DK361989A - N15-alkyl og n15,n15,-dialkylderivater af teicoplanin-antibiotika med funktionelle grupper paa alkyl-sidekaeden - Google Patents

N15-alkyl og n15,n15,-dialkylderivater af teicoplanin-antibiotika med funktionelle grupper paa alkyl-sidekaeden Download PDF

Info

Publication number: DK361989A
Authority: DK; Denmark
Prior art keywords: alkyl; teicoplanine; antibiotics; functional groups; side chain
Prior art date: 1988-07-21

Application number

DK361989A

Other languages

English (en)

Other versions

DK361989D0 (da

Inventor

Adriano Malabarba

Aldo Trani

Original Assignee

Lepetit Spa

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1988-07-21

Filing date

1989-07-21

Publication date

1990-01-22

1989-07-21 Application filed by Lepetit Spa filed Critical Lepetit Spa

1989-07-21 Publication of DK361989D0 publication Critical patent/DK361989D0/da

1990-01-22 Publication of DK361989A publication Critical patent/DK361989A/da

Links

BJNLLBUOHPVGFT-CAYRISATSA-N (1S,2R,19R,22R,34S,37R,40R,52S)-2-[(2R,3R,4R,5S,6R)-3-acetamido-4,5-dihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-22-amino-5,15-dichloro-64-[(2S,3R,4R,5S,6R)-3-(decanoylamino)-4,5-dihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-26,31,44,49-tetrahydroxy-21,35,38,54,56,59-hexaoxo-47-[(3S,4S,5S,6R)-3,4,5-trihydroxy-6-(hydroxymethyl)oxan-2-yl]oxy-7,13,28-trioxa-20,36,39,53,55,58-hexazaundecacyclo[38.14.2.23,6.214,17.219,34.18,12.123,27.129,33.141,45.010,37.046,51]hexahexaconta-3,5,8,10,12(64),14,16,23(61),24,26,29(60),30,32,41(57),42,44,46(51),47,49,62,65-henicosaene-52-carboxylic acid Chemical class CCCCCCCCCC(=O)N[C@@H]1[C@@H](O)[C@H](O)[C@@H](CO)O[C@H]1Oc1c2Oc3ccc(C[C@H]4NC(=O)[C@H](N)c5ccc(O)c(Oc6cc(O)cc(c6)[C@H](NC4=O)C(=O)N[C@@H]4c(c2)cc1Oc1ccc(cc1Cl)[C@@H](O[C@@H]1O[C@H](CO)[C@@H](O)[C@H](O)[C@H]1NC(C)=O)[C@@H]1NC(=O)[C@H](NC4=O)c2ccc(O)c(c2)-c2c(OC4O[C@H](CO)[C@@H](O)[C@H](O)[C@@H]4O)cc(O)cc2[C@H](NC1=O)C(O)=O)c5)cc3Cl BJNLLBUOHPVGFT-CAYRISATSA-N 0.000 title 1
239000003242 anti bacterial agent Substances 0.000 title 1
229940088710 antibiotic agent Drugs 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K9/00—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof
- C07K9/006—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure
- C07K9/008—Peptides having up to 20 amino acids, containing saccharide radicals and having a fully defined sequence; Derivatives thereof the peptide sequence being part of a ring structure directly attached to a hetero atom of the saccharide radical, e.g. actaplanin, avoparcin, ristomycin, vancomycin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents

Landscapes

Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Biochemistry (AREA)
Oncology (AREA)
Pharmacology & Pharmacy (AREA)
General Chemical & Material Sciences (AREA)
Animal Behavior & Ethology (AREA)
Communicable Diseases (AREA)
Public Health (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Biophysics (AREA)
Genetics & Genomics (AREA)
Molecular Biology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Fodder In General (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Peptides Or Proteins (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

DK361989A 1988-07-21 1989-07-21 N15-alkyl og n15,n15,-dialkylderivater af teicoplanin-antibiotika med funktionelle grupper paa alkyl-sidekaeden DK361989A (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB888817397A GB8817397D0 (en)	1988-07-21	1988-07-21	N15-alkyl & n15 n15-di-alkyl derivatives of teicoplanin antibiotics carrying functional groups on alkyl side chain

Publications (2)

Publication Number	Publication Date
DK361989D0 DK361989D0 (da)	1989-07-21
DK361989A true DK361989A (da)	1990-01-22

Family

ID=10640877

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK361989A DK361989A (da)	1988-07-21	1989-07-21	N15-alkyl og n15,n15,-dialkylderivater af teicoplanin-antibiotika med funktionelle grupper paa alkyl-sidekaeden

Country Status (4)

Country	Link
EP (1)	EP0351597A3 (da)
JP (1)	JPH0269500A (da)
DK (1)	DK361989A (da)
GB (1)	GB8817397D0 (da)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
WO1992010516A1 (en) *	1990-12-05	1992-06-25	Gruppo Lepetit S.P.A.	38-decarboxy-38-hydroxymethyl derivatives of teicoplanin antibiotics, and a process for preparing them
PT836619E (pt) *	1995-07-05	2004-11-30	Aventis Bulk S P A	Purificacao de antibioticos dalba-heptidicos por focagem isoelectrica
EP0912604B1 (en)	1996-04-23	2001-11-14	Biosearch Italia S.p.A.	Improved chemical process for preparing amide derivatives of antibiotic A 40926
US5936074A (en) *	1997-04-17	1999-08-10	Eli Lilly And Company	Teicoplanin deacylation process and product
PT1140993E (pt)	1998-12-23	2003-10-31	Theravance Inc	Derivados de glicopeptidos e composicoes farmaceuticas contendo os mesmos
SG87877A1 (en) *	1998-12-23	2002-04-16	Advanced Medicine Inc	Glycopeptide derivatives and pharmaceutical compositions containing the same

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8522574D0 (en) *	1985-09-12	1985-10-16	Lepetit Spa	Amides of teicoplanin compounds

1988
- 1988-07-21 GB GB888817397A patent/GB8817397D0/en active Pending
1989
- 1989-06-28 EP EP19890111730 patent/EP0351597A3/en not_active Ceased
- 1989-07-19 JP JP1184850A patent/JPH0269500A/ja active Pending
- 1989-07-21 DK DK361989A patent/DK361989A/da not_active Application Discontinuation

Also Published As

Publication number	Publication date
DK361989D0 (da)	1989-07-21
EP0351597A2 (en)	1990-01-24
GB8817397D0 (en)	1988-08-24
JPH0269500A (ja)	1990-03-08
EP0351597A3 (en)	1991-06-19

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Legal Events

Date	Code	Title	Description
1994-03-28	AHB	Application shelved due to non-payment