DK41180A - Fremgangsmaade til fremstilling af krystallinske 3-hydroxycephalosporin-solvater - Google Patents

Fremgangsmaade til fremstilling af krystallinske 3-hydroxycephalosporin-solvater

Info

Publication number: DK41180A
Authority: DK; Denmark
Prior art keywords: hydroxycephalosporine; crystallinic; solvates; procedure; preparation
Prior art date: 1979-02-01

Application number

DK41180A

Other languages

English (en)

Other versions

DK159157C (da

DK159157B (da

Inventor

J W Fisher

Original Assignee

Lilly Co Eli

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1979-02-01

Filing date

1980-01-31

Publication date

1980-08-02

1980-01-31 Application filed by Lilly Co Eli filed Critical Lilly Co Eli

1980-08-02 Publication of DK41180A publication Critical patent/DK41180A/da

1990-09-10 Publication of DK159157B publication Critical patent/DK159157B/da

1991-02-11 Application granted granted Critical

1991-02-11 Publication of DK159157C publication Critical patent/DK159157C/da

Links

239000012453 solvate Substances 0.000 title 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/26—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group
- C07D501/32—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group with the 7-amino radical acylated by an araliphatic carboxylic acid, which is substituted on the aliphatic radical by hetero atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/59—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3 with hetero atoms directly attached in position 3
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D501/00—Heterocyclic compounds containing 5-thia-1-azabicyclo [4.2.0] octane ring systems, i.e. compounds containing a ring system of the formula:, e.g. cephalosporins; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D501/14—Compounds having a nitrogen atom directly attached in position 7
- C07D501/16—Compounds having a nitrogen atom directly attached in position 7 with a double bond between positions 2 and 3
- C07D501/20—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids
- C07D501/24—7-Acylaminocephalosporanic or substituted 7-acylaminocephalosporanic acids in which the acyl radicals are derived from carboxylic acids with hydrocarbon radicals, substituted by hetero atoms or hetero rings, attached in position 3
- C07D501/26—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group
- C07D501/30—Methylene radicals, substituted by oxygen atoms; Lactones thereof with the 2-carboxyl group with the 7-amino-radical acylated by an araliphatic carboxylic acid

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Communicable Diseases (AREA)
Pharmacology & Pharmacy (AREA)
Oncology (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Cephalosporin Compounds (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DK041180A 1979-02-01 1980-01-31 Krystallinske 3-hydroxy-cephalosporin-solvater DK159157C (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US846879A	1979-02-01	1979-02-01
US846879		1979-02-01

Publications (3)

Publication Number	Publication Date
DK41180A true DK41180A (da)	1980-08-02
DK159157B DK159157B (da)	1990-09-10
DK159157C DK159157C (da)	1991-02-11

Family

ID=21731772

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK041180A DK159157C (da)	1979-02-01	1980-01-31	Krystallinske 3-hydroxy-cephalosporin-solvater

Country Status (32)

Country	Link
EP (1)	EP0014565B1 (da)
JP (1)	JPS55104288A (da)
KR (1)	KR830001890B1 (da)
AR (1)	AR228342A1 (da)
AT (1)	AT366052B (da)
AU (1)	AU532573B2 (da)
BE (1)	BE881423A (da)
BG (1)	BG32857A3 (da)
CA (1)	CA1142173A (da)
CH (1)	CH647525A5 (da)
CS (1)	CS214694B2 (da)
DD (1)	DD148953A5 (da)
DE (1)	DE3062095D1 (da)
DK (1)	DK159157C (da)
ES (1)	ES488229A0 (da)
FI (1)	FI68239C (da)
FR (1)	FR2447925A1 (da)
GB (1)	GB2041934B (da)
GR (1)	GR72785B (da)
HU (2)	HU181761B (da)
IE (1)	IE49374B1 (da)
IL (1)	IL59265A (da)
IT (1)	IT1130239B (da)
LU (1)	LU82118A1 (da)
NZ (1)	NZ192750A (da)
PH (1)	PH15152A (da)
PL (1)	PL122609B1 (da)
PT (1)	PT70742A (da)
RO (2)	RO79181A (da)
SU (2)	SU897109A3 (da)
YU (1)	YU22480A (da)
ZA (1)	ZA80523B (da)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
DE3128949A1 (de) *	1981-07-22	1983-02-10	Basf Ag, 6700 Ludwigshafen	Lichtempfindliche aufzeichnungsmaterialien zur herstellung von abriebs- und kratzfesten tiefdruckformen sowie verfahren zur herstellung von tiefdruckformen mittels dieser aufzeichnungsmaterialien
JPS6011491A (ja) *	1983-03-04	1985-01-21	Shionogi & Co Ltd	セフアロチンナトリウムの結晶性凍結乾燥粉末の製造法
US4782144A (en) *	1987-09-14	1988-11-01	Eli Lilly And Company	1-carba(dethia)-3-hydroxy-3-cephem ester crystalline and crystalline solvate thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3985747A (en) *	1974-05-24	1976-10-12	Bristol-Myers Company	Crystalline sesquihydrate of 7-[D-α-amino-α-(p-hydroxyphenyl)acetamido]-3-(1,2,3-triazol-5-ylthiomethyl)-3-cephem-4-carboxylic acid
US4044002A (en) *	1976-06-09	1977-08-23	Eli Lilly And Company	Reduction process for cephalosporin sulfoxides

