DK280783A - Fremgangsmaade til fremstilling af (3s)-3-(((2-amino-4-thiazolyl)-((1-carboxy-1-methyloxy)imino)acetyl)amino)-2-oxo-1-azetidinsulfonsyre og 4-substituerede derivater deraf - Google Patents

Fremgangsmaade til fremstilling af (3s)-3-(((2-amino-4-thiazolyl)-((1-carboxy-1-methyloxy)imino)acetyl)amino)-2-oxo-1-azetidinsulfonsyre og 4-substituerede derivater deraf Download PDF

Info

Publication number: DK280783A
Authority: DK; Denmark
Prior art keywords: amino; methyloxy; imino; oxo; carboxy
Prior art date: 1982-06-21

Application number

DK280783A

Other languages

English (en)

Other versions

DK163510C (da

DK280783D0 (da

DK163510B (da

Inventor

Jerome Leon Moniot

Christopher Michael Cimarusti

Rita Theresa Fox

Original Assignee

Squibb & Sons Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1982-06-21

Filing date

1983-06-17

Publication date

1983-12-22

1983-06-17 Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc

1983-06-17 Publication of DK280783D0 publication Critical patent/DK280783D0/da

1983-12-22 Publication of DK280783A publication Critical patent/DK280783A/da

1992-03-09 Publication of DK163510B publication Critical patent/DK163510B/da

1992-07-27 Application granted granted Critical

1992-07-27 Publication of DK163510C publication Critical patent/DK163510C/da

Links

-1 2-AMINO-4-THIAZOLYL Chemical class 0.000 title 3
101000740162 Homo sapiens Sodium- and chloride-dependent transporter XTRP3 Proteins 0.000 title 1
102100037189 Sodium- and chloride-dependent transporter XTRP3 Human genes 0.000 title 1
125000002777 acetyl group Chemical class [H]C([H])([H])C(*)=O 0.000 title 1
BDHFUVZGWQCTTF-UHFFFAOYSA-N sulfonic acid Chemical compound OS(=O)=O BDHFUVZGWQCTTF-UHFFFAOYSA-N 0.000 title 1
125000000218 acetic acid group Chemical group C(C)(=O)* 0.000 abstract 1
239000002253 acid Substances 0.000 abstract 1
125000001841 imino group Chemical group [H]N=* 0.000 abstract 1
238000004519 manufacturing process Methods 0.000 abstract 1
125000002924 primary amino group Chemical group [H]N([H])* 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D277/00—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings
- C07D277/02—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings
- C07D277/20—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
- C07D277/32—Heterocyclic compounds containing 1,3-thiazole or hydrogenated 1,3-thiazole rings not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D277/38—Nitrogen atoms
- C07D277/44—Acylated amino or imino radicals
- C07D277/46—Acylated amino or imino radicals by carboxylic acids, or sulfur or nitrogen analogues thereof
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Veterinary Medicine (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Oncology (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Communicable Diseases (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Saccharide Compounds (AREA)
Thiazole And Isothizaole Compounds (AREA)
Cephalosporin Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

DK280783A 1982-06-21 1983-06-17 Fremgangsmaade til fremstilling af (3s)-3-oeoe(2-amino-4-thioazolyl)-oe(1-carboxy-1-methylethoxy)iminoaaacetylaaaminoaa-2-oxo-1-azetidinsulfonsyre og 4-alkylsubstituerede derivater deraf samt mellemprodukt til brug ved fremgangsmaaden DK163510C (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US39072882		1982-06-21
US06/390,728 US4704457A (en)	1982-06-21	1982-06-21	Process for the preparation of (3S)-3-[[[2-(protected amino)-4-thiazolyl]-oxoacetyl]amino]-2-oxo-1-azetidinesulfonic acid and 4-substituted derivatives thereof

Publications (4)

Publication Number	Publication Date
DK280783D0 DK280783D0 (da)	1983-06-17
DK280783A true DK280783A (da)	1983-12-22
DK163510B DK163510B (da)	1992-03-09
DK163510C DK163510C (da)	1992-07-27

