DK662787A - Anvendelse af en 5-ht-receptorantagonist - Google Patents

Anvendelse af en 5-ht-receptorantagonist

Info

Publication number: DK662787A
Authority: DK; Denmark
Prior art keywords: anagonist; receptor; methyl; carbazol; imidazol
Prior art date: 1986-12-17

Application number

DK662787A

Other languages

English (en)

Other versions

DK662787D0 (da

Inventor

Michael Brian Tyers

Original Assignee

Glaxo Group Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1986-12-17

Filing date

1987-12-16

Publication date

1988-06-18

1987-12-16 Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd

1987-12-16 Publication of DK662787D0 publication Critical patent/DK662787D0/da

1988-06-18 Publication of DK662787A publication Critical patent/DK662787A/da

Links

108091032151 5-hydroxytryptamine receptor family Proteins 0.000 title 1
102000014630 G protein-coupled serotonin receptor activity proteins Human genes 0.000 title 1
-1 2-methyl-1H-imidazol-1-yl Chemical group 0.000 abstract 1
208000020401 Depressive disease Diseases 0.000 abstract 1
125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 abstract 1
150000003839 salts Chemical class 0.000 abstract 1
239000012453 solvate Substances 0.000 abstract 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/415—1,2-Diazoles
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/26—Psychostimulants, e.g. nicotine, cocaine

Landscapes

Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Life Sciences & Earth Sciences (AREA)
Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Epidemiology (AREA)
Neurosurgery (AREA)
Psychiatry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Neurology (AREA)
Biomedical Technology (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
General Chemical & Material Sciences (AREA)
Pain & Pain Management (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Plural Heterocyclic Compounds (AREA)
Connection Of Batteries Or Terminals (AREA)
Emergency Protection Circuit Devices (AREA)
Electrotherapy Devices (AREA)
Saccharide Compounds (AREA)

DK662787A 1986-12-17 1987-12-16 Anvendelse af en 5-ht-receptorantagonist DK662787A (da)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
GB868630071A GB8630071D0 (en)	1986-12-17	1986-12-17	Medicaments

Publications (2)

Publication Number	Publication Date
DK662787D0 DK662787D0 (da)	1987-12-16
DK662787A true DK662787A (da)	1988-06-18

Family

ID=10609112

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK662787A DK662787A (da)	1986-12-17	1987-12-16	Anvendelse af en 5-ht-receptorantagonist

Country Status (18)

Country	Link
US (1)	US4835173A (da)
EP (1)	EP0276559B1 (da)
JP (1)	JP2732844B2 (da)
KR (1)	KR880007073A (da)
AT (1)	ATE79031T1 (da)
AU (1)	AU608794B2 (da)
CY (1)	CY1693A (da)
DE (1)	DE3780940T2 (da)
DK (1)	DK662787A (da)
ES (1)	ES2051754T3 (da)
GB (1)	GB8630071D0 (da)
GR (1)	GR3005682T3 (da)
HK (1)	HK36593A (da)
IE (1)	IE60135B1 (da)
IL (1)	IL84844A0 (da)
NZ (1)	NZ222949A (da)
PH (1)	PH25503A (da)
ZA (1)	ZA879458B (da)

