DK329185A - Fremgangsmaade til syntetisering af farmakologisk aktive forbindelser og mellemprodukter ved en saadan syntese - Google Patents

Fremgangsmaade til syntetisering af farmakologisk aktive forbindelser og mellemprodukter ved en saadan syntese Download PDF

Info

Publication number: DK329185A
Authority: DK; Denmark
Prior art keywords: compound; synthetization; intermediates; synthesis; procedure
Prior art date: 1984-08-13

Application number

DK329185A

Other languages

English (en)

Other versions

DK329185D0 (da

Inventor

Bo Robert Lamm

Original Assignee

Haessle Ab

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1984-08-13

Filing date

1985-07-19

Publication date

1986-02-14

1985-07-19 Application filed by Haessle Ab filed Critical Haessle Ab

1985-07-19 Publication of DK329185D0 publication Critical patent/DK329185D0/da

1986-02-14 Publication of DK329185A publication Critical patent/DK329185A/da

Links

150000001875 compounds Chemical class 0.000 title abstract 3
230000015572 biosynthetic process Effects 0.000 title abstract 2
238000000034 method Methods 0.000 title abstract 2
239000000543 intermediate Substances 0.000 title 1
230000000144 pharmacologic effect Effects 0.000 title 1
238000003786 synthesis reaction Methods 0.000 title 1
FBPFZTCFMRRESA-KVTDHHQDSA-N D-Mannitol Chemical compound OC[C@@H](O)[C@@H](O)[C@H](O)[C@H](O)CO FBPFZTCFMRRESA-KVTDHHQDSA-N 0.000 abstract 1
ZNZYKNKBJPZETN-WELNAUFTSA-N Dialdehyde 11678 Chemical compound N1C2=CC=CC=C2C2=C1[C@H](C[C@H](/C(=C/O)C(=O)OC)[C@@H](C=C)C=O)NCC2 ZNZYKNKBJPZETN-WELNAUFTSA-N 0.000 abstract 1
229930195725 Mannitol Natural products 0.000 abstract 1
DHKHKXVYLBGOIT-UHFFFAOYSA-N acetaldehyde Diethyl Acetal Natural products CCOC(C)OCC DHKHKXVYLBGOIT-UHFFFAOYSA-N 0.000 abstract 1
125000002777 acetyl group Chemical class [H]C([H])([H])C(*)=O 0.000 abstract 1
239000002253 acid Substances 0.000 abstract 1
125000000217 alkyl group Chemical group 0.000 abstract 1
238000005576 amination reaction Methods 0.000 abstract 1
125000006615 aromatic heterocyclic group Chemical group 0.000 abstract 1
125000002837 carbocyclic group Chemical group 0.000 abstract 1
125000004432 carbon atom Chemical group C* 0.000 abstract 1
230000007062 hydrolysis Effects 0.000 abstract 1
238000006460 hydrolysis reaction Methods 0.000 abstract 1
235000010355 mannitol Nutrition 0.000 abstract 1
239000000594 mannitol Substances 0.000 abstract 1
229910052757 nitrogen Inorganic materials 0.000 abstract 1
IJGRMHOSHXDMSA-UHFFFAOYSA-N nitrogen Substances N#N IJGRMHOSHXDMSA-UHFFFAOYSA-N 0.000 abstract 1
230000001590 oxidative effect Effects 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
125000000547 substituted alkyl group Chemical group 0.000 abstract 1
LMBFAGIMSUYTBN-MPZNNTNKSA-N teixobactin Chemical compound C([C@H](C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H](CCC(N)=O)C(=O)N[C@H]([C@@H](C)CC)C(=O)N[C@@H]([C@@H](C)CC)C(=O)N[C@@H](CO)C(=O)N[C@H]1C(N[C@@H](C)C(=O)N[C@@H](C[C@@H]2NC(=N)NC2)C(=O)N[C@H](C(=O)O[C@H]1C)[C@@H](C)CC)=O)NC)C1=CC=CC=C1 LMBFAGIMSUYTBN-MPZNNTNKSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
- C07D295/16—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms
- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D321/00—Heterocyclic compounds containing rings having two oxygen atoms as the only ring hetero atoms, not provided for by groups C07D317/00 - C07D319/00
- C07D321/02—Seven-membered rings
- C07D321/04—Seven-membered rings not condensed with other rings
- C07D321/06—1,3-Dioxepines; Hydrogenated 1,3-dioxepines
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)

