DOP2023000246A - Terapias de combinación - Google Patents

Terapias de combinación

Info

Publication number
DOP2023000246A
DOP2023000246A DO2023000246A DO2023000246A DOP2023000246A DO P2023000246 A DOP2023000246 A DO P2023000246A DO 2023000246 A DO2023000246 A DO 2023000246A DO 2023000246 A DO2023000246 A DO 2023000246A DO P2023000246 A DOP2023000246 A DO P2023000246A
Authority
DO
Dominican Republic
Prior art keywords
effective amount
combinations
formula
combination therapies
therapeutically effective
Prior art date
Application number
DO2023000246A
Other languages
English (en)
Spanish (es)
Inventor
Xu Yanping
Pande Vineet
Fu Liqiang
Li Ming
Fang Lichao
Freddy J Darville Nicolas
Alexis Georges Querolle Olivier
Tee Fuay Ng Alicia
Philippar Ulrike
Daskalakis Nikki
Diane Guttke Christina
Chul Kwon Min
Elizabeth Packman Kathryn
Christine Pietsch Eva
Bhogal Balpreet
Dai Xuedong
Cai Wei
Liu Yingtao
Liu Lianzhu
Deng Xiangjun
Angela Ferrante Lucille
Sun Yu
Ann J Verhulst Tinne
Wilhelmus J Thuring Johannes
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of DOP2023000246A publication Critical patent/DOP2023000246A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/53Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with three nitrogens as the only ring hetero atoms, e.g. chlorazanil, melamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4965Non-condensed pyrazines
    • A61K31/497Non-condensed pyrazines containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/63Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide
    • A61K31/635Compounds containing para-N-benzenesulfonyl-N-groups, e.g. sulfanilamide, p-nitrobenzenesulfonyl hydrazide having a heterocyclic ring, e.g. sulfadiazine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7052Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
    • A61K31/706Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides containing six-membered rings with nitrogen as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2300/00Mixtures or combinations of active ingredients, wherein at least one active ingredient is fully defined in groups A61K31/00 - A61K41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
DO2023000246A 2021-05-11 2023-11-08 Terapias de combinación DOP2023000246A (es)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
CN2021093036 2021-05-11
CN2021100523 2021-06-17
CN2022086004 2022-04-11
PCT/CN2022/091679 WO2022237720A1 (fr) 2021-05-11 2022-05-09 Multithérapies

Publications (1)

Publication Number Publication Date
DOP2023000246A true DOP2023000246A (es) 2024-04-30

Family

ID=81753154

Family Applications (1)

Application Number Title Priority Date Filing Date
DO2023000246A DOP2023000246A (es) 2021-05-11 2023-11-08 Terapias de combinación

Country Status (16)

Country Link
EP (1) EP4337216A1 (fr)
JP (1) JP2024518497A (fr)
KR (1) KR20240006631A (fr)
CN (2) CN117460513A (fr)
AU (1) AU2022274071A1 (fr)
CA (1) CA3215313A1 (fr)
CL (2) CL2023003239A1 (fr)
CO (1) CO2023014322A2 (fr)
DO (1) DOP2023000246A (fr)
IL (1) IL308335A (fr)
MX (1) MX2023013410A (fr)
PE (1) PE20240593A1 (fr)
PH (1) PH12023552974A1 (fr)
TW (1) TW202308643A (fr)
UY (1) UY39761A (fr)
WO (1) WO2022237720A1 (fr)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TW202525813A (zh) 2019-12-19 2025-07-01 比利時商健生藥品公司 經取代之直鏈螺環接衍生物
EP4626426A1 (fr) * 2022-11-30 2025-10-08 JANSSEN Pharmaceutica NV Associations comprenant un inhibiteur de ménine-mll et au moins un autre agent thérapeutique
WO2024114666A1 (fr) * 2022-11-30 2024-06-06 Janssen Pharmaceutica Nv Combinaisons comprenant un inhibiteur de ménine-mll et un inhibiteur de bcl-2
EP4698182A1 (fr) * 2023-04-17 2026-02-25 Janssen Pharmaceutica NV Combinaison d'un inhibiteur ménine-ll1, d'un agent intercalant de l'adn et d'un analogue de pyrimidine pour traiter un trouble hématopoïétique
WO2025082444A2 (fr) * 2023-10-20 2025-04-24 Janssen Pharmaceutica Nv (r)-n-éthyl-5-fluoro-n-isopropyl-2-((5-(2-(6-((2-méthoxyéthyl)(méthyl)amino)-2-méthylhexan-3-yl)-2, 6-diazaspiro[3,4]octan-6-yl)-1, 2, 4-triazin-6-yl)oxy)benzamide, formulations et schémas posologiques de celui-ci, destinés à être utilisés pour le traitement du cancer

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
TN2017000080A1 (en) 2014-12-18 2018-07-04 Takeda Pharmaceuticals Co Solid state forms of fused heteroaromatic pyrrolidinones
AU2016378579A1 (en) * 2015-12-22 2018-06-14 Vitae Pharmaceuticals, Inc. Inhibitors of the menin-MLL interaction
WO2017214367A1 (fr) * 2016-06-10 2017-12-14 Vitae Pharmaceuticals, Inc. Inhibiteurs de l'interaction ménine-mll
TW202104207A (zh) 2019-04-17 2021-02-01 美商健生生物科技公司 二氫乳清酸脫氫酶抑制劑
TW202525813A (zh) 2019-12-19 2025-07-01 比利時商健生藥品公司 經取代之直鏈螺環接衍生物

Also Published As

Publication number Publication date
AU2022274071A1 (en) 2024-01-04
MX2023013410A (es) 2023-12-06
JP2024518497A (ja) 2024-05-01
CO2023014322A2 (es) 2023-11-20
IL308335A (en) 2024-01-01
CL2024002832A1 (es) 2025-02-14
CA3215313A1 (fr) 2022-11-17
PH12023552974A1 (en) 2024-03-11
CL2023003239A1 (es) 2024-06-07
PE20240593A1 (es) 2024-03-21
TW202308643A (zh) 2023-03-01
CN118845787A (zh) 2024-10-29
UY39761A (es) 2022-11-30
CN117460513A (zh) 2024-01-26
EP4337216A1 (fr) 2024-03-20
WO2022237720A1 (fr) 2022-11-17
KR20240006631A (ko) 2024-01-15

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