DK547181A - Fremgangsmaade til fremstilling af halogenmethylestere af penicillansyresulfon og mellemprodukter ved fremgangsmaaden - Google Patents

Fremgangsmaade til fremstilling af halogenmethylestere af penicillansyresulfon og mellemprodukter ved fremgangsmaaden

Info

Publication number
DK547181A
DK547181A DK547181A DK547181A DK547181A DK 547181 A DK547181 A DK 547181A DK 547181 A DK547181 A DK 547181A DK 547181 A DK547181 A DK 547181A DK 547181 A DK547181 A DK 547181A
Authority
DK
Denmark
Prior art keywords
procedure
halogene
methylesters
penicillanic
sulphones
Prior art date
Application number
DK547181A
Other languages
English (en)
Other versions
DK158228B (da
DK158228C (da
Inventor
D L Hageman
T C Crawford
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of DK547181A publication Critical patent/DK547181A/da
Publication of DK158228B publication Critical patent/DK158228B/da
Application granted granted Critical
Publication of DK158228C publication Critical patent/DK158228C/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/04Preparation
    • C07D499/08Modification of a carboxyl radical directly attached in position 2, e.g. esterification
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D499/00Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Oncology (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK547181A 1980-12-11 1981-12-10 Fremgangsmaade til fremstilling af halogenalkylestere af penicillansyresulfon og udgangsmateriale til anvendelse ved fremgangsmaaden DK158228C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US21521580 1980-12-11
US06/215,215 US4361513A (en) 1980-12-11 1980-12-11 Esters of penicillanic acid sulfone

Publications (3)

Publication Number Publication Date
DK547181A true DK547181A (da) 1982-06-12
DK158228B DK158228B (da) 1990-04-16
DK158228C DK158228C (da) 1990-09-24

Family

ID=22802118

Family Applications (1)

Application Number Title Priority Date Filing Date
DK547181A DK158228C (da) 1980-12-11 1981-12-10 Fremgangsmaade til fremstilling af halogenalkylestere af penicillansyresulfon og udgangsmateriale til anvendelse ved fremgangsmaaden

Country Status (20)

Country Link
US (1) US4361513A (da)
EP (1) EP0054397B1 (da)
JP (1) JPS57122089A (da)
KR (1) KR850001340B1 (da)
AR (1) AR229599A1 (da)
AT (1) ATE12233T1 (da)
AU (1) AU527159B2 (da)
CA (1) CA1177068A (da)
DE (1) DE3169462D1 (da)
DK (1) DK158228C (da)
ES (1) ES507867A0 (da)
FI (1) FI75824C (da)
GR (1) GR76963B (da)
IE (1) IE52111B1 (da)
IL (1) IL64497A0 (da)
NO (1) NO160517C (da)
PH (1) PH17469A (da)
PT (1) PT74111B (da)
YU (1) YU43053B (da)
ZA (1) ZA818579B (da)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4746754A (en) * 1986-05-16 1988-05-24 The Dow Chemical Company Preparation of carbonate diisocyanates and related compounds
US7968279B2 (en) * 2008-08-13 2011-06-28 Beckman Coulter, Inc. Reference control for cell by cell analysis
PL2969715T3 (pl) 2013-03-13 2021-07-19 Andrew Bacon Ulepszenia efektywności paliwowej pojazdów drogowych

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS512477A (en) * 1974-06-25 1976-01-10 Zekoo Kk Ijokeisha shindonokanchisochi
JPS512476A (ja) * 1974-06-25 1976-01-10 Inoue Japax Res Hokokei
JPS6056160B2 (ja) * 1977-06-07 1985-12-09 フアイザ−・インコ−ポレ−テツド β−ラクタマ−ゼ阻害剤としてのペニシラン酸1,1−ジオキシド
US4272439A (en) * 1978-06-02 1981-06-09 Schering Corporation 6-(Substituted-hydroxymethylene penams)
US4241050A (en) * 1978-09-01 1980-12-23 Pfizer Inc. Penam 1,1-dioxides as beta-lactamase inhibitors
US4331677A (en) * 1978-11-24 1982-05-25 Farmitalia Carlo Erba S.P.A. 7-Oxo-4-1-aza-bicyclo-[3,2,0]-heptane derivatives
US4256733A (en) * 1979-09-26 1981-03-17 Pfizer Inc. Acetoxymethyl penam compounds as β-lactamase inhibitors

Also Published As

Publication number Publication date
EP0054397B1 (en) 1985-03-20
GR76963B (da) 1984-09-04
DK158228B (da) 1990-04-16
YU288181A (en) 1983-12-31
PH17469A (en) 1984-08-29
ES8302717A1 (es) 1983-01-16
IE52111B1 (en) 1987-06-24
PT74111B (en) 1983-12-19
ZA818579B (en) 1982-11-24
NO160517C (no) 1989-04-26
FI813956L (fi) 1982-06-12
KR830007672A (ko) 1983-11-04
NO160517B (no) 1989-01-16
IL64497A0 (en) 1982-03-31
IE812899L (en) 1982-06-11
FI75824C (fi) 1988-08-08
DK158228C (da) 1990-09-24
CA1177068A (en) 1984-10-30
PT74111A (en) 1982-01-01
AU7844681A (en) 1982-06-17
AU527159B2 (en) 1983-02-17
FI75824B (fi) 1988-04-29
AR229599A1 (es) 1983-09-30
DE3169462D1 (en) 1985-04-25
YU43053B (en) 1989-02-28
US4361513A (en) 1982-11-30
JPS57122089A (en) 1982-07-29
ES507867A0 (es) 1983-01-16
KR850001340B1 (ko) 1985-09-19
JPS6251959B2 (da) 1987-11-02
ATE12233T1 (de) 1985-04-15
NO814226L (no) 1982-06-14
EP0054397A1 (en) 1982-06-23

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