DK266083A - Fremgangsmaade til fremstilling af 2-heterocyclyl-1,3-bis(1h-1,2,4-triazol-1-yl)propan-2-oler eller farmaceutisk acceptable syreadditionssalte deraf - Google Patents
Fremgangsmaade til fremstilling af 2-heterocyclyl-1,3-bis(1h-1,2,4-triazol-1-yl)propan-2-oler eller farmaceutisk acceptable syreadditionssalte deraf Download PDFInfo
- Publication number
- DK266083A DK266083A DK266083A DK266083A DK266083A DK 266083 A DK266083 A DK 266083A DK 266083 A DK266083 A DK 266083A DK 266083 A DK266083 A DK 266083A DK 266083 A DK266083 A DK 266083A
- Authority
- DK
- Denmark
- Prior art keywords
- triazol
- propan
- heterocyclyl
- bis
- oles
- Prior art date
Links
- -1 1H-1,2,4-TRIAZOL-1-YL Chemical class 0.000 title 1
- 239000002253 acid Substances 0.000 title 1
- 150000003839 salts Chemical class 0.000 title 1
- 206010017533 Fungal infection Diseases 0.000 abstract 1
- 241001465754 Metazoa Species 0.000 abstract 1
- 208000031888 Mycoses Diseases 0.000 abstract 1
- 229940121375 antifungal agent Drugs 0.000 abstract 1
- 239000003429 antifungal agent Substances 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing three or more hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/60—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings condensed with carbocyclic rings or ring systems
- C07D277/62—Benzothiazoles
- C07D277/68—Benzothiazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
- C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D213/61—Halogen atoms or nitro radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/10—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D231/12—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
- C07D233/56—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, attached to ring carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D249/00—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms
- C07D249/02—Heterocyclic compounds containing five-membered rings having three nitrogen atoms as the only ring hetero atoms not condensed with other rings
- C07D249/08—1,2,4-Triazoles; Hydrogenated 1,2,4-triazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
- C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
- C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
- C07D333/26—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D333/28—Halogen atoms
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB8217114 | 1982-06-12 | ||
| GB8217114 | 1982-06-12 |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| DK266083D0 DK266083D0 (da) | 1983-06-10 |
| DK266083A true DK266083A (da) | 1983-12-13 |
| DK160825B DK160825B (da) | 1991-04-22 |
| DK160825C DK160825C (da) | 1991-10-14 |
Family
ID=10531001
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK266083A DK160825C (da) | 1982-06-12 | 1983-06-10 | Analogifremgangsmaade til fremstilling af 2-(halogensubstitueret pyridyl)-1,3-bis(1h-1,2,4-triazol-1-yl)propan-2-ol-derivater eller farmaceutisk acceptable syreadditionssalte deraf |
Country Status (16)
| Country | Link |
|---|---|
| US (1) | US4510148A (da) |
| EP (1) | EP0097014B1 (da) |
| JP (1) | JPS5962587A (da) |
| KR (1) | KR870000358B1 (da) |
| AT (1) | ATE24909T1 (da) |
| AU (1) | AU542450B2 (da) |
| CA (1) | CA1238909A (da) |
| DE (1) | DE3369137D1 (da) |
| DK (1) | DK160825C (da) |
| ES (1) | ES8407488A1 (da) |
| FI (1) | FI74465C (da) |
| GR (1) | GR77534B (da) |
| IE (1) | IE55233B1 (da) |
| IL (1) | IL68945A (da) |
| PH (1) | PH21493A (da) |
| PT (1) | PT76846B (da) |
Families Citing this family (14)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8305377D0 (en) * | 1983-02-25 | 1983-03-30 | Pfizer Ltd | Antifungal agents |
| GB8306351D0 (en) * | 1983-03-08 | 1983-04-13 | Ici Plc | Azole fungicides |
| DK159205C (da) * | 1983-03-16 | 1991-03-04 | Pfizer | Bis(triazol)alkanol-forbindelser, anvendelse af disse, farmaceutiske praeparater og landbrugsfungicider indeholdende disse og fremgangsmaade til behandling af planter eller froe, som har en svampeinfektion |
| US4992454A (en) * | 1983-03-16 | 1991-02-12 | Pfizer Inc. | Antifungal 1,3-bis (1H-1,2,4-triazol-1-yl)-2-aryl butan-2-ols and derivatives thereof |
| GB8313235D0 (en) * | 1983-05-13 | 1983-06-22 | Pfizer Ltd | Antifungal agents |
| IE58738B1 (en) * | 1984-09-05 | 1993-11-03 | Ici Plc | Antifungal azole compounds |