Families Citing this family (18)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5246941A (en) *	1986-12-17	1993-09-21	Glaxo Group Limited	Method for the treatment of depression
US4973594A (en) *	1986-12-17	1990-11-27	Glaxo Group Limited	Medicaments
US5221687A (en) *	1988-09-01	1993-06-22	Glaxo Group Limited	Medicaments
GB8820653D0 (en) *	1988-09-01	1988-10-05	Glaxo Group Ltd	Medicaments
US5180728A (en) *	1989-09-25	1993-01-19	Fujisawa Pharmaceutical Company, Ltd.	Pyrimidoindole derivatives and processes for preparation thereof
US5225407A (en) *	1990-02-22	1993-07-06	Glaxo Group Limited	5-HT3 receptor antagonists for the treatment of autism
WO1993000074A1 (en) *	1991-06-26	1993-01-07	Sepracor, Inc.	Method and compositions for treating emesis, nausea and other disorders using optically pure r(+) ondansetron
WO2000051582A2 (en) *	1999-03-01	2000-09-08	Sepracor Inc.	Methods for treating apnea and apnea disorders using optically pure r(+)ondansetron
EP1339707A2 (en) *	2000-10-30	2003-09-03	Teva Pharmaceutical Industries Ltd.	Novel crystal and solvate forms of ondansetron hydrochloride and processes for their preparation
EP1207160A1 (en) *	2000-11-20	2002-05-22	Hanmi Pharm. Co., Ltd.	Process for the preparation of 1,2,3,9-tetrahydro-9-methyl-3-((2-methyl-1H-imidazol-1-yl)-methyl)-4H-carbazol-4-one
US20020115707A1 (en) *	2001-01-11	2002-08-22	Rami Lidor-Hadas	Process for preparing pure ondansetron hydrochloride dihydrate
EP1355881A4 (en) *	2001-01-11	2004-03-31	Teva Pharma	IMPROVED METHOD FOR PRODUCING PURE ONDANSETRONHYDROCHLORIDE DIHYDRATE
PT1499623E (pt) *	2002-04-29	2007-08-10	Teva Gyogyszergyar Zartkoeruee	''processo papa a preparação de 1, 2, 3, 9-tetra-hidro-9-metil-3- [(2-metil-1h-imidazol-1-il) metil] -4h-carbazol-4-ona''
US20050131045A1 (en) *	2002-04-30	2005-06-16	Judith Aronhime	Novel crystal forms of ondansetron, processes for their preparation, pharmaceutical, compositions containing the novel forms and methods for treating nausea using them
MXPA04010845A (es) *	2002-04-30	2005-01-25	Biogal Gyogyszergyar	Formas cristalinas novedosas de ondansetron, procesos para su preparacion, composiciones farmaceuticas que contienen las formas novedosas y metodos para tratar las nauseas utilizando las mismas.
HU225885B1 (en) *	2002-10-17	2007-11-28	Richter Gedeon Nyrt	Process for producing ondansetron hydrochlorid dihydrate of high purity
EP2186517A4 (en) *	2007-08-08	2010-08-18	Ibanez Juan Jose Legarda	USE AND METHODS OF USING A SEROTONIN3 (5-HT3) RECEPTOR ANTAGONIST AND CHLORIDE CHANNEL MODULATOR FOR THE TREATMENT OF DRUG OR DRUG ADDICTION OR DEPENDENCE OR CENTER NERVOUS DISORDERS
EP3810120A2 (en)	2018-06-21	2021-04-28	Société des Produits Nestlé S.A.	Compositions and methods using a nicotinamide adenine dinucleotide (nad+) precursor and at least one ketone or ketone precursor

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
IN158970B (da) *	1981-06-09	1987-02-28	Ici Plc
LU88268I2 (da) *	1984-01-25	1994-02-03
GB8401888D0 (en) *	1984-01-25	1984-02-29	Glaxo Group Ltd	Heterocyclic compounds
DE201165T1 (de) *	1985-03-14	1989-04-20	Beecham Group P.L.C., Brentford	Arzneimittel zur behandlung von emesis, anxietas und "irritable bowel syndrome".
GB8516083D0 (en) *	1985-06-25	1985-07-31	Glaxo Group Ltd	Heterocyclic compounds
GB8518743D0 (en) *	1985-07-24	1985-08-29	Glaxo Group Ltd	Heterocyclic compounds
HU895334D0 (en) *	1986-07-30	1990-01-28	Sandoz Ag	Process for the preparation of nasal pharmaceutical compositions

1986
- 1986-12-17 GB GB868630071A patent/GB8630071D0/en active Pending
1987
- 1987-12-16 ES ES87311082T patent/ES2051754T3/es not_active Expired - Lifetime
- 1987-12-16 AT AT87311082T patent/ATE79031T1/de not_active IP Right Cessation
- 1987-12-16 AU AU82617/87A patent/AU608794B2/en not_active Ceased
- 1987-12-16 DE DE8787311082T patent/DE3780940T2/de not_active Expired - Lifetime
- 1987-12-16 NZ NZ222949A patent/NZ222949A/en unknown
- 1987-12-16 PH PH36241A patent/PH25503A/en unknown
- 1987-12-16 IL IL84844A patent/IL84844A0/xx not_active IP Right Cessation
- 1987-12-16 EP EP87311082A patent/EP0276559B1/en not_active Expired - Lifetime
- 1987-12-16 DK DK662787A patent/DK662787A/da not_active Application Discontinuation
- 1987-12-16 US US07/133,887 patent/US4835173A/en not_active Expired - Lifetime
- 1987-12-16 IE IE341587A patent/IE60135B1/en not_active IP Right Cessation
- 1987-12-16 JP JP62318455A patent/JP2732844B2/ja not_active Expired - Lifetime
- 1987-12-17 KR KR870014390A patent/KR880007073A/ko not_active Ceased
- 1987-12-17 ZA ZA879458A patent/ZA879458B/xx unknown
1992
- 1992-09-10 GR GR920402010T patent/GR3005682T3/el unknown
1993
- 1993-04-15 HK HK365/93A patent/HK36593A/en not_active IP Right Cessation
1994
- 1994-01-14 CY CY169394A patent/CY1693A/xx unknown

