DK377882A - METHOD FOR PREPARING (3H) -IMIDAZO- (5,1-D) -1,2,3,5-TETRAZIN-4-ON DERIVATIVES - Google Patents

METHOD FOR PREPARING (3H) -IMIDAZO- (5,1-D) -1,2,3,5-TETRAZIN-4-ON DERIVATIVES Download PDF

Info

Publication number: DK377882A
Authority: DK; Denmark
Prior art keywords: tetrazin; imidazo; derivatives; preparing
Prior art date: 1981-08-24

Application number

DK377882A

Other languages

Danish (da)

Other versions

DK161147B (en

DK161147C (en

Inventor

Edward Lunt

Malcolm Francis Graham Stevens

Robert Stone

Kenneth Robert Harr Wooldridge

Original Assignee

May & Baker Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1981-08-24

Filing date

1982-08-23

Publication date

1983-02-25

1982-08-23 Application filed by May & Baker Ltd filed Critical May & Baker Ltd

1983-02-25 Publication of DK377882A publication Critical patent/DK377882A/en

1991-06-03 Publication of DK161147B publication Critical patent/DK161147B/en

1991-11-18 Application granted granted Critical

1991-11-18 Publication of DK161147C publication Critical patent/DK161147C/en

Links

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
- C07D407/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Hematology (AREA)
Oncology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

DK377882A 1981-08-24 1982-08-23 METHOD OF ANALOGY FOR THE PREPARATION OF OE3HAA-IMIDAZO-OE5,1-DAA-1,2,3,5-TETRAZIN-4-UNDIVERIVES DK161147C (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
GB8125791		1981-08-24
GB8125791		1981-08-24

Publications (3)

Publication Number	Publication Date
DK377882A true DK377882A (en)	1983-02-25
DK161147B DK161147B (en)	1991-06-03
DK161147C DK161147C (en)	1991-11-18

Family

ID=10524141

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK377882A DK161147C (en)	1981-08-24	1982-08-23	METHOD OF ANALOGY FOR THE PREPARATION OF OE3HAA-IMIDAZO-OE5,1-DAA-1,2,3,5-TETRAZIN-4-UNDIVERIVES

Country Status (29)

Country	Link
JP (1)	JPS5843975A (en)
KR (1)	KR890000094B1 (en)
AT (1)	AT380256B (en)
AU (1)	AU571430B2 (en)
BE (1)	BE894175A (en)
CA (1)	CA1197247A (en)
CH (1)	CH655114A5 (en)
DE (2)	DE19975037I2 (en)
DK (1)	DK161147C (en)
ES (1)	ES8400438A1 (en)
FI (1)	FI73434C (en)
FR (1)	FR2511679A1 (en)
GB (1)	GB2104522B (en)
GE (1)	GEP19960641B (en)
GR (1)	GR76863B (en)
HU (1)	HU186107B (en)
IE (1)	IE53408B1 (en)
IL (1)	IL66606A (en)
IT (1)	IT1152505B (en)
LT (1)	LT2436B (en)
LU (1)	LU84347A1 (en)
LV (2)	LV5511A3 (en)
NL (2)	NL192739C (en)
NZ (1)	NZ201668A (en)
OA (1)	OA07174A (en)
SE (1)	SE448543B (en)
SU (1)	SU1447284A3 (en)
UA (1)	UA5971A1 (en)
ZA (1)	ZA826120B (en)

