DOP2002000419A - SELF-EMULSIONING FORMULATIONS OF INHIBITORS OF THE ESTER CHOLESTERILE TRANSFER PROTECTION. - Google Patents
SELF-EMULSIONING FORMULATIONS OF INHIBITORS OF THE ESTER CHOLESTERILE TRANSFER PROTECTION.Info
- Publication number
- DOP2002000419A DOP2002000419A DO2002000419A DO2002000419A DOP2002000419A DO P2002000419 A DOP2002000419 A DO P2002000419A DO 2002000419 A DO2002000419 A DO 2002000419A DO 2002000419 A DO2002000419 A DO 2002000419A DO P2002000419 A DOP2002000419 A DO P2002000419A
- Authority
- DO
- Dominican Republic
- Prior art keywords
- self
- inhibitors
- cholesterile
- emulsioning
- formulations
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 2
- 239000003112 inhibitor Substances 0.000 title 1
- 239000004094 surface-active agent Substances 0.000 abstract 3
- 239000003354 cholesterol ester transfer protein inhibitor Substances 0.000 abstract 2
- 229940125881 cholesteryl ester transfer protein inhibitor Drugs 0.000 abstract 1
- 239000006184 cosolvent Substances 0.000 abstract 1
- 239000002904 solvent Substances 0.000 abstract 1
Landscapes
- Medicinal Preparation (AREA)
Abstract
Inhibidores de CETP que tienen mejor solubilidad y biodisponibilidad en un vehículo lipófilo que comprende un aceite digerible, un disolvente lipófilo o un tensioactivo. Tales composiciones preferidas son autoemulsionantes o automicroemulsionantes y comprenden 1. un inhibidor de CETP; 2. un codisolvente; 3. un tensioactivo que tiene un HLB de 1 a 8; 4. un tensioactivo que tiene un HLB de 8 a 20; y 5. opcionalmente, un aceite digerible.CETP inhibitors that have better solubility and bioavailability in a lipophilic vehicle comprising a digestible oil, a lipophilic solvent or a surfactant. Such preferred compositions are self-emulsifying or self-emulsifying and comprise 1. a CETP inhibitor; 2. a co-solvent; 3. a surfactant having an HLB of 1 to 8; 4. a surfactant having an HLB of 8 to 20; and 5. optionally, a digestible oil.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DO2002000419A DOP2002000419A (en) | 2002-06-18 | 2002-06-18 | SELF-EMULSIONING FORMULATIONS OF INHIBITORS OF THE ESTER CHOLESTERILE TRANSFER PROTECTION. |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DO2002000419A DOP2002000419A (en) | 2002-06-18 | 2002-06-18 | SELF-EMULSIONING FORMULATIONS OF INHIBITORS OF THE ESTER CHOLESTERILE TRANSFER PROTECTION. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DOP2002000419A true DOP2002000419A (en) | 2003-01-15 |
Family
ID=44261084
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DO2002000419A DOP2002000419A (en) | 2002-06-18 | 2002-06-18 | SELF-EMULSIONING FORMULATIONS OF INHIBITORS OF THE ESTER CHOLESTERILE TRANSFER PROTECTION. |
Country Status (1)
| Country | Link |
|---|---|
| DO (1) | DOP2002000419A (en) |
-
2002
- 2002-06-18 DO DO2002000419A patent/DOP2002000419A/en unknown
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