DK297486A - Benzoxazinonderivater - Google Patents

Benzoxazinonderivater Download PDF

Info

Publication number: DK297486A
Authority: DK; Denmark
Prior art keywords: benzoxazinone derivatives; benzoxazinone; derivatives
Prior art date: 1985-06-25

Application number

DK297486A

Other languages

English (en)

Other versions

DK297486D0 (da

Inventor

Alexander Krantz

Robin W Spencer

Tim Tam

Teng J Liak

Original Assignee

Syntex Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1985-06-25

Filing date

1986-06-24

Publication date

1986-12-26

1986-06-24 Application filed by Syntex Inc filed Critical Syntex Inc

1986-06-24 Publication of DK297486D0 publication Critical patent/DK297486D0/da

1986-12-26 Publication of DK297486A publication Critical patent/DK297486A/da

Links

HQQTZCPKNZVLFF-UHFFFAOYSA-N 4h-1,2-benzoxazin-3-one Chemical class C1=CC=C2ONC(=O)CC2=C1 HQQTZCPKNZVLFF-UHFFFAOYSA-N 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
- C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
- C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D265/24—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in positions 2 and 4
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
- C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
- C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D265/24—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in positions 2 and 4
- C07D265/26—Two oxygen atoms, e.g. isatoic anhydride
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
- C07D265/04—1,3-Oxazines; Hydrogenated 1,3-oxazines
- C07D265/12—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems
- C07D265/14—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring
- C07D265/18—1,3-Oxazines; Hydrogenated 1,3-oxazines condensed with carbocyclic rings or ring systems condensed with one six-membered ring with hetero atoms directly attached in position 2
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6527—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having nitrogen and oxygen atoms as the only ring hetero atoms
- C07F9/6533—Six-membered rings
- C07F9/65335—Six-membered rings condensed with carbocyclic rings or carbocyclic ring systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Biochemistry (AREA)
Molecular Biology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)

DK297486A 1985-06-25 1986-06-24 Benzoxazinonderivater DK297486A (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US06/748,631 US4665070A (en)	1985-06-25	1985-06-25	2-oxy-4H-3,1-benzoxazin-4-ones and pharmaceutical use

Publications (2)

Publication Number	Publication Date
DK297486D0 DK297486D0 (da)	1986-06-24
DK297486A true DK297486A (da)	1986-12-26

Family

ID=25010264

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK297486A DK297486A (da)	1985-06-25	1986-06-24	Benzoxazinonderivater

Country Status (13)

Country	Link
US (1)	US4665070A (da)
EP (1)	EP0206323A1 (da)
JP (1)	JPS6230770A (da)
KR (1)	KR900004319B1 (da)
AU (2)	AU599320B2 (da)
CA (1)	CA1270487A (da)
DK (1)	DK297486A (da)
ES (4)	ES8802223A1 (da)
FI (1)	FI862691A7 (da)
HU (1)	HU196772B (da)
IL (1)	IL79222A0 (da)
NO (1)	NO163486C (da)
ZA (1)	ZA864715B (da)

Families Citing this family (15)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4745116A (en) *	1985-06-25	1988-05-17	Syntex (U.S.A.) Inc.	2-oxy-4H-3,1-benzoxazin-4-ones and related compounds and pharmaceutical use
CA1309556C (en) *	1987-06-09	1992-10-27	Masayuki Kokubo	4h-3,1-benzoxazin-4-one compounds and pharmaceutical composition thereoffor the inhibition of serine proteases
CA2056453A1 (en) *	1990-03-30	1991-10-01	Koji Kobayashi	4h-3, 1-benzoxazin-4-one derivative
US5985872A (en) *	1995-05-24	1999-11-16	G.D. Searle & Co.	2-amino-benzoxazinones for the treatment of viral infections
DE19708846A1 (de) *	1997-03-05	1998-09-17	Gruenenthal Gmbh	Neue Benzoxazindionderivate, Verfahren zu ihrer Herstellung und ihre Verwendung
FR2763944B1 (fr) *	1997-06-03	2000-12-15	Centre Nat Rech Scient	Nouveaux derives de coumarines, leurs procedes de preparation et leur application comme medicaments en tant qu'inhibiteurs de proteases
US6180625B1 (en)	1998-03-24	2001-01-30	Novo Nordisk A/S	Heterocyclic compounds regulating clotting
AU2826099A (en) *	1998-03-24	1999-10-18	Novo Nordisk A/S	Heterocyclic compounds regulating clotting
AU1375000A (en) *	1998-11-26	2000-06-13	Novo Nordisk A/S	Heterocyclic compounds regulating clotting
AR022204A1 (es) *	1999-01-08	2002-09-04	Norgine Bv	Compuesto, proceso para su preparacion, composicion farmaceutica y producto comestible que lo comprende.
GB9900416D0 (en)	1999-01-08	1999-02-24	Alizyme Therapeutics Ltd	Inhibitors
PE20010588A1 (es) *	1999-09-10	2001-06-23	Procter & Gamble	Conjugados polimericos inhibidores de enzimas proteoliticas y lipoliticas
EP1628674A2 (en) *	2003-05-06	2006-03-01	Cytovia, Inc.	Protease inhibitors for coronaviruses and sars-cov and the use thereof
ES2380135T3 (es) *	2006-11-22	2012-05-08	Ajinomoto Co., Inc.	MÃ©todo de preparaciÃ³n de derivados de fenilalanina que tienen esqueleto de quinazolinadiona e intermedios para su preparaciÃ³n
JP2010254623A (ja) *	2009-04-24	2010-11-11	Takeda Chem Ind Ltd	ベンゾオキサジノン化合物の結晶

