ECSP003476A - SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRIMIDINONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL - Google Patents
SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRIMIDINONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALLInfo
- Publication number
- ECSP003476A ECSP003476A ECSP003476A ECSP003476A EC SP003476 A ECSP003476 A EC SP003476A EC SP003476 A ECSP003476 A EC SP003476A EC SP003476 A ECSP003476 A EC SP003476A
- Authority
- EC
- Ecuador
- Prior art keywords
- useful
- pirimidinones
- heteroaril
- substituted
- selective inhibition
- Prior art date
Links
- 230000015271 coagulation Effects 0.000 title abstract 2
- 238000005345 coagulation Methods 0.000 title abstract 2
- 230000005764 inhibitory process Effects 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 2
- 102000012479 Serine Proteases Human genes 0.000 abstract 1
- 108010022999 Serine Proteases Proteins 0.000 abstract 1
- 239000003146 anticoagulant agent Substances 0.000 abstract 1
- 229940127219 anticoagulant drug Drugs 0.000 abstract 1
- 208000026106 cerebrovascular disease Diseases 0.000 abstract 1
- 208000029078 coronary artery disease Diseases 0.000 abstract 1
- 210000004351 coronary vessel Anatomy 0.000 abstract 1
- -1 heteroaryl pyrimidinones Chemical class 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 238000002560 therapeutic procedure Methods 0.000 abstract 1
- 230000001732 thrombotic effect Effects 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
El invento se relaciona con los compuestos sustitutos del arilo policíclico y pirimidinonas heteroarilos útiles como inhibidores de las proteasas de serina de la cascada de coagulación y compuestos, composiciones y métodos utilizados para terapias anticuagulantes para el tratamiento y prevención de una variedad de condiciones trombóticas, incluyendo la arteria coronaria y enfermedades cerebrovasculares.The invention relates to polycyclic aryl and heteroaryl pyrimidinones substitute compounds useful as inhibitors of coagulation cascade serine proteases and compounds, compositions and methods used for anticoagulant therapies for the treatment and prevention of a variety of thrombotic conditions, including coronary artery and cerebrovascular diseases.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003476 ECSP003476A (en) | 2000-05-19 | 2000-05-19 | SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRIMIDINONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003476 ECSP003476A (en) | 2000-05-19 | 2000-05-19 | SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRIMIDINONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP003476A true ECSP003476A (en) | 2000-10-24 |
Family
ID=42041102
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP003476 ECSP003476A (en) | 2000-05-19 | 2000-05-19 | SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PIRIMIDINONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP003476A (en) |
-
2000
- 2000-05-19 EC ECSP003476 patent/ECSP003476A/en unknown
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