Family

ID=23543684

Family Applications (3)

Application Number	Title	Priority Date	Filing Date
DK280783A DK163510C (da)	1982-06-21	1983-06-17	Fremgangsmaade til fremstilling af (3s)-3-oeoe(2-amino-4-thioazolyl)-oe(1-carboxy-1-methylethoxy)iminoaaacetylaaaminoaa-2-oxo-1-azetidinsulfonsyre og 4-alkylsubstituerede derivater deraf samt mellemprodukt til brug ved fremgangsmaaden
DK146591A DK166322C (da)	1982-06-21	1991-08-14	Fremgangsmaade til fremstilling af azetidinsulfonsyrederivater
DK106592A DK166209C (da)	1982-06-21	1992-08-27	Mellemprodukt til fremstilling af azetidinsulfonsyrederivater

Family Applications After (2)

Application Number	Title	Priority Date	Filing Date
DK146591A DK166322C (da)	1982-06-21	1991-08-14	Fremgangsmaade til fremstilling af azetidinsulfonsyrederivater
DK106592A DK166209C (da)	1982-06-21	1992-08-27	Mellemprodukt til fremstilling af azetidinsulfonsyrederivater

Country Status (18)

Country	Link
US (1)	US4704457A (da)
EP (1)	EP0097352B1 (da)
JP (1)	JPS597190A (da)
KR (1)	KR880001048B1 (da)
AT (1)	ATE30155T1 (da)
AU (1)	AU563938B2 (da)
CA (1)	CA1205076A (da)
DE (1)	DE3374008D1 (da)
DK (3)	DK163510C (da)
ES (2)	ES523420A0 (da)
GR (1)	GR78278B (da)
HU (3)	HU194560B (da)
IE (1)	IE55234B1 (da)
NO (1)	NO832229L (da)
NZ (1)	NZ204214A (da)
PH (2)	PH18423A (da)
PT (1)	PT76896B (da)
ZA (1)	ZA833623B (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5484928A (en) *	1984-04-10	1996-01-16	Biochemie Gesellschaft M.B.H.	2-(2-aminothiazol-4-yl)-2-oxoacetic acid derivatives
US4647660A (en) *	1985-05-02	1987-03-03	E. R. Squibb & Sons, Inc.	3-acylamino-2-oxo-1-azetidinesulfonic acids
US4675398A (en) *	1985-08-16	1987-06-23	E. R. Squibb & Sons, Inc.	Copper-mediated oximation reaction
US4684722A (en) *	1986-01-06	1987-08-04	E. R. Squibb & Sons, Inc.	Monosulfactams

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1575803A (en) *	1976-03-09	1980-10-01	Fujisawa Pharmaceutical Co	3,7 disubstituted 3 cephem 4 carboxylic acid compounds andprocesses for the preparation thereof
US4166115A (en) *	1976-04-12	1979-08-28	Fujisawa Pharmaceutical Co., Ltd.	Syn 7-oxoimino substituted derivatives of cephalosporanic acid
US4237128A (en) *	1979-04-12	1980-12-02	E. R. Squibb & Sons, Inc.	7-[2-(2-Amino-4-thiazolyl)-2-[(1-carboxy-1,1-dialkyl)alkoxyimino]acetamido]cephem sulfoxides
NZ196202A (en) *	1980-02-07	1984-07-31	Squibb & Sons Inc	Beta-lactam antibiotics (of azetidine-sulphonic acid type)
EP0048953B1 (en) *	1980-09-29	1988-03-09	E.R. Squibb & Sons, Inc.	Beta-lactam antibiotics
US4443374A (en) *	1982-02-01	1984-04-17	E. R. Squibb & Sons, Inc.	Process for preparing (3S)-3-[[(2-amino-4-thiazolyl)[(1-carboxy-1-methylethoxy)imino]-acetyl]amino]-2-oxo-1-azetidinesulfonic acid, and 4-substituted derivatives