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
HU173974B (hu) *	1971-08-30	1979-10-28	Chinoin Gyogyszer Es Vegyeszet	Sposob poluchenija proizvodnykh 3,1-benzoksazin-4-ona

1985
- 1985-06-25 US US06/748,631 patent/US4665070A/en not_active Expired - Fee Related
1986
- 1986-06-24 JP JP61149323A patent/JPS6230770A/ja active Pending
- 1986-06-24 KR KR1019860005053A patent/KR900004319B1/ko not_active Expired
- 1986-06-24 IL IL79222A patent/IL79222A0/xx unknown
- 1986-06-24 ZA ZA864715A patent/ZA864715B/xx unknown
- 1986-06-24 DK DK297486A patent/DK297486A/da not_active Application Discontinuation
- 1986-06-24 AU AU59150/86A patent/AU599320B2/en not_active Ceased
- 1986-06-24 ES ES556514A patent/ES8802223A1/es not_active Expired
- 1986-06-24 NO NO862534A patent/NO163486C/no unknown
- 1986-06-24 EP EP86108617A patent/EP0206323A1/en not_active Ceased
- 1986-06-24 CA CA000512310A patent/CA1270487A/en not_active Expired - Lifetime
- 1986-06-24 HU HU862647A patent/HU196772B/hu not_active IP Right Cessation
- 1986-06-24 FI FI862691A patent/FI862691A7/fi not_active Application Discontinuation
1987
- 1987-09-16 ES ES557732A patent/ES8801808A1/es not_active Expired
- 1987-09-16 ES ES557731A patent/ES8801807A1/es not_active Expired
- 1987-09-16 ES ES557730A patent/ES8801806A1/es not_active Expired
1990
- 1990-02-07 AU AU49120/90A patent/AU4912090A/en not_active Abandoned

Also Published As

Publication number	Publication date
ES8801806A1 (es)	1988-03-01
CA1270487A (en)	1990-06-19
ZA864715B (en)	1988-02-24
ES8801808A1 (es)	1988-03-01
US4665070A (en)	1987-05-12
HU196772B (en)	1989-01-30
JPS6230770A (ja)	1987-02-09
DK297486D0 (da)	1986-06-24
AU599320B2 (en)	1990-07-19
ES557731A0 (es)	1988-03-01
HUT41750A (en)	1987-05-28
ES557732A0 (es)	1988-03-01
EP0206323A1 (en)	1986-12-30
FI862691A0 (fi)	1986-06-24
ES8801807A1 (es)	1988-03-01
ES8802223A1 (es)	1988-05-01
ES557730A0 (es)	1988-03-01
IL79222A0 (en)	1986-09-30
FI862691L (fi)	1986-12-26
AU4912090A (en)	1990-05-31
NO163486C (no)	1990-06-13
KR870000310A (ko)	1987-02-17
NO163486B (no)	1990-02-26
NO862534D0 (no)	1986-06-24
AU5915086A (en)	1987-01-08
ES556514A0 (es)	1988-05-01
FI862691A7 (fi)	1986-12-26
KR900004319B1 (ko)	1990-06-22
NO862534L (no)	1986-12-29

Legal Events

Date	Code	Title	Description
1992-02-24	AHB	Application shelved due to non-payment

Publication	Publication Date	Title
DK263587D0 (da)	1987-05-22	Imidazoquinolinyletherderivater
DK82087D0 (da)	1987-02-18	Pyrocatecholderivater
ATE49403T1 (de)	1990-01-15	N-aralkylpiperidinmethanol-derivate.
ATA312487A (de)	1993-05-15	Tetrahydrocarbazolonderivate
DE3675232D1 (de)	1990-12-06	Pyridinderivate.
DE3678805D1 (de)	1991-05-23	Indolderivate.
DK297486A (da)	1986-12-26	Benzoxazinonderivater
DK693587D0 (da)	1987-12-30	Alkansulfonanilidderivater
BR8606663A (pt)	1987-08-11	Derivados de triazolil-quinolina
DK81888D0 (da)	1988-02-17	Dibenzoxepinderivater
DK109186D0 (da)	1986-03-10	Dihydropyridazinonderivater
ATE41655T1 (de)	1989-04-15	Phenaethanolaminderivate.
DE3680067D1 (de)	1991-08-08	Fluorphenylcyclohexanderivate.
DK491786D0 (da)	1986-10-14	Dichloranilinderivater
DK444687A (da)	1988-02-28	Alfa-substituerede ketonitron-derivater
DK556386A (da)	1987-06-21	Quinilinderivater
FI865230L (fi)	1987-06-21	Antikonvulsiva -tiobutyrolaktonderivat.
DK303886A (da)	1986-12-29	Secocanthinderivater
DK440687D0 (da)	1987-08-24	Bicyclooctanderivater
DK619187A (da)	1988-05-28	Isoindolderivater
DK229887D0 (da)	1987-05-05	Alkenamidderivater
DE3662889D1 (de)	1989-05-24	Tetrahydrofurancarboxylic-acid derivatives
KR880700821A (ko)	1988-04-12	데--데옥시테이코플라닌 유도체
DK435087D0 (da)	1987-08-20	Isoprenderivater
DK440787D0 (da)	1987-08-24	Bicyclooctanderivater