DK588785A - Imidazo(1,2-a)pyrimidiner og fremgangsmaade til deres fremstilling - Google Patents

Imidazo(1,2-a)pyrimidiner og fremgangsmaade til deres fremstilling Download PDF

Info

Publication number: DK588785A
Authority: DK; Denmark
Prior art keywords: carbon atoms; alkyl; group; oxadiazol; alkenyl
Prior art date: 1984-12-19

Application number

DK588785A

Other languages

English (en)

Other versions

DK588785D0 (da

Inventor

Roger John Gillespie

Wilfred Roger Tully

Original Assignee

Roussel Uclaf

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1984-12-19

Filing date

1985-12-18

Publication date

1986-06-20

1985-12-18 Application filed by Roussel Uclaf filed Critical Roussel Uclaf

1985-12-18 Publication of DK588785D0 publication Critical patent/DK588785D0/da

1986-06-20 Publication of DK588785A publication Critical patent/DK588785A/da

Links

238000000034 method Methods 0.000 title abstract 2
150000005238 imidazo[1,2-a]pyrimidines Chemical class 0.000 title 1
125000004432 carbon atom Chemical group C* 0.000 abstract 9
125000000217 alkyl group Chemical group 0.000 abstract 5
125000003342 alkenyl group Chemical group 0.000 abstract 3
125000001766 1,2,4-oxadiazol-3-yl group Chemical group [H]C1=NC(*)=NO1 0.000 abstract 1
125000004505 1,2,4-oxadiazol-5-yl group Chemical group O1N=CN=C1* 0.000 abstract 1
125000004509 1,3,4-oxadiazol-2-yl group Chemical group O1C(=NN=C1)* 0.000 abstract 1
125000004521 1,3,4-thiadiazol-2-yl group Chemical group S1C(=NN=C1)* 0.000 abstract 1
PXGOKWXKJXAPGV-UHFFFAOYSA-N Fluorine Chemical compound FF PXGOKWXKJXAPGV-UHFFFAOYSA-N 0.000 abstract 1
239000002253 acid Substances 0.000 abstract 1
125000002947 alkylene group Chemical group 0.000 abstract 1
239000002249 anxiolytic agent Substances 0.000 abstract 1
230000000949 anxiolytic effect Effects 0.000 abstract 1
150000001875 compounds Chemical class 0.000 abstract 1
229910052731 fluorine Inorganic materials 0.000 abstract 1
239000011737 fluorine Substances 0.000 abstract 1
229910052739 hydrogen Inorganic materials 0.000 abstract 1
239000001257 hydrogen Substances 0.000 abstract 1
125000004435 hydrogen atom Chemical class [H]* 0.000 abstract 1
230000000147 hypnotic effect Effects 0.000 abstract 1
239000000543 intermediate Substances 0.000 abstract 1
231100000252 nontoxic Toxicity 0.000 abstract 1
230000003000 nontoxic effect Effects 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
239000000932 sedative agent Substances 0.000 abstract 1
230000001624 sedative effect Effects 0.000 abstract 1

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/20—Hypnotics; Sedatives
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Bioinformatics & Cheminformatics (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Engineering & Computer Science (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Veterinary Medicine (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
Biomedical Technology (AREA)
Public Health (AREA)
Anesthesiology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)

DK588785A 1984-12-19 1985-12-18 Imidazo(1,2-a)pyrimidiner og fremgangsmaade til deres fremstilling DK588785A (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB848432073A GB8432073D0 (en)	1984-12-19	1984-12-19	Chemical compounds

Publications (2)

Publication Number	Publication Date
DK588785D0 DK588785D0 (da)	1985-12-18
DK588785A true DK588785A (da)	1986-06-20

Family

ID=10571440

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK588785A DK588785A (da)	1984-12-19	1985-12-18	Imidazo(1,2-a)pyrimidiner og fremgangsmaade til deres fremstilling

Country Status (16)

Country	Link
US (1)	US4703049A (da)
EP (1)	EP0197230B1 (da)
JP (1)	JPS61180786A (da)
AT (1)	ATE49971T1 (da)
AU (1)	AU581713B2 (da)
CA (1)	CA1248528A (da)
DE (1)	DE3575726D1 (da)
DK (1)	DK588785A (da)
ES (2)	ES8705432A1 (da)
FI (1)	FI82247C (da)
GB (2)	GB8432073D0 (da)
GR (1)	GR853021B (da)
HU (1)	HU193843B (da)
PT (1)	PT81693B (da)
SU (1)	SU1650013A3 (da)
ZA (1)	ZA859650B (da)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB8613591D0 (en) *	1986-06-04	1986-07-09	Roussel Lab Ltd	Chemical compounds
DK522187D0 (da) *	1987-10-06	1987-10-06	Ferrosan As	Imidozothienopyrimidiner, deres fremstilling og anvendelse
GB8905130D0 (en) *	1989-03-07	1989-04-19	Pfizer Ltd	Therapeutic agents
US5185446A (en) *	1990-09-04	1993-02-09	Neurogen Corporation	Certain cycloalkyl imidazopyrimidines; a new class of gaba brainreceptor ligands
US5646152A (en) *	1994-06-15	1997-07-08	Pfizer Inc.	Methods of administering CRF antagonists
WO2019155066A1 (en) *	2018-02-12	2019-08-15	Bayer Aktiengesellschaft	Fungicidal oxadiazoles

