DK474288D0 - Benzimidazolderivater og fremgangsmaade til fremstilling deraf samt laegemiddel indeholdende benzimidazolderivaterne - Google Patents

Benzimidazolderivater og fremgangsmaade til fremstilling deraf samt laegemiddel indeholdende benzimidazolderivaterne

Info

Publication number: DK474288D0
Authority: DK; Denmark
Prior art keywords: benzimidazold; derivatives; procedures; preparing; benzimidazold derivatives
Prior art date: 1987-08-25

Application number

DK474288A

Other languages

English (en)

Other versions

DK474288A (da

DK169701B1 (da

Inventor

Klaus Schoellkopf

Helmut Wachtel

Original Assignee

Schering Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1987-08-25

Filing date

1988-08-25

Publication date

1988-08-25

1988-08-25 Application filed by Schering Ag filed Critical Schering Ag

1988-08-25 Publication of DK474288D0 publication Critical patent/DK474288D0/da

1989-02-26 Publication of DK474288A publication Critical patent/DK474288A/da

1995-01-16 Application granted granted Critical

1995-01-16 Publication of DK169701B1 publication Critical patent/DK169701B1/da

Links

229940126601 medicinal product Drugs 0.000 title 1
238000000034 method Methods 0.000 title 1
IWPAPERMAWYYDD-UHFFFAOYSA-N 4-(2-aminoethyl)-1,3-dihydrobenzimidazol-2-one Chemical compound NCCC1=CC=CC2=C1NC(=O)N2 IWPAPERMAWYYDD-UHFFFAOYSA-N 0.000 abstract 1
125000001183 hydrocarbyl group Chemical group 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
- C07D409/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings
- C07D409/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/12—Antihypertensives
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/26—Oxygen atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D235/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings
- C07D235/02—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, condensed with other rings condensed with carbocyclic rings or ring systems
- C07D235/04—Benzimidazoles; Hydrogenated benzimidazoles
- C07D235/24—Benzimidazoles; Hydrogenated benzimidazoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 2
- C07D235/28—Sulfur atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Urology & Nephrology (AREA)
Vascular Medicine (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Plural Heterocyclic Compounds (AREA)
Medicinal Preparation (AREA)

DK474288A 1987-08-25 1988-08-25 Benzimidazolderivater og fremgangsmåder til fremstilling deraf samt lægemiddel indeholdende benzimidazolderivaterne DK169701B1 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE3728695		1987-08-25
DE19873728695 DE3728695A1 (de)	1987-08-25	1987-08-25	Neue benzimidazol-derivate

Publications (3)

Publication Number	Publication Date
DK474288D0 true DK474288D0 (da)	1988-08-25
DK474288A DK474288A (da)	1989-02-26
DK169701B1 DK169701B1 (da)	1995-01-16

Family

ID=6334659

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK474288A DK169701B1 (da)	1987-08-25	1988-08-25	Benzimidazolderivater og fremgangsmåder til fremstilling deraf samt lægemiddel indeholdende benzimidazolderivaterne

Country Status (17)

Country	Link
US (1)	US4925854A (da)
EP (1)	EP0304789B1 (da)
JP (1)	JP2818170B2 (da)
AT (1)	ATE86982T1 (da)
AU (1)	AU615939B2 (da)
CA (1)	CA1330440C (da)
DD (1)	DD274215A5 (da)
DE (2)	DE3728695A1 (da)
DK (1)	DK169701B1 (da)
ES (1)	ES2054752T3 (da)
FI (1)	FI99013C (da)
HU (1)	HU201746B (da)
IE (1)	IE63283B1 (da)
IL (1)	IL87561A (da)
NO (1)	NO170852C (da)
PT (1)	PT88326B (da)
ZA (1)	ZA886336B (da)

Families Citing this family (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IE914003A1 (en) *	1990-11-20	1992-05-20	Astra Pharma Prod	Biologically Active Amines
US5371102A (en) *	1992-03-11	1994-12-06	University Of Hawaii	Compositions and methods of inhibiting thyroid activity
PE27997A1 (es)	1994-04-29	1997-09-20	Lilly Co Eli	Antagonistas de receptores de taquicininas
US5565454A (en) *	1995-05-31	1996-10-15	Ergo Science, Incorporated	Method for preventing intervention-associated stenosis and other symptoms associated with stenosis of blood vessels following non-bypass, invasive interventions
TW356468B (en) *	1995-09-15	1999-04-21	Astra Pharma Prod	Benzothiazolone compounds useful as beta2-adrenoreceptor and dopamine DA2 receptor agonists process for preparing same and pharmaceutical compositions containing same
GB9526511D0 (en) *	1995-12-23	1996-02-28	Astra Pharma Prod	Pharmaceutically active compounds
WO2004032861A2 (en) *	2002-10-11	2004-04-22	Bristol-Myers Squibb Company	Hexahydro-benzimidazolone compounds useful as anti-inflammatory agents
MX346346B (es)	2011-12-16	2017-03-14	Colgate Palmolive Co	Composiciones que cambian de color.

