DK464386A - 2-substituerede e-kondenserede (1,2,4)-triazolo(1,5-c)pyrimidiner samt deres fremstilling og anvendelse - Google Patents
2-substituerede e-kondenserede (1,2,4)-triazolo(1,5-c)pyrimidiner samt deres fremstilling og anvendelse Download PDFInfo
- Publication number
- DK464386A DK464386A DK464386A DK464386A DK464386A DK 464386 A DK464386 A DK 464386A DK 464386 A DK464386 A DK 464386A DK 464386 A DK464386 A DK 464386A DK 464386 A DK464386 A DK 464386A
- Authority
- DK
- Denmark
- Prior art keywords
- triazolo
- pyrimidines
- condensed
- substituted
- preparation
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
- C07D471/14—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/12—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
- C07D487/14—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
- C07D491/12—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains three hetero rings
- C07D491/14—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
- C07D495/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
- C07D495/14—Ortho-condensed systems
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US78223485A | 1985-09-30 | 1985-09-30 | |
| US78223485 | 1985-09-30 | ||
| US84198686A | 1986-03-20 | 1986-03-20 | |
| US84198686 | 1986-03-20 |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| DK464386D0 DK464386D0 (da) | 1986-09-29 |
| DK464386A true DK464386A (da) | 1987-03-31 |
| DK168046B1 DK168046B1 (da) | 1994-01-24 |
Family
ID=27119971
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK464386A DK168046B1 (da) | 1985-09-30 | 1986-09-29 | 2-substituerede cycloalkenooeeaaoe1,2,4aatriazolooe1,5-caapyrimidiner, deres tautomerer og farmaceutisk acceptable salte samt fremgangsmaade til fremstilling deraf |
Country Status (9)
| Country | Link |
|---|---|
| EP (1) | EP0217748B1 (da) |
| CA (1) | CA1288097C (da) |
| DE (1) | DE3677445D1 (da) |
| DK (1) | DK168046B1 (da) |
| ES (1) | ES2002012A6 (da) |
| FI (1) | FI84068C (da) |
| GR (1) | GR862456B (da) |
| IE (1) | IE58968B1 (da) |
| PT (1) | PT83453B (da) |
Families Citing this family (22)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3781080T2 (de) * | 1986-09-30 | 1992-12-24 | Ciba Geigy Ag | 2-substituierte-e-kondensierte(1,2,4)triazolo-(1,5-c)pyrimidine, pharmazeutische zubereitungen und ihre verwendung. |
| IE64917B1 (en) * | 1988-02-05 | 1995-09-20 | Riker Laboratories Inc | Triazolo[1,5-c]pyrimido[1,4]azines as bronchodilators |
| EP0459702A1 (en) * | 1990-05-29 | 1991-12-04 | Zeneca Limited | Azole Derivatives |
| US5095015A (en) * | 1990-07-24 | 1992-03-10 | Neurogen Corporation | Certain azacycloalkyl imidazopyrimidines; a new class of gaba brain receptor ligands |
| US5185446A (en) * | 1990-09-04 | 1993-02-09 | Neurogen Corporation | Certain cycloalkyl imidazopyrimidines; a new class of gaba brainreceptor ligands |
| GB9111131D0 (en) * | 1991-05-23 | 1991-07-17 | Ici Plc | Heterocyclic compounds |
| GB9111130D0 (en) * | 1991-05-23 | 1991-07-17 | Ici Plc | Azole derivatives |
| GB9125002D0 (en) * | 1991-11-25 | 1992-01-22 | Ici Plc | Azole derivatives |
| DE4241562A1 (de) * | 1992-12-10 | 1994-06-16 | Basf Ag | Neue Triazolopyrimidone, ihre Herstellung und Verwendung |
| IT1264901B1 (it) * | 1993-06-29 | 1996-10-17 | Schering Plough S P A | Analoghi eterociclici di 1,2,4-triazolo(15-c)pirimidine ad attivita' antagonista per il recettore a2 dell'adenosina |
| US5565460A (en) * | 1993-07-27 | 1996-10-15 | Kyowa Hakko Koygo Co., Ltd. | Therapeutic purine agents for parkinson's disease |
| US5494887A (en) * | 1994-07-11 | 1996-02-27 | Dowelanco | Ring annulated 5-alkoxy-n-aryl[1,2,4]triazolo[1,5-C]-pyrimidine-2-sulfonamide herbicides |
