DK519984D0 - Milbemycinderivater samt deres fremstilling og anvendelse - Google Patents

Milbemycinderivater samt deres fremstilling og anvendelse

Info

Publication number: DK519984D0
Authority: DK; Denmark
Prior art keywords: formula; image; derivatives; milbemycine; preparation
Prior art date: 1983-11-02

Application number

DK519984A

Other languages

English (en)

Other versions

DK519984A (da

Inventor

Jean-Claude Gehret

Original Assignee

Ciba Geigy Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1983-11-02

Filing date

1984-11-01

Publication date

1984-11-01

1984-11-01 Application filed by Ciba Geigy Ag filed Critical Ciba Geigy Ag

1984-11-01 Publication of DK519984D0 publication Critical patent/DK519984D0/da

1985-05-03 Publication of DK519984A publication Critical patent/DK519984A/da

Links

FXWHFKOXMBTCMP-WMEDONTMSA-N milbemycin Natural products COC1C2OCC3=C/C=C/C(C)CC(=CCC4CC(CC5(O4)OC(C)C(C)C(OC(=O)C(C)CC(C)C)C5O)OC(=O)C(C=C1C)C23O)C FXWHFKOXMBTCMP-WMEDONTMSA-N 0.000 abstract 2
241001465754 Metazoa Species 0.000 abstract 1
241000244206 Nematoda Species 0.000 abstract 1
125000002252 acyl group Chemical group 0.000 abstract 1
QVGXLLKOCUKJST-UHFFFAOYSA-N atomic oxygen Chemical compound [O] QVGXLLKOCUKJST-UHFFFAOYSA-N 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
244000078703 ectoparasite Species 0.000 abstract 1
125000001495 ethyl group Chemical group [H]C([H])([H])C([H])([H])* 0.000 abstract 1
239000001257 hydrogen Substances 0.000 abstract 1
229910052739 hydrogen Inorganic materials 0.000 abstract 1
125000004435 hydrogen atom Chemical group [H]* 0.000 abstract 1
239000000543 intermediate Substances 0.000 abstract 1
125000001449 isopropyl group Chemical group [H]C([H])([H])C([H])(*)C([H])([H])[H] 0.000 abstract 1
125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
239000000203 mixture Substances 0.000 abstract 1
230000003647 oxidation Effects 0.000 abstract 1
238000007254 oxidation reaction Methods 0.000 abstract 1
239000001301 oxygen Substances 0.000 abstract 1
229910052760 oxygen Inorganic materials 0.000 abstract 1
244000045947 parasite Species 0.000 abstract 1
125000002914 sec-butyl group Chemical group [H]C([H])([H])C([H])([H])C([H])(*)C([H])([H])[H] 0.000 abstract 1
125000003808 silyl group Chemical group [H][Si]([H])([H])[*] 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
- C07D493/22—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains four or more hetero rings
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
- C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N55/00—Biocides, pest repellants or attractants, or plant growth regulators, containing organic compounds containing elements other than carbon, hydrogen, halogen, oxygen, nitrogen and sulfur
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents

Landscapes

Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Zoology (AREA)
Dentistry (AREA)
Environmental Sciences (AREA)
Wood Science & Technology (AREA)
Agronomy & Crop Science (AREA)
Pest Control & Pesticides (AREA)
Plant Pathology (AREA)
Genetics & Genomics (AREA)
Veterinary Medicine (AREA)
Biotechnology (AREA)
Biochemistry (AREA)
Molecular Biology (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Tropical Medicine & Parasitology (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Pyrane Compounds (AREA)

DK519984A 1983-11-02 1984-11-01 Milbemycinderivater samt deres fremstilling og anvendelse DK519984A (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
CH590983		1983-11-02
CH473684		1984-10-02

Publications (2)

Publication Number	Publication Date
DK519984D0 true DK519984D0 (da)	1984-11-01
DK519984A DK519984A (da)	1985-05-03

Family

ID=25696163

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK519984A DK519984A (da)	1983-11-02	1984-11-01	Milbemycinderivater samt deres fremstilling og anvendelse

Country Status (10)

