ECSP003477A - SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PYRIDONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL - Google Patents
SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PYRIDONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALLInfo
- Publication number
- ECSP003477A ECSP003477A ECSP003477A ECSP003477A EC SP003477 A ECSP003477 A EC SP003477A EC SP003477 A ECSP003477 A EC SP003477A EC SP003477 A ECSP003477 A EC SP003477A
- Authority
- EC
- Ecuador
- Prior art keywords
- heteroaril
- substituted
- selective inhibition
- pyridones
- polyclic
- Prior art date
Links
- 230000015271 coagulation Effects 0.000 title abstract 2
- 238000005345 coagulation Methods 0.000 title abstract 2
- 230000005764 inhibitory process Effects 0.000 title 1
- 239000003146 anticoagulant agent Substances 0.000 abstract 1
- 229940127219 anticoagulant drug Drugs 0.000 abstract 1
- 208000026106 cerebrovascular disease Diseases 0.000 abstract 1
- 208000029078 coronary artery disease Diseases 0.000 abstract 1
- 210000004351 coronary vessel Anatomy 0.000 abstract 1
- -1 heterocyclic pyridones Chemical class 0.000 abstract 1
- 239000003112 inhibitor Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 238000006467 substitution reaction Methods 0.000 abstract 1
- 238000002560 therapeutic procedure Methods 0.000 abstract 1
- 230000001732 thrombotic effect Effects 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyridine Compounds (AREA)
Abstract
El invento se relaciona con la substitución de los componentes de aril policíclico y de las piridonas heterociclicas que se utilizan como inhibidores en las variables dentadas en la coagulación en cascada y sus componentes, las composiciones y métodos para las terapias anticoagulante para el tratamiento y prevención de una variedad de condiciones trombóticas incluyendo la arteria coronaria y males cerebrovasculares.The invention relates to the substitution of the polycyclic aryl components and of the heterocyclic pyridones that are used as inhibitors in the toothed variables in cascade coagulation and its components, the compositions and methods for anticoagulant therapies for the treatment and prevention of a variety of thrombotic conditions including the coronary artery and cerebrovascular disease.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003477 ECSP003477A (en) | 2000-05-19 | 2000-05-19 | SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PYRIDONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003477 ECSP003477A (en) | 2000-05-19 | 2000-05-19 | SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PYRIDONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP003477A true ECSP003477A (en) | 2000-11-24 |
Family
ID=42041103
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP003477 ECSP003477A (en) | 2000-05-19 | 2000-05-19 | SUBSTITUTED POLYCLIC ARYL AND HETEROARIL PYRIDONES USEFUL FOR THE SELECTIVE INHIBITION OF THE COAGULATION WATERFALL |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP003477A (en) |
-
2000
- 2000-05-19 EC ECSP003477 patent/ECSP003477A/en unknown
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