1980
- 1980-01-03 IE IE191/80A patent/IE49374B1/en not_active IP Right Cessation
- 1980-01-29 GR GR61064A patent/GR72785B/el unknown
- 1980-01-29 IL IL59265A patent/IL59265A/xx unknown
- 1980-01-29 NZ NZ192750A patent/NZ192750A/xx unknown
- 1980-01-29 PT PT70742A patent/PT70742A/pt active IP Right Revival
- 1980-01-29 HU HU80189A patent/HU181761B/hu unknown
- 1980-01-29 AU AU55026/80A patent/AU532573B2/en not_active Expired
- 1980-01-29 YU YU00224/80A patent/YU22480A/xx unknown
- 1980-01-29 ZA ZA00800523A patent/ZA80523B/xx unknown
- 1980-01-29 HU HU80192A patent/HU182095B/hu unknown
- 1980-01-30 FR FR8001966A patent/FR2447925A1/fr active Granted
- 1980-01-30 BE BE1/9699A patent/BE881423A/fr not_active IP Right Cessation
- 1980-01-30 BG BG046408A patent/BG32857A3/xx unknown
- 1980-01-30 CA CA000344677A patent/CA1142173A/en not_active Expired
- 1980-01-31 CH CH795/80A patent/CH647525A5/fr not_active IP Right Cessation
- 1980-01-31 LU LU82118A patent/LU82118A1/fr unknown
- 1980-01-31 AT AT0049980A patent/AT366052B/de not_active IP Right Cessation
- 1980-01-31 EP EP80300281A patent/EP0014565B1/en not_active Expired
- 1980-01-31 DE DE8080300281T patent/DE3062095D1/de not_active Expired
- 1980-01-31 DK DK041180A patent/DK159157C/da not_active IP Right Cessation
- 1980-01-31 JP JP1196280A patent/JPS55104288A/ja active Granted
- 1980-01-31 CS CS80658A patent/CS214694B2/cs unknown
- 1980-01-31 IT IT19607/80A patent/IT1130239B/it active
- 1980-01-31 GB GB8003294A patent/GB2041934B/en not_active Expired
- 1980-02-01 PH PH23579A patent/PH15152A/en unknown
- 1980-02-01 RO RO80100063A patent/RO79181A/ro unknown
- 1980-02-01 PL PL1980221748A patent/PL122609B1/pl unknown
- 1980-02-01 AR AR279834A patent/AR228342A1/es active
- 1980-02-01 DD DD80218815A patent/DD148953A5/de unknown
- 1980-02-01 FI FI800300A patent/FI68239C/fi not_active IP Right Cessation
- 1980-02-01 RO RO107056A patent/RO83702B/ro unknown
- 1980-02-01 ES ES488229A patent/ES488229A0/es active Granted
- 1980-02-01 SU SU802877808A patent/SU897109A3/ru active
- 1980-02-01 KR KR1019800000402A patent/KR830001890B1/ko not_active Expired
1981
- 1981-01-26 SU SU813233006A patent/SU938740A3/ru active