Country	Link
US (1)	US4582852A (da)
EP (1)	EP0144285B1 (da)
JP (1)	JPS60120880A (da)
KR (1)	KR850003894A (da)
AT (1)	ATE38230T1 (da)
AU (1)	AU575871B2 (da)
CA (1)	CA1257586A (da)
DE (1)	DE3474825D1 (da)
DK (1)	DK519984A (da)
IL (1)	IL73384A (da)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS60126289A (ja) *	1983-11-14	1985-07-05	Sankyo Co Ltd	ミルベマイシン類の５−カ−ボネ−ト誘導体
US4584314A (en) *	1983-11-25	1986-04-22	Ciba-Geigy Corporation	Lactone derivative, process for the preparation thereof, and use thereof in pest control
DK614084A (da) *	1983-12-30	1985-07-01	Ciba Geigy Ag	Milbemycim-derivater samt deres fremstilling og anvendelse
US4696922A (en) *	1984-11-26	1987-09-29	Ciba-Geigy Corporation	5-azolylacetoxymilbemycins as ecto- and endoparasites
US4857509A (en) *	1985-01-22	1989-08-15	Ciba-Geigy Corporation	13β-alkylmilbemycin derivatives for controlling parasites of animals and plants
US4666937A (en) *	1985-03-04	1987-05-19	Merck & Co., Inc.	Avermectin bioconversion products
AR243528A1 (es) *	1986-12-11	1993-08-31	Sankyo Co	Procedimiento para preparar compuestos de macrolida y un procedimiento para producir con los mismos una composicion parasiticida.
US5212322A (en) *	1986-12-11	1993-05-18	Sankyo Company, Limited	Macrolide compounds, their preparation and their use
EP0285561A3 (de) *	1987-03-27	1989-10-25	Ciba-Geigy Ag	Parasitizide und insektizide Milbemycin-Derivate
JPH0631246B2 (ja) *	1988-02-02	1994-04-27	三共株式会社	５−オキソミルベマイシン誘導体の製造方法
EP0524686A1 (en) *	1991-07-23	1993-01-27	Merck & Co. Inc.	A process for the 14a-hydroxylation of avermectin compounds
US5312753A (en) *	1992-03-23	1994-05-17	Merck & Co., Inc.	Strain of streptomyces avermitilis capable of glycosylating avermectin compounds at the 13- and 14A positions
JP4373080B2 (ja) *	2002-12-24	2009-11-25	三井化学アグロ株式会社	ミルベマイシン類の精製法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4201861A (en) *	1977-10-03	1980-05-06	Merck & Co., Inc.	Acyl derivatives of C-076 compounds
US4173571A (en) *	1977-12-19	1979-11-06	Merck & Co., Inc.	13-Halo and 13-deoxy derivatives of C-076 compounds
US4328335A (en) *	1979-08-13	1982-05-04	Merck & Co., Inc.	Process for the interconversion of C-076 compounds
US4289760A (en) *	1980-05-02	1981-09-15	Merck & Co., Inc.	23-Keto derivatives of C-076 compounds
US4469682A (en) *	1983-01-28	1984-09-04	Merck & Co., Inc.	Avermectin and milbemycin phosphate esters, pharmaceutical compositions, and method of use
US4584314A (en) *	1983-11-25	1986-04-22	Ciba-Geigy Corporation	Lactone derivative, process for the preparation thereof, and use thereof in pest control
DK614084A (da) *	1983-12-30	1985-07-01	Ciba Geigy Ag	Milbemycim-derivater samt deres fremstilling og anvendelse
EP0165900A3 (de) *	1984-06-08	1986-05-28	Ciba-Geigy Ag	Neue Lactone, Verfahren zu ihrer Herstellung und ihre Verwendung in der Schädlingsbekämpfung