Families Citing this family (22)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5260291A (en) *	1981-08-24	1993-11-09	Cancer Research Campaign Technology Limited	Tetrazine derivatives
GB2125402B (en) *	1982-08-17	1985-11-13	May & Baker Ltd	New tetrazine derivatives
FR2531958B1 (en) *	1982-08-17	1986-10-31	May & Baker Ltd	NEW DERIVATIVES
US4517182A (en) *	1983-05-24	1985-05-14	Warner-Lambert Company	3-(Haloethyl)-4-oxopyrazolo-[5,1-d]-1,2,3,5-tetrazine-8-carboxamide composition
GB8616125D0 (en) *	1986-07-02	1986-08-06	May & Baker Ltd	Compositions of matter
AU622330B2 (en) *	1989-06-23	1992-04-02	Takeda Chemical Industries Ltd.	Condensed heterocyclic compounds having a nitrogen atom in the bridgehead for use as fungicides
DE69636837T2 (en) *	1995-09-25	2007-10-25	Sanofi-Aventis U.S. Llc	1,2,4-benzotriazine FORMULATIONS
EP2275425A1 (en) *	2003-12-30	2011-01-19	Chemagis Ltd.	Novel crystalline forms of temozolomide
MX2007008781A (en)	2005-01-21	2007-09-11	Astex Therapeutics Ltd	Pharmaceutical compounds.
AR060635A1 (en)	2006-04-27	2008-07-02	Banyu Pharma Co Ltd	DERIVATIVES OF 1,2-DIHIDRO-3H-PIRAZOLO [3,4-D] PIRIMIDIN-3-ONA, PHARMACEUTICAL COMPOSITIONS THAT INCLUDE THEM AND THEIR USE IN THE TREATMENT OF CANCER
JP2008081492A (en)	2006-08-31	2008-04-10	Banyu Pharmaceut Co Ltd	Novel aminopyridine derivatives having selective inhibition of Aurora A
JP5528807B2 (en)	2006-10-12	2014-06-25	アステックス、セラピューティックス、リミテッド	Compound drug
WO2008044041A1 (en)	2006-10-12	2008-04-17	Astex Therapeutics Limited	Pharmaceutical combinations
EP2213673B1 (en)	2007-10-23	2013-06-05	Msd K.K.	Pyridone-substituted-dihydropyrazolopyrimidinone derivative
PE20091101A1 (en) *	2007-12-18	2009-07-26	Pharminox Ltd	3-SUBSTITUTED-4-OXO-3,4-DIHYDRO-IMIDAZO [5,1-d] [1,2,3,5-TETRACINE-8-CARBOXYL ACID AMIDES AND ITS USE
KR20110111383A (en) *	2008-11-24	2011-10-11	리라이언스 라이프 사이언시스 프라이빗. 리미티드	Method for preparing tetrazine derivative
WO2010101734A1 (en)	2009-03-06	2010-09-10	Merck Sharp & Dohme Corp.	Combination cancer therapy with an akt inhibitor and other anticancer agents
CA2763766A1 (en)	2009-06-23	2010-12-29	Pharminox Limited	3-substituted-8-substituted-3h-imidazo[5,1-d][1,2,3,5-tetrazin-4-one compounds and their use
RU2462466C1 (en) *	2011-06-24	2012-09-27	Автономная Некоммерческая Организация "Научно-Исследовательский Центр Биотехнологии Антибиотиков И Других Биологически Активных Веществ "Биоан"	Substituted azolo[1,2,4,5]tetrazines - inhibitors of antibacterial serine-threonine protein kinases
EP2766041B1 (en)	2011-10-12	2018-12-05	Children's Medical Center Corporation	Combinatorial compositions and methods of treating hemoglobinopathies
ES3057783T3 (en)	2016-03-15	2026-03-04	Oryzon Genomics Sa	Combinations of lsd1 inhibitors for use in the treatment of neoplastic diseases
KR101847342B1 (en) *	2017-05-08	2018-04-11	(주)센텍코리아	Wearable body fat burning measurement device

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE2932305A1 (en) *	1979-08-09	1981-02-26	Basf Ag	Pyrrolo-, pyrazolo-, imidazo- and thiazolo-tetrazin-4-one derivs. - prepd. from amino-azole cpds. by diazotisation and reaction with isocyanate