1982
- 1982-06-21 US US06/390,728 patent/US4704457A/en not_active Expired - Lifetime
1983
- 1983-05-10 CA CA000427829A patent/CA1205076A/en not_active Expired
- 1983-05-12 NZ NZ204214A patent/NZ204214A/en unknown
- 1983-05-12 AU AU14499/83A patent/AU563938B2/en not_active Expired
- 1983-05-19 ZA ZA833623A patent/ZA833623B/xx unknown
- 1983-05-20 PH PH28939A patent/PH18423A/en unknown
- 1983-06-03 JP JP58100110A patent/JPS597190A/ja active Granted
- 1983-06-03 GR GR71555A patent/GR78278B/el unknown
- 1983-06-13 IE IE1382/83A patent/IE55234B1/en not_active IP Right Cessation
- 1983-06-17 DK DK280783A patent/DK163510C/da not_active IP Right Cessation
- 1983-06-20 EP EP83106005A patent/EP0097352B1/en not_active Expired
- 1983-06-20 HU HU831047A patent/HU194560B/hu unknown
- 1983-06-20 ES ES523420A patent/ES523420A0/es active Granted
- 1983-06-20 DE DE8383106005T patent/DE3374008D1/de not_active Expired
- 1983-06-20 AT AT83106005T patent/ATE30155T1/de not_active IP Right Cessation
- 1983-06-20 HU HU831046A patent/HU194558B/hu unknown
- 1983-06-20 HU HU832191A patent/HU190903B/hu unknown
- 1983-06-20 KR KR1019830002746A patent/KR880001048B1/ko not_active Expired
- 1983-06-20 PT PT76896A patent/PT76896B/pt unknown
- 1983-06-20 NO NO832229A patent/NO832229L/no unknown
1984
- 1984-11-26 ES ES537960A patent/ES8601984A1/es not_active Expired
- 1984-12-10 PH PH31557A patent/PH22121A/en unknown
1991
- 1991-08-14 DK DK146591A patent/DK166322C/da not_active IP Right Cessation
1992
- 1992-08-27 DK DK106592A patent/DK166209C/da not_active IP Right Cessation

Also Published As

Publication number	Publication date
DK163510C (da)	1992-07-27
ZA833623B (en)	1984-02-29
US4704457A (en)	1987-11-03
DK166322C (da)	1993-08-23
EP0097352A3 (en)	1984-09-12
GR78278B (da)	1984-09-26
EP0097352B1 (en)	1987-10-07
DE3374008D1 (en)	1987-11-12
ATE30155T1 (de)	1987-10-15
KR880001048B1 (ko)	1988-06-18
NO832229L (no)	1983-12-22
DK280783D0 (da)	1983-06-17
DK146591A (da)	1991-08-14
JPH0348910B2 (da)	1991-07-25
PT76896A (en)	1983-07-01
DK146591D0 (da)	1991-08-14
NZ204214A (en)	1986-01-24
ES537960A0 (es)	1985-11-01
AU563938B2 (en)	1987-07-30
CA1205076A (en)	1986-05-27
IE55234B1 (en)	1990-07-04
PH22121A (en)	1988-06-01
DK163510B (da)	1992-03-09
JPS597190A (ja)	1984-01-14
ES8503682A1 (es)	1985-03-16
KR840005114A (ko)	1984-11-03
HU190903B (en)	1986-12-28
AU1449983A (en)	1984-01-05
PH18423A (en)	1985-06-26
ES523420A0 (es)	1985-03-16
PT76896B (en)	1986-01-24
DK106592D0 (da)	1992-08-27
HU194558B (en)	1988-02-29
ES8601984A1 (es)	1985-11-01
DK166209C (da)	1993-08-16
HU194560B (en)	1988-02-29
EP0097352A2 (en)	1984-01-04
DK106592A (da)	1992-08-27
DK166209B (da)	1993-03-22
IE831382L (en)	1983-12-21
DK166322B (da)	1993-04-05