| GB8819308D0 (en) * | 1988-08-13 | 1988-09-14 | Pfizer Ltd | Triazole antifungal agents |
| GB9002375D0 (en) * | 1990-02-02 | 1990-04-04 | Pfizer Ltd | Triazole antifungal agents |
| US5068333A (en) * | 1990-03-07 | 1991-11-26 | Pfizer Inc. | 6-chloro-3,4-dihydro-pyrano [2,3-b]pyridines having the R configuration |
| NZ270418A (en) * | 1994-02-07 | 1997-09-22 | Eisai Co Ltd | Polycyclic triazole & imidazole derivatives, antifungal compositions |
| US6291463B1 (en) | 1998-06-30 | 2001-09-18 | Neurogen Corporation | 1-(Benzothiazol-2-yl)-4-(1-phenylmethyl) piperazines: dopamine receptor subtype specific ligands |
| EP1089990A1 (en) * | 1998-06-30 | 2001-04-11 | Neurogen Corporation | 1-(benzothiazol-2-yl)-4-(1-phenylmethyl)piperazines: dopamine receptor subtype specific ligands |
| CN105308032B (zh) * | 2013-04-12 | 2017-05-24 | 拜耳作物科学股份公司 | 新的三唑衍生物 |
| CN106231901A (zh) * | 2014-04-15 | 2016-12-14 | 美国陶氏益农公司 | 作为杀真菌剂的金属酶抑制剂化合物 |
Family Cites Families (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3658813A (en) * | 1970-01-13 | 1972-04-25 | Janssen Pharmaceutica Nv | 1-(beta-aryl-beta-(r-oxy)-ethyl)-imidazoles |
| DE2738725A1 (de) * | 1977-08-27 | 1979-03-08 | Basf Ag | Azolylalkohole |
| DE2926280A1 (de) * | 1979-06-29 | 1981-01-08 | Basf Ag | Fungizide alpha -triazolylglykolderivate, ihre herstellung und verwendung |
| GB2078719B (en) * | 1980-06-02 | 1984-04-26 | Ici Ltd | Heterocyclic compounds |
| EP0046337A3 (en) * | 1980-08-20 | 1982-09-15 | Imperial Chemical Industries Plc | Triazole compounds, a process for preparing them, their use as plant and pharmaceutical fungicides and as plant growth regulators and compositions containing them |
| JPS5758671A (en) * | 1980-09-25 | 1982-04-08 | Ishihara Sangyo Kaisha Ltd | Phenoxyalkylazole type compound and agricultural and gardening fungicide comprising it |
| GB2099818A (en) * | 1981-06-06 | 1982-12-15 | Pfizer Ltd | Triazoles |
| EP0069442B1 (en) * | 1981-06-06 | 1985-02-20 | Pfizer Limited | Antifungal agents, processes for their preparation, and pharmaceutical compositions containing them |
-
1983
- 1983-05-27 US US06/499,073 patent/US4510148A/en not_active Expired - Lifetime
- 1983-06-07 EP EP83303267A patent/EP0097014B1/en not_active Expired
- 1983-06-07 DE DE8383303267T patent/DE3369137D1/de not_active Expired
- 1983-06-07 AT AT83303267T patent/ATE24909T1/de not_active IP Right Cessation
- 1983-06-08 KR KR1019830002555A patent/KR870000358B1/ko not_active Expired
- 1983-06-09 PT PT76846A patent/PT76846B/pt not_active IP Right Cessation
- 1983-06-09 GR GR71600A patent/GR77534B/el unknown
- 1983-06-10 IE IE1371/83A patent/IE55233B1/en unknown
- 1983-06-10 AU AU15702/83A patent/AU542450B2/en not_active Ceased
- 1983-06-10 DK DK266083A patent/DK160825C/da not_active IP Right Cessation
- 1983-06-10 CA CA000430189A patent/CA1238909A/en not_active Expired
- 1983-06-10 FI FI832101A patent/FI74465C/fi not_active IP Right Cessation
- 1983-06-10 ES ES523146A patent/ES8407488A1/es not_active Expired
- 1983-06-10 IL IL68945A patent/IL68945A/xx not_active IP Right Cessation
- 1983-06-10 PH PH29034A patent/PH21493A/en unknown
- 1983-06-13 JP JP58105637A patent/JPS5962587A/ja active Granted
Also Published As
| Publication number | Publication date |
|---|---|
| DK266083D0 (da) | 1983-06-10 |
| AU1570283A (en) | 1983-12-15 |
| PT76846A (en) | 1983-07-01 |
| KR840005134A (ko) | 1984-11-03 |
| FI832101L (fi) | 1983-12-13 |
| KR870000358B1 (ko) | 1987-03-05 |
| ATE24909T1 (de) | 1987-01-15 |
| EP0097014A2 (en) | 1983-12-28 |
| IE831371L (en) | 1983-12-12 |
| CA1238909A (en) | 1988-07-05 |
| EP0097014A3 (en) | 1984-07-25 |
| IE55233B1 (en) | 1990-07-04 |
| IL68945A0 (en) | 1983-10-31 |
| AU542450B2 (en) | 1985-02-21 |
| FI832101A0 (fi) | 1983-06-10 |
| DK160825C (da) | 1991-10-14 |
| EP0097014B1 (en) | 1987-01-14 |
| FI74465B (fi) | 1987-10-30 |
| PT76846B (en) | 1986-04-09 |
| JPS5962587A (ja) | 1984-04-10 |
| ES523146A0 (es) | 1984-10-01 |
| DE3369137D1 (en) | 1987-02-19 |
| ES8407488A1 (es) | 1984-10-01 |
| GR77534B (da) | 1984-09-24 |
| FI74465C (fi) | 1988-02-08 |
| IL68945A (en) | 1986-09-30 |
| US4510148A (en) | 1985-04-09 |
| DK160825B (da) | 1991-04-22 |
| JPS6330308B2 (da) | 1988-06-17 |
| PH21493A (en) | 1987-11-10 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PBP | Patent lapsed |