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
JPS57123180A (en) *	1980-12-17	1982-07-31	Schering Ag	3-substituted beta-carboline, manufacture and psychotropic drug containing same
IL69417A (en) *	1982-08-27	1987-12-20	Roussel Uclaf	2-acyl imidazo(1,2-a)pyrimidines,their preparation and pharmaceutical compositions containing them
GB8305245D0 (en) *	1983-02-25	1983-03-30	Fujisawa Pharmaceutical Co	Imidazo-heterocyclic compounds

1984
- 1984-12-19 GB GB848432073A patent/GB8432073D0/en active Pending
1985
- 1985-12-12 US US06/808,844 patent/US4703049A/en not_active Expired - Fee Related
- 1985-12-16 JP JP60281254A patent/JPS61180786A/ja active Pending
- 1985-12-16 GR GR853021A patent/GR853021B/el unknown
- 1985-12-17 PT PT81693A patent/PT81693B/pt not_active IP Right Cessation
- 1985-12-18 GB GB08531161A patent/GB2170199B/en not_active Expired
- 1985-12-18 SU SU854005003A patent/SU1650013A3/ru active
- 1985-12-18 ZA ZA859650A patent/ZA859650B/xx unknown
- 1985-12-18 ES ES550100A patent/ES8705432A1/es not_active Expired
- 1985-12-18 DK DK588785A patent/DK588785A/da not_active Application Discontinuation
- 1985-12-18 HU HU854857A patent/HU193843B/hu not_active IP Right Cessation
- 1985-12-18 FI FI855060A patent/FI82247C/fi not_active IP Right Cessation
- 1985-12-18 CA CA000498010A patent/CA1248528A/en not_active Expired
- 1985-12-19 AU AU51487/85A patent/AU581713B2/en not_active Ceased
- 1985-12-19 EP EP85402558A patent/EP0197230B1/fr not_active Expired - Lifetime
- 1985-12-19 DE DE8585402558T patent/DE3575726D1/de not_active Expired - Fee Related
- 1985-12-19 AT AT85402558T patent/ATE49971T1/de not_active IP Right Cessation
1987
- 1987-01-16 ES ES557324A patent/ES8900049A1/es not_active Expired

Also Published As

Publication number	Publication date
ES550100A0 (es)	1987-05-01
PT81693A (en)	1986-01-01
ES8705432A1 (es)	1987-05-01
JPS61180786A (ja)	1986-08-13
GR853021B (da)	1986-04-15
FI82247C (fi)	1991-02-11
HUT40437A (en)	1986-12-28
GB2170199A (en)	1986-07-30
DK588785D0 (da)	1985-12-18
FI855060A0 (fi)	1985-12-18
DE3575726D1 (de)	1990-03-08
US4703049A (en)	1987-10-27
ES557324A0 (es)	1988-11-16
AU5148785A (en)	1986-06-26
EP0197230B1 (fr)	1990-01-31
SU1650013A3 (ru)	1991-05-15
CA1248528A (en)	1989-01-10
GB8432073D0 (en)	1985-01-30
PT81693B (pt)	1988-02-17
GB8531161D0 (en)	1986-01-29
GB2170199B (en)	1988-03-16
AU581713B2 (en)	1989-03-02
HU193843B (en)	1987-12-28
EP0197230A1 (fr)	1986-10-15
ATE49971T1 (de)	1990-02-15
ZA859650B (en)	1987-02-25
FI855060A7 (fi)	1986-06-20
ES8900049A1 (es)	1988-11-16
FI82247B (fi)	1990-10-31

Legal Events

Date	Code	Title	Description
1992-08-24	AHB	Application shelved due to non-payment

Publication	Publication Date	Title
GB2191196B (en)	1990-03-28	Imidazo pyrimidines
DK588785D0 (da)	1985-12-18	Imidazo(1,2-a)pyrimidiner og fremgangsmaade til deres fremstilling
DK0383686T3 (da)	1993-12-20	Carboxyalkylethere af 2-amino-7-hydroxytetralin samt fremgangsmåde til fremstilling deraf
DK160308C (da)	1991-07-29	Analogifremgangsmaade til fremstilling af 1,2,4-triazolo(4,3-a)quinazolin-5-(4h)-oner eller deres syreadditionssalte
FI881582A0 (fi)	1988-04-06	Foerfarande foer framstaellning av 3h-1,2,3-triazolo (4,5-d) pyrimidiner.
ES538933A0 (es)	1986-03-16	Un procedimiento para preparar imidazo(1,2-c)pirimidinas
ES8501416A1 (es)	1984-11-16	5'-alquil o alquenil-fosfatos de nucleosidos.
NO167286C (no)	1991-10-23	Fremgangsmaate for fremstilling av terapeutisk aktive benzotiazepin-derivater.
SE9702306L (sv)	1997-08-25	Diklavulanatsalt med en diaminoeter och process av preparation
DK470888A (da)	1989-03-01	Imidazobenzodiazepinderivater, deres fresmtilling samt laegemidler med indholdd deraf
ES8800938A1 (es)	1987-12-16	Procedimiento para preparar derivados berbanicos biologicamente activos.
NZ217276A (en)	1988-10-28	Bicyclic heterocyclic compounds and pharmaceutical compositions
GR852568B (da)	1986-02-21
ES500108A0 (es)	1982-06-01	Procedimiento para preparar nuevas benzotiopirano (2,3-c)pi-ridinas