| US5792766A (en) * | 1996-03-13 | 1998-08-11 | Neurogen Corporation | Imidazo 1,5-c! quinazolines; a new class of GABA brain receptor ligands |
| US5677309A (en) * | 1996-03-22 | 1997-10-14 | Neurogen Corporation | 1,2,4-triazolo 4,3-c! quinazolin-3-ones and 1,2,4-triazolo 4,3-c!quinazolin-3-thiones; a new class of GABA brain receptor ligands |
| US5955465A (en) * | 1996-03-22 | 1999-09-21 | Neurogen Corporation | 1,2,4-triazolo 4,3-c!quinazolin-3-ones and 1,2,4-triazolo 4,3-c!quinazolin-3-thiones |
| ES2137113B1 (es) * | 1997-07-29 | 2000-09-16 | Almirall Prodesfarma Sa | Nuevos derivados de triazolo-piridazinas heterociclicos. |
| CA2326716C (en) * | 1998-04-03 | 2006-12-12 | Otsuka Pharmaceutical Factory, Inc. | Triazolopurine derivative, pharmaceutical composition containing the derivative, adenosine a3 receptor ligand, and remedy for asthma |
| PT1283839E (pt) | 2000-05-26 | 2005-08-31 | Schering Corp | Antagonistas do receptor a2a da adenosina |
| PA8539501A1 (es) * | 2001-02-14 | 2002-09-30 | Warner Lambert Co | Compuestos triazolo como inhibidores de mmp |
| JP4545437B2 (ja) | 2001-10-15 | 2010-09-15 | シェーリング コーポレイション | アデノシンａ２ａ受容体アンタゴニストとしてのイミダゾ（４，３−ｅ）−１，２，４−トリアゾロ（１，５−ｃ）ピリミジン |
| US7196106B2 (en) | 2002-11-05 | 2007-03-27 | Merck & Co., Inc | Cyanothiophene derivatives, compositions containing such compounds and methods of use |
| US9499562B2 (en) | 2012-06-18 | 2016-11-22 | Dart Neuroscience (Cayman) Ltd. | Substituted thiophene- and furan-fused azolopyrimidine-5-(6H)-one compounds |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3045015A (en) * | 1958-10-03 | 1962-07-17 | Ici Ltd | Triazolo-[2, 3-c]-pyrimidines |
| BE792856A (fr) * | 1971-12-17 | 1973-06-15 | Sandoz Sa | Nouveaux derives de la triazolo-quinazoline, leur preparation et medicaments contenant ces |
| US4252945A (en) * | 1979-07-11 | 1981-02-24 | E. R. Squibb & Sons, Inc. | Process for preparing pyrazolo[1,5-c]-quinazoline derivatives and novel intermediates |
| DE3146599A1 (de) * | 1981-11-25 | 1983-07-07 | Basf Ag, 6700 Ludwigshafen | Neue triazolochinazoline, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische zubereitungen |
| EP0181282A1 (de) * | 1984-10-01 | 1986-05-14 | Ciba-Geigy Ag | Triazolochinazolinverbindungen |
-
1986
- 1986-09-25 DE DE8686810421T patent/DE3677445D1/de not_active Expired - Lifetime
- 1986-09-25 EP EP86810421A patent/EP0217748B1/en not_active Expired - Lifetime
- 1986-09-26 CA CA000519161A patent/CA1288097C/en not_active Expired - Lifetime
- 1986-09-26 FI FI863904A patent/FI84068C/fi not_active IP Right Cessation
- 1986-09-29 IE IE257586A patent/IE58968B1/en not_active IP Right Cessation
- 1986-09-29 GR GR862456A patent/GR862456B/el unknown
- 1986-09-29 DK DK464386A patent/DK168046B1/da not_active IP Right Cessation
- 1986-09-29 ES ES8602265A patent/ES2002012A6/es not_active Expired
- 1986-09-29 PT PT83453A patent/PT83453B/pt not_active IP Right Cessation
Also Published As
| Publication number | Publication date |
|---|---|
| EP0217748A2 (en) | 1987-04-08 |
| FI84068B (fi) | 1991-06-28 |
| FI863904A7 (fi) | 1987-03-31 |
| PT83453A (en) | 1986-10-01 |
| EP0217748A3 (en) | 1988-01-07 |
| PT83453B (pt) | 1989-05-12 |
| DE3677445D1 (de) | 1991-03-14 |
| IE862575L (en) | 1987-03-30 |
| EP0217748B1 (en) | 1991-02-06 |
| DK464386D0 (da) | 1986-09-29 |
| IE58968B1 (en) | 1993-12-01 |
| ES2002012A6 (es) | 1988-07-01 |
| DK168046B1 (da) | 1994-01-24 |
| FI863904A0 (fi) | 1986-09-26 |
| GR862456B (en) | 1987-01-29 |
| FI84068C (fi) | 1991-10-10 |
| CA1288097C (en) | 1991-08-27 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B1 | Patent granted (law 1993) | ||
| PBP | Patent lapsed |