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US3813409A (en) *	1972-07-31	1974-05-28	Squibb & Sons Inc	Benzimidazolinone compounds
DE3042481A1 (de) *	1980-11-11	1982-06-16	A. Nattermann & Cie GmbH, 5000 Köln	(omega)-(2-oxo-benzazolinyl)-alkansaeure-derivate, verfahren zu ihrer herstellung und diese enthaltende pharmazeutische praeparate
US4367337A (en) *	1981-01-05	1983-01-04	The Sherwin-Williams Company	Process for conversion of benzimidazolones to benzotriazoles
WO1986001204A1 (en) *	1984-08-15	1986-02-27	Schering Aktiengesellschaft	New dopamine derivatives, process for their production, and their use as medicinal products
US4554287A (en) *	1984-09-12	1985-11-19	Smithkline Beckman Corporation	Antihypertensive 7-[2-(dialkylamino)ethyl]-4-hydroxy-1,3-benzimidazol-2-ones

1987
- 1987-08-25 DE DE19873728695 patent/DE3728695A1/de not_active Withdrawn
1988
- 1988-08-17 ES ES88113339T patent/ES2054752T3/es not_active Expired - Lifetime
- 1988-08-17 DE DE8888113339T patent/DE3879322D1/de not_active Expired - Lifetime
- 1988-08-17 EP EP88113339A patent/EP0304789B1/de not_active Expired - Lifetime
- 1988-08-17 AT AT88113339T patent/ATE86982T1/de active
- 1988-08-22 IE IE255288A patent/IE63283B1/en not_active IP Right Cessation
- 1988-08-23 DD DD88319141A patent/DD274215A5/de not_active IP Right Cessation
- 1988-08-23 JP JP63207486A patent/JP2818170B2/ja not_active Expired - Lifetime
- 1988-08-24 NO NO883776A patent/NO170852C/no unknown
- 1988-08-24 CA CA000575617A patent/CA1330440C/en not_active Expired - Fee Related
- 1988-08-24 PT PT88326A patent/PT88326B/pt not_active IP Right Cessation
- 1988-08-24 HU HU884447A patent/HU201746B/hu not_active IP Right Cessation
- 1988-08-25 IL IL87561A patent/IL87561A/xx not_active IP Right Cessation
- 1988-08-25 FI FI883930A patent/FI99013C/fi not_active IP Right Cessation
- 1988-08-25 US US07/236,383 patent/US4925854A/en not_active Expired - Fee Related
- 1988-08-25 AU AU21498/88A patent/AU615939B2/en not_active Ceased
- 1988-08-25 DK DK474288A patent/DK169701B1/da not_active IP Right Cessation
- 1988-08-25 ZA ZA886336A patent/ZA886336B/xx unknown

Also Published As

Publication number	Publication date
FI883930L (fi)	1989-02-26
ATE86982T1 (de)	1993-04-15
PT88326A (pt)	1989-06-30
IL87561A0 (en)	1989-01-31
IE63283B1 (en)	1995-04-05
FI99013B (fi)	1997-06-13
ZA886336B (en)	1989-04-26
HU201746B (en)	1990-12-28
DE3728695A1 (de)	1989-03-09
AU2149888A (en)	1989-03-02
DK474288A (da)	1989-02-26
CA1330440C (en)	1994-06-28
FI99013C (fi)	1997-09-25
NO170852B (no)	1992-09-07
NO883776L (no)	1989-02-27
ES2054752T3 (es)	1994-08-16
IE882552L (en)	1989-02-25
FI883930A0 (fi)	1988-08-25
EP0304789A3 (en)	1989-10-04
DK169701B1 (da)	1995-01-16
HUT49589A (en)	1989-10-30
NO883776D0 (no)	1988-08-24
AU615939B2 (en)	1991-10-17
JPS6468359A (en)	1989-03-14
JP2818170B2 (ja)	1998-10-30
IL87561A (en)	1993-02-21
DE3879322D1 (de)	1993-04-22
EP0304789B1 (de)	1993-03-17
DD274215A5 (de)	1989-12-13
PT88326B (pt)	1995-03-31
EP0304789A2 (de)	1989-03-01
US4925854A (en)	1990-05-15
NO170852C (no)	1992-12-16

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Legal Events

Date	Code	Title	Description
1995-01-16	B1	Patent granted (law 1993)
1999-05-10	PBP	Patent lapsed