DK329185A 1984-08-13 1985-07-19 Fremgangsmaade til syntetisering af farmakologisk aktive forbindelser og mellemprodukter ved en saadan syntese DK329185A (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
SE8404073A SE8404073D0 (sv)	1984-08-13	1984-08-13	Method for the synthesis of pharmacologically acitve compounds and intermediates for such synthesis

Publications (2)

Publication Number	Publication Date
DK329185D0 DK329185D0 (da)	1985-07-19
DK329185A true DK329185A (da)	1986-02-14

Family

ID=20356705

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK329185A DK329185A (da)	1984-08-13	1985-07-19	Fremgangsmaade til syntetisering af farmakologisk aktive forbindelser og mellemprodukter ved en saadan syntese

Country Status (9)

Country	Link
US (1)	US4777293A (da)
EP (1)	EP0179031B1 (da)
JP (1)	JPS6147447A (da)
AT (1)	ATE40108T1 (da)
DE (1)	DE3567641D1 (da)
DK (1)	DK329185A (da)
FI (1)	FI853089L (da)
NO (1)	NO853179L (da)
SE (1)	SE8404073D0 (da)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JP2801768B2 (ja) *	1990-11-17	1998-09-21	日東電工株式会社	新規な光学活性メトプロロール・酒石酸誘導体塩及びその製法、並びにこの塩を用いる光学活性メトプロロールの製法
WO1992016197A1 (en) *	1991-03-18	1992-10-01	Sepracor Inc.	Composition and method containing optically pure (s) metoprolol

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3729461A (en) *	1970-12-23	1973-04-24	Us Agriculture	Synthesis of glycosyl glycerides
CH635573A5 (en) *	1977-03-24	1983-04-15	Sandoz Ag	Process for preparing novel 1,2-dihydroxypropane derivatives
CA1074308A (en) *	1977-04-22	1980-03-25	Walter A. Szarek	L-sucrose and process for producing same

1984
- 1984-08-13 SE SE8404073A patent/SE8404073D0/xx unknown
1985
- 1985-07-10 US US06/753,682 patent/US4777293A/en not_active Expired - Fee Related
- 1985-07-19 DK DK329185A patent/DK329185A/da not_active Application Discontinuation
- 1985-08-08 DE DE8585850255T patent/DE3567641D1/de not_active Expired
- 1985-08-08 EP EP85850255A patent/EP0179031B1/en not_active Expired
- 1985-08-08 AT AT85850255T patent/ATE40108T1/de not_active IP Right Cessation
- 1985-08-12 JP JP60175983A patent/JPS6147447A/ja active Pending
- 1985-08-12 NO NO853179A patent/NO853179L/no unknown
- 1985-08-12 FI FI853089A patent/FI853089L/fi not_active Application Discontinuation

Also Published As

Publication number	Publication date
US4777293A (en)	1988-10-11
DK329185D0 (da)	1985-07-19
EP0179031A2 (en)	1986-04-23
NO853179L (no)	1986-02-14
ATE40108T1 (de)	1989-02-15
JPS6147447A (ja)	1986-03-07
EP0179031B1 (en)	1989-01-18
SE8404073D0 (sv)	1984-08-13
FI853089A7 (fi)	1986-02-14
DE3567641D1 (en)	1989-02-23
EP0179031A3 (en)	1986-08-13
FI853089L (fi)	1986-02-14
FI853089A0 (fi)	1985-08-12

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Legal Events

Date	Code	Title	Description
1991-03-25	AHB	Application shelved due to non-payment