DK287085A - Triazolobenzodiazepin og farmaceutisk praeparat indeholdende en saadanforbindelse - Google Patents
Triazolobenzodiazepin og farmaceutisk praeparat indeholdende en saadanforbindelse Download PDFInfo
- Publication number
- DK287085A DK287085A DK287085A DK287085A DK287085A DK 287085 A DK287085 A DK 287085A DK 287085 A DK287085 A DK 287085A DK 287085 A DK287085 A DK 287085A DK 287085 A DK287085 A DK 287085A
- Authority
- DK
- Denmark
- Prior art keywords
- triazolobenzodiazepine
- pharmaceutical preparation
- preparation containing
- seed connection
- seed
- Prior art date
Links
- 239000000825 pharmaceutical preparation Substances 0.000 title 1
- KYTREVLPRJOBEM-UHFFFAOYSA-N triazolo[4,5-i][1,2]benzodiazepine Chemical compound C1=CC2=CC=CN=NC2=C2C1=NN=N2 KYTREVLPRJOBEM-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
- C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
- C07D243/20—Nitrogen atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
- C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
- C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
- C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
- C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals
- C07D243/18—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals substituted in position 2 by nitrogen, oxygen or sulfur atoms
- C07D243/22—Sulfur atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US62485084A | 1984-06-26 | 1984-06-26 | |
| US06/741,971 US4663321A (en) | 1984-06-26 | 1985-06-10 | Triazolobenzodiazepines and pharmaceutical use |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| DK287085D0 DK287085D0 (da) | 1985-06-25 |
| DK287085A true DK287085A (da) | 1986-03-05 |
Family
ID=27089769
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK287085A DK287085A (da) | 1984-06-26 | 1985-06-25 | Triazolobenzodiazepin og farmaceutisk praeparat indeholdende en saadanforbindelse |
Country Status (4)
| Country | Link |
|---|---|
| US (1) | US4663321A (fr) |
| EP (1) | EP0169392A3 (fr) |
| DK (1) | DK287085A (fr) |
| ES (2) | ES8704946A1 (fr) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| YU136287A (en) * | 1986-07-25 | 1990-06-30 | Boehringer Kg | Process for preparing new 1,4 benzodiazepines |
| EP0272866A1 (fr) * | 1986-12-23 | 1988-06-29 | Merck & Co. Inc. | 1,4-Benzodiazépines avec hétérocycles à 5 chaînons |
| US4735941A (en) * | 1986-12-23 | 1988-04-05 | Merck & Co., Inc. | 1,4-benzodiazepines with 5- and 6-membered heterocyclic rings, useful as gastrointestinal and CNS agents |
| EP0272868A1 (fr) * | 1986-12-23 | 1988-06-29 | Merck & Co. Inc. | 1,4-Benzodiazépines avec hétérocycles à 6 chaînons |
| EP0273697A3 (fr) * | 1986-12-30 | 1989-11-29 | Merck & Co. Inc. | 2-Benzazépines à cycles hétérocycliques de 5 et 6 côtés |
| US5185331A (en) * | 1991-05-14 | 1993-02-09 | Merck & Co., Inc. | Triazolobenzodiazepines |
| CA2071092A1 (fr) * | 1991-06-14 | 1992-12-15 | Roger M. Freidinger | 1,4-benzodiazepines avec heterocycles a 5 chainons |
| EP0730596A4 (fr) * | 1993-11-22 | 1997-07-30 | Merck & Co Inc | Benzodiazepines |
| US5929071A (en) * | 1996-07-02 | 1999-07-27 | Merck & Co., Inc. | Method for the treatment of preterm labor |
| WO1998000406A1 (fr) * | 1996-07-02 | 1998-01-08 | Merck & Co., Inc. | Procede de traitement du travail preterme |
| US7119088B2 (en) * | 2003-02-19 | 2006-10-10 | Pfizer Inc. | Triazole compounds useful in therapy |
| WO2012075456A1 (fr) | 2010-12-02 | 2012-06-07 | Constellation Pharmaceuticals | Inhibiteurs de bromodomaines et leurs utilisations |
| AR084070A1 (es) | 2010-12-02 | 2013-04-17 | Constellation Pharmaceuticals Inc | Inhibidores del bromodominio y usos de los mismos |
| US9422292B2 (en) | 2011-05-04 | 2016-08-23 | Constellation Pharmaceuticals, Inc. | Bromodomain inhibitors and uses thereof |
| WO2012174487A2 (fr) | 2011-06-17 | 2012-12-20 | Constellation Pharmaceuticals, Inc. | Inhibiteurs à bromodomaine et leurs utilisations |
| TWI602820B (zh) | 2012-06-06 | 2017-10-21 | 星宿藥物公司 | 溴域抑制劑及其用途 |
| US9624244B2 (en) | 2012-06-06 | 2017-04-18 | Constellation Pharmaceuticals, Inc. | Benzo [B] isoxazoloazepine bromodomain inhibitors and uses thereof |
| PL3157928T3 (pl) | 2014-06-20 | 2019-07-31 | Constellation Pharmaceuticals, Inc. | Krystaliczne postacie 2-((4S)-6-(4-chlorofenylo)-1-metylo-4H-benzo[ c]izoksazolo-[4,5-e]azepin-4-ylo)acetamidu |
| US11040049B2 (en) | 2014-10-29 | 2021-06-22 | Glycom A/S | Composition comprising HMSs/HMOs and use thereof |
| US11040050B2 (en) | 2014-10-29 | 2021-06-22 | Glycom A/S | Composition comprising HMSs/HMOs and use thereof |
| US20160243139A1 (en) * | 2014-10-29 | 2016-08-25 | Glycom A/S | Composition comprising HMSs/HMOs and use thereof |
| EP3212197A4 (fr) | 2014-10-29 | 2018-07-11 | Glycom A/S | Composition synthétique et procédé de traitement de syndrome de l'intestin irritable |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3880877A (en) * | 1972-11-03 | 1975-04-29 | American Home Prod | Process for the preparation of 6-aryl-4H-s-triazolo(4,3-a)(1,4)benzodiazepines |
| JPS5747914B2 (fr) * | 1974-04-12 | 1982-10-13 | ||
| US3910944A (en) * | 1974-11-20 | 1975-10-07 | Upjohn Co | Spiro(cyclopropane-1,4{40 -(4H)-s-triazolo-(4,3-a)(1,4)benzodiazepines) |
| US4180668A (en) * | 1977-06-08 | 1979-12-25 | The Upjohn Company | Piperidino-4H-s-triazolo[4,3-a][1,4]benzodiazepines |
-
1985
- 1985-06-10 US US06/741,971 patent/US4663321A/en not_active Expired - Fee Related
- 1985-06-25 EP EP85107843A patent/EP0169392A3/fr not_active Withdrawn
- 1985-06-25 DK DK287085A patent/DK287085A/da not_active Application Discontinuation
- 1985-06-25 ES ES544521A patent/ES8704946A1/es not_active Expired
-
1986
- 1986-10-01 ES ES557126A patent/ES8707733A1/es not_active Expired
Also Published As
| Publication number | Publication date |
|---|---|
| ES8704946A1 (es) | 1987-04-16 |
| EP0169392A3 (fr) | 1986-11-05 |
| ES8707733A1 (es) | 1987-08-16 |
| US4663321A (en) | 1987-05-05 |
| DK287085D0 (da) | 1985-06-25 |
| EP0169392A2 (fr) | 1986-01-29 |
| ES557126A0 (es) | 1987-08-16 |
| ES544521A0 (es) | 1987-04-16 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| AHB | Application shelved due to non-payment |