DK3298008T3 - Krystallinsk form af forbindelsen (s)-3-{4-[5-(2-cyclopentyl-6-methoxy-pyridin-4-yl)-[1,2,4]oxadiazol-3-yl]-2-ethyl-6-methyl-phenoxy}-propan-1,2-diol - Google Patents

Krystallinsk form af forbindelsen (s)-3-{4-[5-(2-cyclopentyl-6-methoxy-pyridin-4-yl)-[1,2,4]oxadiazol-3-yl]-2-ethyl-6-methyl-phenoxy}-propan-1,2-diol Download PDF

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DK3298008T3
DK3298008T3 DK16724387.2T DK16724387T DK3298008T3 DK 3298008 T3 DK3298008 T3 DK 3298008T3 DK 16724387 T DK16724387 T DK 16724387T DK 3298008 T3 DK3298008 T3 DK 3298008T3
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oxadiazol
pyridin
cyclopentyl
phenoxy
diol
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DK16724387.2T
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Cyrille Lescop
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Idorsia Pharmaceuticals Ltd
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/045—Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates
    • A61K31/047—Hydroxy compounds, e.g. alcohols; Salts thereof, e.g. alcoholates having two or more hydroxy groups, e.g. sorbitol
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4245—Oxadiazoles
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    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
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    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
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    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
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    • C07B2200/13—Crystalline forms, e.g. polymorphs
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DK16724387.2T 2015-05-20 2016-05-19 Krystallinsk form af forbindelsen (s)-3-{4-[5-(2-cyclopentyl-6-methoxy-pyridin-4-yl)-[1,2,4]oxadiazol-3-yl]-2-ethyl-6-methyl-phenoxy}-propan-1,2-diol DK3298008T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP2015061153 2015-05-20
PCT/EP2016/061200 WO2016184939A1 (en) 2015-05-20 2016-05-19 Crystalline form of the compound (s)-3-{4-[5-(2-cyclopentyl-6-methoxy-pyridin-4-yl)-[1,2,4]oxadiazol-3-yl]-2-ethyl-6-methyl-phenoxy}-propane-1,2-diol

Publications (1)

Publication Number Publication Date
DK3298008T3 true DK3298008T3 (da) 2020-02-10

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DK16724387.2T DK3298008T3 (da) 2015-05-20 2016-05-19 Krystallinsk form af forbindelsen (s)-3-{4-[5-(2-cyclopentyl-6-methoxy-pyridin-4-yl)-[1,2,4]oxadiazol-3-yl]-2-ethyl-6-methyl-phenoxy}-propan-1,2-diol

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US (4) US10385043B2 (da)
EP (1) EP3298008B1 (da)
JP (1) JP6674967B2 (da)
KR (2) KR102220848B1 (da)
CN (2) CN107667104B (da)
AU (1) AU2016263472B2 (da)
BR (1) BR112017024785B1 (da)
CA (1) CA2981130C (da)
CL (1) CL2017002822A1 (da)
CY (1) CY1122506T1 (da)
DK (1) DK3298008T3 (da)
EA (1) EA035133B1 (da)
ES (1) ES2770348T3 (da)
HR (1) HRP20200001T1 (da)
HU (1) HUE047646T2 (da)
IL (1) IL255718B (da)
LT (1) LT3298008T (da)
MA (1) MA42107B1 (da)
MX (1) MX373293B (da)
MY (1) MY192358A (da)
PH (1) PH12017502097B1 (da)
PL (1) PL3298008T3 (da)
PT (1) PT3298008T (da)
RS (1) RS59788B1 (da)
SG (1) SG11201708794PA (da)
SI (1) SI3298008T1 (da)
TW (1) TWI711609B (da)
UA (1) UA119818C2 (da)
WO (1) WO2016184939A1 (da)

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JP7749552B2 (ja) 2019-10-31 2025-10-06 イドルシア・ファーマシューティカルズ・リミテッド Ｃｘｃｒ７アンタゴニストのｓ１ｐ１受容体調節剤との合剤
WO2021148314A1 (en) 2020-01-20 2021-07-29 Idorsia Pharmaceuticals Ltd Accelerated elimination of (s)-3-{4-[5-(2-cyclopentyl-6-methoxy-pyridin-4-yl)-[1,2,4]oxadiazol-3-yl]-2-ethyl-6-methyl-phenoxy}-propane-1,2-diol
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