Also Published As

Publication number	Publication date
FI800300A7 (fi)	1980-08-02
GR72785B (da)	1983-12-05
NZ192750A (en)	1982-05-25
LU82118A1 (fr)	1980-04-23
ATA49980A (de)	1981-07-15
FI68239C (fi)	1985-08-12
FR2447925A1 (fr)	1980-08-29
RO83702B (ro)	1984-03-30
IL59265A (en)	1983-05-15
DE3062095D1 (en)	1983-03-31
YU22480A (en)	1983-02-28
AT366052B (de)	1982-03-10
CS214694B2 (en)	1982-05-28
DK159157C (da)	1991-02-11
BE881423A (fr)	1980-07-30
CH647525A5 (fr)	1985-01-31
JPS55104288A (en)	1980-08-09
GB2041934B (en)	1983-03-23
AU5502680A (en)	1980-08-07
ES8103098A1 (es)	1981-02-16
IE800191L (en)	1980-08-01
ZA80523B (en)	1981-09-30
RO83702A (ro)	1984-03-15
FI68239B (fi)	1985-04-30
KR830001951A (ko)	1983-05-21
PH15152A (en)	1982-08-24
PL122609B1 (en)	1982-08-31
PT70742A (en)	1980-02-01
ES488229A0 (es)	1981-02-16
EP0014565B1 (en)	1983-02-23
BG32857A3 (bg)	1982-10-15
HU181761B (en)	1983-11-28
RO79181A (ro)	1982-06-25
DD148953A5 (de)	1981-06-17
SU938740A3 (ru)	1982-06-23
GB2041934A (en)	1980-09-17
IT1130239B (it)	1986-06-11
IL59265A0 (en)	1980-05-30
HU182095B (en)	1983-12-28
AR228342A1 (es)	1983-02-28
CA1142173A (en)	1983-03-01
JPH0128035B2 (da)	1989-05-31
IT8019607A0 (it)	1980-01-31
SU897109A3 (ru)	1982-01-07
EP0014565A1 (en)	1980-08-20
FR2447925B1 (da)	1984-02-03
PL221748A1 (da)	1980-12-15
KR830001890B1 (ko)	1983-09-17
DK159157B (da)	1990-09-10
IE49374B1 (en)	1985-09-18
AU532573B2 (en)	1983-10-06

Legal Events

Date	Code	Title	Description
2000-02-14	PUP	Patent expired

Publication	Publication Date	Title
DK29681A (da)	1981-01-22	Fremgangsmaade til fremstilling af immunogammaglobulin
DK546080A (da)	1981-06-21	Fremgangsmaade til fremstilling af galactosaccharosederivater
DK311580A (da)	1981-01-22	Fremgangsmaade til fremstilling af oxoalkylxanthiner
DK6180A (da)	1980-07-11	Fremgangsmaade til fremstilling af 2-pennemforbindelser
DK365280A (da)	1981-02-28	Fremgangsmaade til fremstilling af ftaliminderivater
DK552180A (da)	1981-06-28	Fremgangsmaade til fremstilling af tetrapeptidsemikarbazidderivater
DK307480A (da)	1981-01-18	Fremgangsmaade til fremstilling af neopentylamin
DK274580A (da)	1980-12-29	Fremgangsmaade til fremstilling af tripeptidamider
DK149623C (da)	1987-06-01	Fremgangsmaade til fremstilling af alfa-hydroxycarboxylsyreamider
DK394080A (da)	1981-03-19	Fremgangsmaade til fremstilling af carbostyrilderivater
DK289480A (da)	1981-01-06	Fremgangsmaade til fremstilling af o-substituerede ketoximer
DK153791C (da)	1989-01-23	Fremgangsmaade til fremstilling af 7-hydroxycumaraner
DK481280A (da)	1981-05-16	Fremgangsmaade til fremstilling af piperidylbenzimidazolinonderivater
DK478079A (da)	1981-05-13	Fremgangsmaade til fremstilling af xremet maelkeis
DK262180A (da)	1980-12-21	Fremgangsmaade til fremstilling af alkyl-2-chlorpropionater
DK187980A (da)	1980-11-05	Fremgangsmaade til fremstilling af benzimidazolderivater
DK274680A (da)	1980-12-29	Fremgangsmaade til fremstilling af tripeptidamider
DK222880A (da)	1980-11-23	Fremgangsmaade til fremstilling af anthracyclinonderivater
DK304080A (da)	1981-01-17	Fremgangsmaade til fremstilling af pyrazoloindazolderivater
DK522180A (da)	1981-06-08	Fremgangsmaade til fremstilling af indolderivater
DK277180A (da)	1980-12-30	Fremgangsmaade til fremstilling af tripeptider
DK69680A (da)	1980-08-21	Fremgangsmaade til fremstilling af diorganomagnesiumforbindelser
DK318280A (da)	1981-01-26	Fremgangsmaade til fremstilling af naphthyridinderivater
DK546180A (da)	1981-06-22	Fremgangsmaade til fremstilling af triazepinderivater
DK199981A (da)	1981-05-05	Fremgangsmaade til fremstilling af thiobiscarbamater