DOP2004000893A - PDE9 INHIBITORS TO TREAT TYPE 2 DIABETES, METABOLIC SYNDROME AND CARDIOVASCULAR DISEASES - Google Patents
PDE9 INHIBITORS TO TREAT TYPE 2 DIABETES, METABOLIC SYNDROME AND CARDIOVASCULAR DISEASESInfo
- Publication number
- DOP2004000893A DOP2004000893A DO2004000893A DO2004000893A DOP2004000893A DO P2004000893 A DOP2004000893 A DO P2004000893A DO 2004000893 A DO2004000893 A DO 2004000893A DO 2004000893 A DO2004000893 A DO 2004000893A DO P2004000893 A DOP2004000893 A DO P2004000893A
- Authority
- DO
- Dominican Republic
- Prior art keywords
- diabetes
- metabolic syndrome
- cardiovascular diseases
- treat type
- pde9 inhibitors
- Prior art date
Links
- 208000024172 Cardiovascular disease Diseases 0.000 title abstract 2
- 208000001145 Metabolic Syndrome Diseases 0.000 title abstract 2
- 201000000690 abdominal obesity-metabolic syndrome Diseases 0.000 title abstract 2
- 208000001072 type 2 diabetes mellitus Diseases 0.000 title abstract 2
- 229940076380 PDE9 inhibitor Drugs 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000008194 pharmaceutical composition Substances 0.000 abstract 2
- 239000000651 prodrug Substances 0.000 abstract 2
- 229940002612 prodrug Drugs 0.000 abstract 2
- 208000032928 Dyslipidaemia Diseases 0.000 abstract 1
- 208000002705 Glucose Intolerance Diseases 0.000 abstract 1
- 208000017170 Lipid metabolism disease Diseases 0.000 abstract 1
- 206010067584 Type 1 diabetes mellitus Diseases 0.000 abstract 1
- 206010012601 diabetes mellitus Diseases 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 201000001421 hyperglycemia Diseases 0.000 abstract 1
- 201000009104 prediabetes syndrome Diseases 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
La invencion proporciona los compuestos de formula (I) los estereoisomeros y los profarmacos de los mismos, y las sales de los compuestos, estereoisomeros, y profarmacos farmaceuticamente aceptables, en la que A, P, J, x y R10 son como se han definido en esta memoria descriptiva; las composiciones farmaceuticas de los mismos; y los procedimientos de use de las composiciones farmaceuticas para el tratamiento de enfermedades, incluyendo diabetes, que incluye diabetes tipo 1 y tipo 2, hiperglucemia, dislipidemia, tolerancia a la glucosa alterada, sindrome metabolico, y/o enfermedad cardiovascular.The invention provides the compounds of formula (I) the stereoisomers and the prodrugs thereof, and the salts of the pharmaceutically acceptable compounds, stereoisomers, and prodrugs, wherein A, P, J, x and R10 are as defined in this descriptive report; the pharmaceutical compositions thereof; and the methods of using the pharmaceutical compositions for the treatment of diseases, including diabetes, which includes type 1 and type 2 diabetes, hyperglycemia, dyslipidemia, impaired glucose tolerance, metabolic syndrome, and / or cardiovascular disease.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DO2004000893A DOP2004000893A (en) | 2004-04-29 | 2004-04-29 | PDE9 INHIBITORS TO TREAT TYPE 2 DIABETES, METABOLIC SYNDROME AND CARDIOVASCULAR DISEASES |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DO2004000893A DOP2004000893A (en) | 2004-04-29 | 2004-04-29 | PDE9 INHIBITORS TO TREAT TYPE 2 DIABETES, METABOLIC SYNDROME AND CARDIOVASCULAR DISEASES |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DOP2004000893A true DOP2004000893A (en) | 2004-11-30 |
Family
ID=44261350
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DO2004000893A DOP2004000893A (en) | 2004-04-29 | 2004-04-29 | PDE9 INHIBITORS TO TREAT TYPE 2 DIABETES, METABOLIC SYNDROME AND CARDIOVASCULAR DISEASES |
Country Status (1)
| Country | Link |
|---|---|
| DO (1) | DOP2004000893A (en) |
-
2004
- 2004-04-29 DO DO2004000893A patent/DOP2004000893A/en unknown
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