1982
- 1982-08-05 OA OA57766BISD patent/OA07174A/en unknown
- 1982-08-12 IL IL66606A patent/IL66606A/en not_active IP Right Cessation
- 1982-08-23 NZ NZ201668A patent/NZ201668A/en unknown
- 1982-08-23 IE IE2026/82A patent/IE53408B1/en not_active IP Right Cessation
- 1982-08-23 NL NL8203286A patent/NL192739C/en not_active IP Right Cessation
- 1982-08-23 LU LU84347A patent/LU84347A1/en unknown
- 1982-08-23 ES ES515176A patent/ES8400438A1/en not_active Expired
- 1982-08-23 CA CA000409950A patent/CA1197247A/en not_active Expired
- 1982-08-23 AT AT0319182A patent/AT380256B/en not_active IP Right Cessation
- 1982-08-23 GR GR69093A patent/GR76863B/el unknown
- 1982-08-23 ZA ZA826120A patent/ZA826120B/en unknown
- 1982-08-23 SU SU823482389A patent/SU1447284A3/en active
- 1982-08-23 GB GB08224155A patent/GB2104522B/en not_active Expired
- 1982-08-23 SE SE8204817A patent/SE448543B/en not_active IP Right Cessation
- 1982-08-23 BE BE0/208860A patent/BE894175A/en not_active IP Right Cessation
- 1982-08-23 DK DK377882A patent/DK161147C/en not_active IP Right Cessation
- 1982-08-23 HU HU822708A patent/HU186107B/en unknown
- 1982-08-23 IT IT22938/82A patent/IT1152505B/en active Protection Beyond IP Right Term
- 1982-08-23 UA UA3482389A patent/UA5971A1/en unknown
- 1982-08-23 FI FI822921A patent/FI73434C/en not_active IP Right Cessation
- 1982-08-23 FR FR8214461A patent/FR2511679A1/en active Granted
- 1982-08-23 JP JP57144902A patent/JPS5843975A/en active Granted
- 1982-08-23 CH CH5007/82A patent/CH655114A5/en not_active IP Right Cessation
- 1982-08-23 DE DE1999175037 patent/DE19975037I2/en active Active
- 1982-08-23 KR KR8203774A patent/KR890000094B1/en not_active Expired
- 1982-08-23 AU AU87493/82A patent/AU571430B2/en not_active Expired
- 1982-08-23 DE DE19823231255 patent/DE3231255A1/en active Granted
1993
- 1993-06-19 LV LV930621A patent/LV5511A3/en unknown
- 1993-09-29 LT LTRP1286A patent/LT2436B/en not_active IP Right Cessation
- 1993-11-16 GE GEAP19931653A patent/GEP19960641B/en unknown
- 1993-12-03 LV LV931303A patent/LV5621A3/en unknown
1999
- 1999-04-01 NL NL990010C patent/NL990010I2/en unknown

Also Published As

Publication number	Publication date
KR840001175A (en)	1984-03-28
FI73434C (en)	1987-10-09
IL66606A0 (en)	1982-12-31
NZ201668A (en)	1985-08-16
SE8204817L (en)	1983-02-25
IL66606A (en)	1987-07-31
JPH045029B2 (en)	1992-01-30
GEP19960641B (en)	1996-11-15
DK161147B (en)	1991-06-03
NL192739B (en)	1997-09-01
ES515176A0 (en)	1983-11-01
GB2104522B (en)	1985-06-12
IT8222938A0 (en)	1982-08-23
SU1447284A3 (en)	1988-12-23
IE53408B1 (en)	1988-11-09
DE3231255A1 (en)	1983-03-03
FI822921L (en)	1983-02-25
FI822921A0 (en)	1982-08-23
AT380256B (en)	1986-05-12
FI73434B (en)	1987-06-30
KR890000094B1 (en)	1989-03-07
NL192739C (en)	1998-01-06
BE894175A (en)	1983-02-23
OA07174A (en)	1984-04-30
NL8203286A (en)	1983-03-16
CH655114A5 (en)	1986-03-27
DK161147C (en)	1991-11-18
ATA319182A (en)	1985-09-15
GR76863B (en)	1984-09-04
HU186107B (en)	1985-06-28
DE19975037I2 (en)	2001-06-13
SE8204817D0 (en)	1982-08-23
FR2511679B1 (en)	1985-02-01
UA5971A1 (en)	1994-12-29
DE3231255C2 (en)	1992-02-27
IE822026L (en)	1983-02-24
LV5621A3 (en)	1994-05-10
JPS5843975A (en)	1983-03-14
AU8749382A (en)	1983-03-03
FR2511679A1 (en)	1983-02-25
NL990010I2 (en)	1999-09-01
LV5511A3 (en)	1994-03-10
AU571430B2 (en)	1988-04-21
NL990010I1 (en)	1999-07-01
CA1197247A (en)	1985-11-26
LU84347A1 (en)	1983-06-07
GB2104522A (en)	1983-03-09
ES8400438A1 (en)	1983-11-01
LT2436B (en)	1994-02-15
IT1152505B (en)	1987-01-07
SE448543B (en)	1987-03-02
IT8222938A1 (en)	1984-02-23
ZA826120B (en)	1983-07-27

Legal Events

Date	Code	Title	Description
1999-08-16	CTFF	Application for supplementary protection certificate (spc) filed	Free format text: CA 1999 00012, 19990511, EXPIRES: 20070823
2002-09-09	PUP	Patent expired

