aryl ketone as MRI
ES2662350T3 (es) 2010-07-01 2018-04-06 Azevan Pharmaceuticals, Inc. Procedimientos para el tratamiento del trastorno por estrés postraumático
AU2015237253B2 (en) 2014-03-28 2019-11-14 Azevan Pharmaceuticals, Inc. Compositions and methods for treating neurodegenerative diseases
MY208313A (en) 2017-09-15 2025-04-30 Azevan Pharmaceuticals Inc Compositions and methods for treating brain injury

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2604845A1 (de) * 1976-02-07 1977-08-18 Knoll Ag Neue piperazinderivate
US4254107A (en) * 1979-11-27 1981-03-03 Merck & Co., Inc. Long-lasting agonists of enkephalin

Also Published As

Publication number Publication date
PH19222A (en) 1986-02-12
IT8049032A0 (it) 1980-06-20
IT1148277B (it) 1986-11-26
DE3022401A1 (de) 1981-01-08
ES492566A0 (es) 1981-06-16
SE447250B (sv) 1986-11-03
IE49834B1 (en) 1985-12-25
NL8003580A (nl) 1980-12-23
GB2132605B (en) 1985-01-03
CH645363A5 (de) 1984-09-28
GB2051821A (en) 1981-01-21
SE460540B (sv) 1989-10-23
NZ193934A (en) 1983-02-15
AU559278B2 (en) 1987-03-05
FR2473042B1 (da) 1983-07-01
SE8004254L (sv) 1980-12-22
GB2051821B (en) 1983-04-27
SE8500877D0 (sv) 1985-02-22
FR2459236B1 (da) 1984-01-06
US4341698A (en) 1982-07-27
GB2106515A (en) 1983-04-13
FR2473042A1 (fr) 1981-07-10
SE460541B (sv) 1989-10-23
CA1161838A (en) 1984-02-07
CH648835A5 (de) 1985-04-15
GB2132605A (en) 1984-07-11
NO801855L (no) 1980-12-22
SE8500878D0 (sv) 1985-02-22
IL60245A (en) 1985-08-30
SE8500877L (sv) 1985-02-22
ES8105720A1 (es) 1981-06-16
AU9187782A (en) 1983-04-21
FR2459236A1 (fr) 1981-01-09
GB2106515B (en) 1983-11-23
IE801152L (en) 1980-12-21

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Legal Events

Date Code Title Description
AHS Application shelved for other reasons than non-payment