DOP2002000405A - 1-BIARIL-1,8-NAFTIRIDIN-4-ONA PHOSPHODISTERASE-4 INHIBITORS. - Google Patents
1-BIARIL-1,8-NAFTIRIDIN-4-ONA PHOSPHODISTERASE-4 INHIBITORS.Info
- Publication number
- DOP2002000405A DOP2002000405A DO2002000405A DO2002000405A DOP2002000405A DO P2002000405 A DOP2002000405 A DO P2002000405A DO 2002000405 A DO2002000405 A DO 2002000405A DO 2002000405 A DO2002000405 A DO 2002000405A DO P2002000405 A DOP2002000405 A DO P2002000405A
- Authority
- DO
- Dominican Republic
- Prior art keywords
- inhibitors
- phosphodisterase
- biaril
- naftiridin
- ona
- Prior art date
Links
- 239000003112 inhibitor Substances 0.000 title abstract 2
- MSYGAHOHLUJIKV-UHFFFAOYSA-N 3,5-dimethyl-1-(3-nitrophenyl)-1h-pyrazole-4-carboxylic acid ethyl ester Chemical compound CC1=C(C(=O)OCC)C(C)=NN1C1=CC=CC([N+]([O-])=O)=C1 MSYGAHOHLUJIKV-UHFFFAOYSA-N 0.000 abstract 1
- 206010061218 Inflammation Diseases 0.000 abstract 1
- 102000011017 Type 4 Cyclic Nucleotide Phosphodiesterases Human genes 0.000 abstract 1
- 108010037584 Type 4 Cyclic Nucleotide Phosphodiesterases Proteins 0.000 abstract 1
- 208000006673 asthma Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000004054 inflammatory process Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Los compuestos representados por la Fórmula (I): o una sal farmacéuticamente aceptable de los mismos, son inhibidores útiles de la fosfodiesterasa 4 en el tratamiento del asma y la inflamación.The compounds represented by Formula (I): or a pharmaceutically acceptable salt thereof, are useful inhibitors of phosphodiesterase 4 in the treatment of asthma and inflammation.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DO2002000405A DOP2002000405A (en) | 2002-05-24 | 2002-05-24 | 1-BIARIL-1,8-NAFTIRIDIN-4-ONA PHOSPHODISTERASE-4 INHIBITORS. |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DO2002000405A DOP2002000405A (en) | 2002-05-24 | 2002-05-24 | 1-BIARIL-1,8-NAFTIRIDIN-4-ONA PHOSPHODISTERASE-4 INHIBITORS. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DOP2002000405A true DOP2002000405A (en) | 2002-11-30 |
Family
ID=44261079
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DO2002000405A DOP2002000405A (en) | 2002-05-24 | 2002-05-24 | 1-BIARIL-1,8-NAFTIRIDIN-4-ONA PHOSPHODISTERASE-4 INHIBITORS. |
Country Status (1)
| Country | Link |
|---|---|
| DO (1) | DOP2002000405A (en) |
-
2002
- 2002-05-24 DO DO2002000405A patent/DOP2002000405A/en unknown
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