Publication	Publication Date	Title
DK377882A (en)	1983-02-25	METHOD FOR PREPARING (3H) -IMIDAZO- (5,1-D) -1,2,3,5-TETRAZIN-4-ON DERIVATIVES
DK280182A (en)	1982-12-24	METHOD FOR PREPARING N-ARYL-PIPERAZINAL CANAMIDES
DK159442C (en)	1991-03-18	ANALOGY PROCEDURE FOR PREPARING 6,7-SUBSTITUTED-4-ETHYL-QUINAZOLINES
DK470583D0 (en)	1983-10-12	METHOD FOR PREPARING 1-PHENYL-2-PIPERIDINOPROPANOL DERIVATIVES
DK492783D0 (en)	1983-10-27	METHOD FOR PREPARING 3-ARYL-5-PYRAZOLE DERIVATIVES
DK95483D0 (en)	1983-02-25	METHOD FOR PREPARING TETRA-HYDROPYRANE DERIVATIVES
DK143491D0 (en)	1991-08-06	METHOD FOR PREPARING 3-OEN-PHENYLACETYLAMINOPIPERIDINAA-2,6-DION
DK262782A (en)	1982-12-13	METHOD FOR PREPARING N-DIHYDROTHIAZOLYL-3-QUINOLINCARBOXAMIDE DERIVATIVES
DK379985A (en)	1986-03-06	METHOD FOR PREPARING 6-CHLOR-N-METHYL-2,3,4,5-TETRAHYDRO-LH-BENZAZEPINE
DK155281C (en)	1989-07-24	METHOD FOR PREPARING 1,2-DIHYDRO-6-METHYL-2-OXO-5- (PYRIDINYL) NICOTINON NITRILS
DK157855C (en)	1990-07-30	METHOD FOR PREPARING 2,3-DICHLOR-5-TRICHLORMETHYLPYRIDINE
ES517022A0 (en)	1984-08-16	PROCEDURE FOR PREPARING 1,4-DIHYDROPYRIDINE COMPOUNDS.
DK156722C (en)	1990-02-19	ANALOGY PROCEDURE FOR PREPARING 2-PIPERAZINOPYRIMIDINE DERIVATIVES
DK40482A (en)	1982-07-31	METHOD FOR PREPARING 2- (2- (1,4-BENZODIOXANYL)) - 2-IMIDAZOLINE DERIVATIVES
DK370582A (en)	1983-02-20	METHOD FOR PREPARING 2-BETA-D-RIBOFURANOSYLTHIAZOL-4-CARBOXAMIDE
DK113483A (en)	1983-03-08	METHOD FOR PREPARING 3,4-DIPHENYL-5-METHYLPYRAZOLE DERIVATIVES
DK158227C (en)	1990-09-17	METHOD OF ANALOGUE FOR THE PREPARATION OF SUBSTITUTED IMIDAZOOE1,5-AAAPYRIDINES OR 5,6,7,8-TETRAHYDRODE DERIVATIVES OR SALTS THEREOF
DK154207C (en)	1989-03-13	METHOD FOR PREPARING 1,8-DIHYDROXY-10-ACYL-9 ANTHRONS
DK153488C (en)	1988-12-19	PROCEDURE FOR PREPARING 5,6,7,7A-TETRAHYDRO-4H-THIENO (3,2-C -) - PYRIDIN-2 UNDERIVATIVES
FI821514A7 (en)	1982-11-02	Method for preparing overvoltage-resistant chromone derivatives.
DK97682A (en)	1982-09-07	METHOD FOR PREPARING 1- (1,3-BENZODIOXOL-5-YL) -2-PYRROLIDINON
DK79982A (en)	1982-08-26	METHOD FOR PREPARING 3- (4-PHENYL-1-PIPERAZINIO-1-YL) -1,2-PROPANDIOL-3- (THEOPHYLLIN-7-YL) -1-PROPAN SULPHONATE
FI822647A7 (en)	1983-01-30	Method for preparing 4-amino-butyramide.
DK513580A (en)	1981-07-08	METHOD FOR PREPARING 4,5-DIARYL-ALFA (POLYHALOGENALKYL) -1H-IMIDAZOL-2-METHANOLS
DK454183A (en)	1984-04-02	METHOD FOR PREPARING 15-CYCLOALIPHATIC DERIVATIVES OF 13,14-DIDEHYDRO-CARBOPROSTANCYCLINES