DK429788A - Thieno(2,3-beta)thiophen-2-sulfonamid og farmaceutisk praeparat indeholdende en saadan forbindelse - Google Patents

Thieno(2,3-beta)thiophen-2-sulfonamid og farmaceutisk praeparat indeholdende en saadan forbindelse

Info

Publication number: DK429788A
Authority: DK; Denmark
Prior art keywords: thieno; sulphonamide; thiophen; beta; compound
Prior art date: 1987-08-03

Application number

DK429788A

Other languages

Danish (da)

English (en)

Other versions

DK429788D0 (da

Inventor

George D Hartman

John D Prugh

Original Assignee

Merck & Co Inc

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-08-03

Filing date

1988-08-02

Publication date

1989-03-30

1988-08-02 Application filed by Merck & Co Inc filed Critical Merck & Co Inc

1988-08-02 Publication of DK429788D0 publication Critical patent/DK429788D0/da

1989-03-30 Publication of DK429788A publication Critical patent/DK429788A/da

Links

KTFDYVNEGTXQCV-UHFFFAOYSA-N 2-Thiophenesulfonamide Chemical compound NS(=O)(=O)C1=CC=CS1 KTFDYVNEGTXQCV-UHFFFAOYSA-N 0.000 title 1
150000001875 compounds Chemical class 0.000 title 1
239000000825 pharmaceutical preparation Substances 0.000 title 1
208000010412 Glaucoma Diseases 0.000 abstract 1
229940006133 antiglaucoma drug and miotics carbonic anhydrase inhibitors Drugs 0.000 abstract 1
239000003489 carbonate dehydratase inhibitor Substances 0.000 abstract 1
230000004406 elevated intraocular pressure Effects 0.000 abstract 1
NOYGIFXRBNFNHM-UHFFFAOYSA-N thieno[2,3-b]thiophene-5-sulfonamide Chemical class C1=CSC2=C1C=C(S(=O)(=O)N)S2 NOYGIFXRBNFNHM-UHFFFAOYSA-N 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D495/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/06—Antiglaucoma agents or miotics

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Ophthalmology & Optometry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Life Sciences & Earth Sciences (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

DK429788A 1987-08-03 1988-08-02 Thieno(2,3-beta)thiophen-2-sulfonamid og farmaceutisk praeparat indeholdende en saadan forbindelse DK429788A (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US8085187A	1987-08-03	1987-08-03

Publications (2)

Publication Number	Publication Date
DK429788D0 DK429788D0 (da)	1988-08-02
DK429788A true DK429788A (da)	1989-03-30

Family

ID=22160036

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK429788A DK429788A (da)	1987-08-03	1988-08-02	Thieno(2,3-beta)thiophen-2-sulfonamid og farmaceutisk praeparat indeholdende en saadan forbindelse

Country Status (6)

Country	Link
EP (1)	EP0307084B1 (de)
JP (1)	JPH064636B2 (de)
AT (1)	ATE98647T1 (de)
CA (1)	CA1320487C (de)
DE (1)	DE3886314T2 (de)
DK (1)	DK429788A (de)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4894390A (en) *	1987-08-03	1990-01-16	Merck & Co., Inc.	Substituted thieno[2,3-b]thiophene-2-sulfonamides as antiglaucoma agents
US4876271A (en) *	1988-12-20	1989-10-24	Merck & Co., Inc.	Substituted thieno[3,2-b]thiophene-2-sulfonamides as topically active carbonic anhydrase inhibitors
US4929549A (en) *	1989-02-08	1990-05-29	Merck & Co., Inc.	5-carbamoylthieno[2,3-b]thiophene-2-sulfon-amides as topically active carbonic anhydrase inhibitors
US5120757A (en) *	1989-07-31	1992-06-09	Merck & Co., Inc.	Substituted aromatic sulfonamides as antiglaucoma agents
US4946859A (en) *	1989-07-31	1990-08-07	Merck & Co., Inc.	4-(2-methyl-2-hydroxypropylamino)-5,6-dihydrothieno-[2,3-b]thiopyran-2-sulfonamide-7,7-dioxide
EP0480745A3 (en) *	1990-10-12	1992-07-29	Merck & Co. Inc.	Substituted dihydrothieno-thiophene-2-sulfonamides and dioxides thereof
US5216020A (en) *	1990-10-12	1993-06-01	Merck & Co., Inc.	Substituted 4,5-dihydrothieno(2,3-b)thiophene-2-sulfonamides and 6,6-dioxides thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IL72070A (en) *	1983-06-20	1988-11-30	Merck & Co Inc	2-sulfamoylbenzo(b)-thiophene derivatives,their preparation and pharmaceutical compositions containing them
US4863922A (en) *	1984-12-12	1989-09-05	Merck & Co., Inc.	Substituted aromatic sulfonamides as antiglaucoma agents, compositions and use
US4665090A (en) *	1985-10-09	1987-05-12	Merck & Co., Inc.	Substituted thiophene-2-sulfonamide antiglaucoma agents
DE3667056D1 (en) *	1985-12-24	1989-12-28	Merck & Co Inc	Substituted thiophene-2-sulfonamide antiglaucoma agents
EP0271273A3 (de) *	1986-12-08	1989-07-12	Merck & Co. Inc.	Thieno- und Furopyridinsulfonamide

1988
- 1988-07-28 CA CA000573233A patent/CA1320487C/en not_active Expired - Fee Related
- 1988-08-01 AT AT88307099T patent/ATE98647T1/de not_active IP Right Cessation
- 1988-08-01 DE DE3886314T patent/DE3886314T2/de not_active Expired - Fee Related
- 1988-08-01 EP EP88307099A patent/EP0307084B1/de not_active Expired - Lifetime
- 1988-08-02 DK DK429788A patent/DK429788A/da not_active Application Discontinuation
- 1988-08-03 JP JP63194322A patent/JPH064636B2/ja not_active Expired - Lifetime

Also Published As

Publication number	Publication date
DK429788D0 (da)	1988-08-02
EP0307084B1 (de)	1993-12-15
DE3886314T2 (de)	1994-06-16
DE3886314D1 (de)	1994-01-27
EP0307084A1 (de)	1989-03-15
JPS6450886A (en)	1989-02-27
CA1320487C (en)	1993-07-20
ATE98647T1 (de)	1994-01-15
JPH064636B2 (ja)	1994-01-19

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Legal Events

Date	Code	Title	Description
1995-05-08	AHB	Application shelved due to non-payment