1984
- 1984-10-25 US US06/664,677 patent/US4582852A/en not_active Expired - Lifetime
- 1984-10-29 EP EP84810519A patent/EP0144285B1/de not_active Expired
- 1984-10-29 DE DE8484810519T patent/DE3474825D1/de not_active Expired
- 1984-10-29 AT AT84810519T patent/ATE38230T1/de not_active IP Right Cessation
- 1984-10-31 CA CA000466670A patent/CA1257586A/en not_active Expired
- 1984-10-31 IL IL73384A patent/IL73384A/xx unknown
- 1984-11-01 JP JP59229065A patent/JPS60120880A/ja active Granted
- 1984-11-01 DK DK519984A patent/DK519984A/da not_active Application Discontinuation
- 1984-11-01 AU AU34907/84A patent/AU575871B2/en not_active Ceased
- 1984-11-02 KR KR1019840006869A patent/KR850003894A/ko not_active Ceased

Also Published As

Publication number	Publication date
DK519984A (da)	1985-05-03
CA1257586A (en)	1989-07-18
IL73384A (en)	1988-01-31
US4582852A (en)	1986-04-15
AU3490784A (en)	1985-05-09
KR850003894A (ko)	1985-06-29
ATE38230T1 (de)	1988-11-15
IL73384A0 (en)	1985-01-31
DE3474825D1 (en)	1988-12-01
JPS60120880A (ja)	1985-06-28
JPH0564154B2 (da)	1993-09-14
EP0144285B1 (de)	1988-10-26
AU575871B2 (en)	1988-08-11
EP0144285A1 (de)	1985-06-12

Legal Events

Date	Code	Title
1985-01-01	AHS	Application shelved for other reasons than non-payment
1988-07-04	AHB	Application shelved due to non-payment
1990-10-01	AHS	Application shelved for other reasons than non-payment

Publication	Publication Date	Title
DK519984A (da)	1985-05-03	Milbemycinderivater samt deres fremstilling og anvendelse
ES8708232A1 (es)	1987-10-01	Procedimiento para la produccion de derivados de la 13-beta-milbemicina
FI864150A0 (fi)	1986-10-14	Kemiska foereningar.
DK369482A (da)	1983-02-19	6alfa-methylprednisolonderivater, deres fremstilling og anvendelse
ATE159885T1 (de)	1997-11-15	Fungizide zusammensetzungen
ES8201560A1 (es)	1981-12-16	Un procedimiento para la preparacion de derivados de oxazo- lidona- o tiazolidona.
PH24355A (en)	1990-06-13	Macrolide compounds,composition said compound and method of use thereof
DK465484D0 (da)	1984-09-28	Cyclohexenon-derivater til anvendelse som herbicider og fremgangsmaade til fremstilling af saadanne derivater
BR8504580A (pt)	1986-07-15	Composto de benzoil-ureia,composicao inseticida,processo para controlar insetos e processo para a preparacao de um composto inseticida
DK251284D0 (da)	1984-05-22	Substituerede 1,2,3-triazino(4',5'.4,5)thieno(2,3-b)-quinolin-4(3h)-oner eller syreadditionssalte deraf og deres fremstilling
PT88462A (pt)	1988-10-01	Process for the preparation of macrolide compounds and of compositions containing them
DE68927070D1 (de)	1996-10-10	Makrolid-Derivate
DE3851190D1 (de)	1994-09-29	Makrolid-Derivate.
AU558254B2 (en)	1987-01-22	Imidazolecarboxylic acid derivatives as cardiotonics
DK484988D0 (da)	1988-08-31	Thionophosphonsyreestere, deres fremstilling og anvendelse til bekaempelse af skadelige organismer
DK378382A (da)	1983-02-26	N-substituerede tetrahydroisophthalimidderivater
FI921848L (fi)	1992-04-24	Nya pleuromutilinderivator.
DK384685A (da)	1986-02-25	Substituerede 1-phenyl-3-benzoyl-(thio)urinstoffer, deres fremstilling og anvendelse til bekaempelse af skadelige organismer samt ved fremstillingen anvendelige udgangsforbindelser og disses fremstilling
JPS53111080A (en)	1978-09-28	2-phenyl-4h-1,3-thiazine derivative, its preparation and use
GEP19970660B (en)	1997-01-04	Macrolide compounds
BG49444A1 (en)	1991-11-15	Acylureidoamynotiasolylni derivatives and method for their preparation
SE7909980L (sv)	1980-06-14	I-amino-indolin-derivat, deras framstellning och farmaceutiska kompositioner innehallande desamma