DK553986D0 - Cykliske peptider, fremgangsmaade til fremstilling heraf samt deres anvendelse som vasopressinantagonister - Google Patents

Cykliske peptider, fremgangsmaade til fremstilling heraf samt deres anvendelse som vasopressinantagonister

Info

Publication number
DK553986D0
DK553986D0 DK553986A DK553986A DK553986D0 DK 553986 D0 DK553986 D0 DK 553986D0 DK 553986 A DK553986 A DK 553986A DK 553986 A DK553986 A DK 553986A DK 553986 D0 DK553986 D0 DK 553986D0
Authority
DK
Denmark
Prior art keywords
preparing
cyclic peptides
vasopressin antagonists
vasopressin
antagonists
Prior art date
Application number
DK553986A
Other languages
English (en)
Other versions
DK553986A (da
Inventor
Fadia Elfehail Ali
William Francis Huffman
Ross Marshall Garland
Michael Lee Moore
Original Assignee
Smithkline Beckman Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Smithkline Beckman Corp filed Critical Smithkline Beckman Corp
Publication of DK553986D0 publication Critical patent/DK553986D0/da
Publication of DK553986A publication Critical patent/DK553986A/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04—Linear peptides containing only normal peptide links
    • C07K7/16—Oxytocins; Vasopressins; Related peptides
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10—TECHNICAL SUBJECTS COVERED BY FORMER USPC
    • Y10S—TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y10S930/00—Peptide or protein sequence
    • Y10S930/01—Peptide or protein sequence
    • Y10S930/15—Oxytocin or vasopressin; related peptides

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biophysics (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Diabetes (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
DK553986A 1985-11-19 1986-11-19 Cykliske peptider, fremgangsmaade til fremstilling heraf samt deres anvendelse som vasopressinantagonister DK553986A (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/799,718 US4687758A (en) 1985-11-19 1985-11-19 Des-proline-N-methylarginine vasopressins

Publications (2)

Publication Number Publication Date
DK553986D0 true DK553986D0 (da) 1986-11-19
DK553986A DK553986A (da) 1987-05-20

Family

ID=25176592

Family Applications (1)

Application Number Title Priority Date Filing Date
DK553986A DK553986A (da) 1985-11-19 1986-11-19 Cykliske peptider, fremgangsmaade til fremstilling heraf samt deres anvendelse som vasopressinantagonister

Country Status (7)

Country Link
US (1) US4687758A (da)
EP (1) EP0225109A3 (da)
JP (1) JPS62155298A (da)
AU (1) AU595258B2 (da)
DK (1) DK553986A (da)
PT (1) PT83760B (da)
ZA (1) ZA868690B (da)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA2027936C (en) 1989-10-23 2001-07-24 Smithkline Beecham Corporation Cyclic anti-aggregatory peptides
JP2003335797A (ja) * 2000-06-28 2003-11-28 Daicel Chem Ind Ltd ペプチド化合物及びそれを有効成分とする医薬組成物

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4469679A (en) * 1983-02-16 1984-09-04 Smithkline Beckman Corporation Octapeptide vasopressin antagonists
CA1238314A (en) * 1983-09-22 1988-06-21 James F. Callahan Process for preparing basic heptapeptide vasopressin antagonists
US4543349A (en) * 1983-09-22 1985-09-24 Smithkline Beckman Corporation Basic heptapeptide vasopressin antagonists
US4551445A (en) * 1983-10-14 1985-11-05 The Medical College Of Ohio Derivatives of arginine vasopressin antagonists
US4481194A (en) * 1984-03-07 1984-11-06 Smithkline Beckman Corporation Des-proline-des-glycine vasopressin antagonists
US4481193A (en) * 1984-03-07 1984-11-06 Smithkline Beckman Corporation Des-proline vasopressin antagonists
PH21037A (en) * 1984-03-07 1987-06-30 Smithkline Beckman Corp Des-proline vasopressin antagonists
US4604378A (en) * 1984-11-21 1986-08-05 Smithkline Beckman Corporation Basic V1 -vasopressin antagonists
US4599324A (en) * 1984-11-21 1986-07-08 Smithkline Beckman Corporation V1-vasopressin antagonists
NZ216417A (en) * 1985-06-18 1990-12-21 Smithkline Beckman Corp Vasopressin antagonists, preparation thereof and pharmaceutical compositions
PT84342B (pt) * 1986-02-25 1989-09-14 Smithkline Beecham Corp Processo de preparacao de compostos de vasopressina

Also Published As

Publication number Publication date
PT83760A (en) 1986-12-01
EP0225109A2 (en) 1987-06-10
AU6538386A (en) 1987-05-21
JPS62155298A (ja) 1987-07-10
PT83760B (en) 1988-12-07
ZA868690B (en) 1987-08-26
DK553986A (da) 1987-05-20
US4687758A (en) 1987-08-18
EP0225109A3 (en) 1989-06-07
AU595258B2 (en) 1990-03-29

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Legal Events

Date Code Title Description
AHB Application shelved due to non-payment