Legal Events

Date	Code	Title	Description
2003-07-07	PUP	Patent expired

Publication	Publication Date	Title
KR850002742A (ko)	1985-05-15	아미노산 유도체의 제조방법
DK144783D0 (da)	1983-03-29	Fremgangsmade til fremstilling af cycloalka(c)pyrrol-carboxylsyrederivater
DE3683791D1 (de)	1992-03-19	Verfahren zur digitalen datenfehlerkorrektur.
AU6845990A (en)	1991-07-04	Karl-fishcher reagent and a process for the determination of water with the aid of this reagent
DK166087C (da)	1993-08-23	Fremgangsmaade til fremstilling af oe(3-amino-3-carboxy)-propyl-1aaphosphinsyrederivater
DK280783D0 (da)	1983-06-17	Fremgangsmade til fremstilling af (3s)-3-(((2-amino-4-thiazolyl)-((1-carboxy-1-methyl-oxy)imino)acetyl)amino)-2-oxo-1-azetidinsulfonsyre og 4-substituerede derivater deraf
DK82682A (da)	1982-08-28	Fremgangsmaade til fremstilling af threo-2-hydroxy-3-(4-methoxyphenyl)-3-(2-nitrophenylthio)-propionsyreestere
DK442083D0 (da)	1983-09-27	Fremgangsmade til fremstilling af mikrobiel alkalisk protease
FI831253A7 (fi)	1983-10-20	Menetelmä uusien oksatsolijohdosten valmistamiseksi.
FI872784A7 (fi)	1987-12-24	Menetelmä terapeuttisesti käyttökelpoisten 2-okso-1-//(substituoitu sulfonyyli)amino/karbonyyli/atsetidiinien valmistamiseksi
FI834340A7 (fi)	1984-05-30	Menetelmä terapeuttisesti käyttökelpoisten rikkipitoisten bentsylideenijohdannaisten valmistamiseksi.
DK541882A (da)	1983-06-09	Fremgangsmaade til fremstilling af n-(vinblastinoyl-23)-derivater af aminosyrer
FI893478L (fi)	1989-07-18	Menetelmä uusien kysteiinijohdannaisten valmistamiseksi
DK148096C (da)	1985-08-12	Fremgangsmaade til fremstilling af (2-aminothiazol-4-yl)-eddikesyre-hydrochlorid
DK193580A (da)	1980-11-05	Fremgangsmaade til fremstilling af 5-(2-( (2,3-dihydro-1,4-benzodioxan-2-yl-methyl)amino)-1-hydroxyethyl)-2-hydroxybenzoesyre-derivater
DK356288D0 (da)	1988-06-28	Fremgangsmaade til fremstilling af n-((4-hydroxy-pyrrolidin-2-on-1-yl)-acetyl)-glycinamid
DK277688A (da)	1988-11-24	Fremgangsmaade til fremstilling af et hmg-coa-lignende protein
FI810542A7 (fi)	1981-08-29	Menetelmä heterosyklisten tioyhdisteiden valmistamiseksi.
FI883139A7 (fi)	1989-01-03	Menetelmä L-fenyylialaniinin valmistamiseksi bentsylideenihydantoiinista.
FI901703A7 (fi)	1991-10-05	Menetelmä kliinisesti tärkeiden metaboliittien määräämiseksi
DK457485D0 (da)	1985-10-08	Polyether-antibiotikum benaevnt a80190 og derivater heraf samt fremgangsmaade til fremstilling af saadanne forbindelser
FI832960A7 (fi)	1984-02-20	Menetelmä angiotensiiniä muuttavan entsyymin inhibiittorien valmistamiseksi.
DK395087D0 (da)	1987-07-29	Fremgangsmaade til fremstilling af n-sulfonyl-n-(phosphonomethylglycyl)aminderivater
DK435381A (da)	1983-04-02	Fremgangsmaade til fremstilling af n-(1-formylamido-2,2,2-trichlorethyl)-morpholin