DK519488D0 - Substituerede pyridiner, fremgangsmaader til fremstilling heraf, mellemprodukter, som er anvendelige ved deres fremstilling samt farmaceutiske midler indeholdende dem - Google Patents

Substituerede pyridiner, fremgangsmaader til fremstilling heraf, mellemprodukter, som er anvendelige ved deres fremstilling samt farmaceutiske midler indeholdende dem

Info

Publication number
DK519488D0
DK519488D0 DK519488A DK519488A DK519488D0 DK 519488 D0 DK519488 D0 DK 519488D0 DK 519488 A DK519488 A DK 519488A DK 519488 A DK519488 A DK 519488A DK 519488 D0 DK519488 D0 DK 519488D0
Authority
DK
Denmark
Prior art keywords
procedures
preparation
production
pharmaceutical agents
agents containing
Prior art date
Application number
DK519488A
Other languages
English (en)
Other versions
DK519488A (da
Inventor
Lawrence Ivan Kruse
Stephen Torey Ross
Original Assignee
Smithkline Beckman Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beckman Corp filed Critical Smithkline Beckman Corp
Publication of DK519488D0 publication Critical patent/DK519488D0/da
Publication of DK519488A publication Critical patent/DK519488A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/63—One oxygen atom
    • C07D213/64—One oxygen atom attached in position 2 or 6
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D213/62—Oxygen or sulfur atoms
    • C07D213/70—Sulfur atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pyridine Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK519488A 1987-09-17 1988-09-16 Substituerede pyridiner, fremgangsmaader til fremstilling heraf, mellemprodukter, som er anvendelige ved deres fremstilling samt farmaceutiske midler indeholdende dem DK519488A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US07/097,988 US4839371A (en) 1987-09-17 1987-09-17 3-aralkyl-2-mercaptoyridines as dopamine-β-hydroxylase inhibitors

Publications (2)

Publication Number Publication Date
DK519488D0 true DK519488D0 (da) 1988-09-16
DK519488A DK519488A (da) 1989-03-18

Family

ID=22266083

Family Applications (1)

Application Number Title Priority Date Filing Date
DK519488A DK519488A (da) 1987-09-17 1988-09-16 Substituerede pyridiner, fremgangsmaader til fremstilling heraf, mellemprodukter, som er anvendelige ved deres fremstilling samt farmaceutiske midler indeholdende dem

Country Status (6)

Country Link
US (1) US4839371A (da)
EP (1) EP0308159A3 (da)
JP (1) JPH01104053A (da)
AU (1) AU2223088A (da)
DK (1) DK519488A (da)
PT (1) PT88509A (da)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US5308854A (en) * 1990-06-18 1994-05-03 Merck & Co., Inc. Inhibitors of HIV reverse transcriptase
DE602004023106D1 (de) 2003-11-07 2009-10-22 Senju Pharma Co Pharmazeutische zusammensetzung mit prostaglandin
US9567316B2 (en) 2012-03-07 2017-02-14 The Mclean Hospital Corporation Aminoquinoline derivatives and uses thereof
KR102172771B1 (ko) 2020-06-16 2020-11-02 주식회사 세화 개별 검지 기능을 갖는 led 신호기 및 이를 이용한 신호 방법

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7016899A (da) * 1969-12-03 1971-06-07
US3853900A (en) * 1973-09-14 1974-12-10 Searle & Co 4-benzyloxy-2 (1h)-pyridones
US4487761A (en) * 1982-04-05 1984-12-11 Merck & Co., Inc. Dopamine β-hydroxylase inhibitors
US4532331A (en) * 1983-04-12 1985-07-30 Smithkline Beckman Corporation 1-Benzyl-2-aminomethyl imidazole derivatives

Also Published As

Publication number Publication date
EP0308159A3 (en) 1990-01-10
US4839371A (en) 1989-06-13
PT88509A (pt) 1989-07-31
EP0308159A2 (en) 1989-03-22
DK519488A (da) 1989-03-18
AU2223088A (en) 1989-03-23
JPH01104053A (ja) 1989-04-21

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Legal Events

Date Code Title Description
AHB Application shelved due to non-payment