Also Published As

Publication number	Publication date
PH25503A (en)	1991-07-24
KR880007073A (ko)	1988-08-26
DE3780940D1 (de)	1992-09-10
HK36593A (en)	1993-04-23
ZA879458B (en)	1988-11-30
CY1693A (en)	1994-01-14
US4835173A (en)	1989-05-30
IE873415L (en)	1988-06-17
JP2732844B2 (ja)	1998-03-30
IE60135B1 (en)	1994-06-01
EP0276559A3 (en)	1989-10-18
DK662787D0 (da)	1987-12-16
IL84844A0 (en)	1988-06-30
EP0276559B1 (en)	1992-08-05
EP0276559A2 (en)	1988-08-03
ATE79031T1 (de)	1992-08-15
GR3005682T3 (da)	1993-06-07
GB8630071D0 (en)	1987-01-28
NZ222949A (en)	1997-06-24
AU8261787A (en)	1988-06-23
AU608794B2 (en)	1991-04-18
ES2051754T3 (es)	1994-07-01
JPS63165314A (ja)	1988-07-08
DE3780940T2 (de)	1992-12-24

Legal Events

Date	Code	Title	Description
2004-12-27	AHS	Application shelved for other reasons than non-payment

Publication	Publication Date	Title
DK662787D0 (da)	1987-12-16	Anvendelse af en 5-ht-receptorantagonist
ITFI910071U1 (it)	1992-12-25	Piastra per osso per la porzione distale dell'omero.
FR2658414B1 (fr)	1992-07-31	Implant pour dispositif d'osteosynthese en particulier du rachis.
ES2079620T3 (es)	1996-01-16	Protesis femoral parcialmente cimentada.
FR2658413B1 (fr)	1997-01-03	Dispositif d'osteosynthese pour la correction des deviations rachidiennes.
FR2599970B1 (fr)	1989-10-06	Composition tinctoriale pour fibres keratiniques humaines sous forme de mousse, a base de 5,6-dihydroxyindole.
FR2670669B1 (fr)	1993-03-12	Instrument de correction chirurgicale de l'astigmatisme.
DE69107329D1 (de)	1995-03-23	Zahnärztliches Handstück.
DK612787D0 (da)	1987-11-20	Anvendelse af imidazolderivater
IT1238825B (it)	1993-09-03	Dispositivo per la correzione chirurgica dell'ametropia.
GR3003327T3 (en)	1993-02-17	Substituted 1,8-naphthyridine derivatives and fungicides containing them
IT8919074A0 (it)	1989-01-12	Composizione per l'igiene orale.
ITBO910103U1 (it)	1992-11-24	Dispositivo per realizzare attacchi rapidi per protesi dentarie.
ATE219083T1 (de)	2002-06-15	4-oxo-und 4h-imidazo(5,1-c)(1,4)benzoxazine nützlich als benzodiazepinrezeptor-bindemittel.
DE69223362D1 (de)	1998-01-15	N1-Trifluoralkyl substituierte 2-Nitro-p-Phenylendiaminfarbstoffe
FR2666979B3 (fr)	1995-10-06	Dispositif pour deposer des couronnes, protheses ou bridges dentaires.
FR2665074B1 (fr)	1994-08-12	Appareil d'orthopedie.
FR2670665B1 (fr)	1997-12-19	Moyen d'ancrage radiculaire pour prothese dentaire.
FR2674435B1 (fr)	1995-03-10	Utilisation de 4-amino-1-(2-pyridyl) piperidines pour la preparation d'agents psychotropes.
IT1192045B (it)	1988-03-31	Articolatore d'anca per protesi ortopediche
IT1217080B (it)	1990-03-14	Acetabolo perfezionato per protesi d'anca.
IT8821443A0 (it)	1988-07-21	Cotile per protesi d'anca.
FR2651673B1 (fr)	1994-06-17	Positionneur prothetique pour l'art dentaire.
IT206741Z2 (it)	1987-10-01	Bastoncino per l'igiene del canale uditivo.
IT1238934B (it)	1993-09-07	Attacco per protesi dentale rimovibile, con ritenzione regolabile