ECSP003523A - N- CYCLOPENTIL MODULATORS OF THE RECEPTORY ACTIVITY OF BEMOQUINE - Google Patents
N- CYCLOPENTIL MODULATORS OF THE RECEPTORY ACTIVITY OF BEMOQUINEInfo
- Publication number
- ECSP003523A ECSP003523A ECSP003523A ECSP003523A EC SP003523 A ECSP003523 A EC SP003523A EC SP003523 A ECSP003523 A EC SP003523A EC SP003523 A ECSP003523 A EC SP003523A
- Authority
- EC
- Ecuador
- Prior art keywords
- modulators
- activity
- bemoquine
- receptory
- cyclopentil
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 2
- 102000004499 CCR3 Receptors Human genes 0.000 abstract 1
- 108010017316 CCR3 Receptors Proteins 0.000 abstract 1
- 102000004274 CCR5 Receptors Human genes 0.000 abstract 1
- 108010017088 CCR5 Receptors Proteins 0.000 abstract 1
- 102000009410 Chemokine receptor Human genes 0.000 abstract 1
- 108050000299 Chemokine receptor Proteins 0.000 abstract 1
- 102000019034 Chemokines Human genes 0.000 abstract 1
- 108010012236 Chemokines Proteins 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención está dirigida a los compuestos de la fórmula I (gráfico), (en que R1, R3, R4, R5, R6, R7, R8, X n, x y y se definen en este trabajo) que son útiles como moduladores de la actividad receptora de la quemoquina. En particular, estos compuestos son útiles como moduladores de los receptores CCR-5 y/o CCR-3 de la quemoquina.The present invention is directed to compounds of formula I (graph), (where R1, R3, R4, R5, R6, R7, R8, X n, x, and y are defined herein) which are useful as modulators of the chemokine receptor activity. In particular, these compounds are useful as modulators of chemokine CCR-5 and / or CCR-3 receptors.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003523 ECSP003523A (en) | 2000-06-09 | 2000-06-09 | N- CYCLOPENTIL MODULATORS OF THE RECEPTORY ACTIVITY OF BEMOQUINE |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003523 ECSP003523A (en) | 2000-06-09 | 2000-06-09 | N- CYCLOPENTIL MODULATORS OF THE RECEPTORY ACTIVITY OF BEMOQUINE |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP003523A true ECSP003523A (en) | 2000-08-18 |
Family
ID=42041147
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP003523 ECSP003523A (en) | 2000-06-09 | 2000-06-09 | N- CYCLOPENTIL MODULATORS OF THE RECEPTORY ACTIVITY OF BEMOQUINE |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP003523A (en) |
-
2000
- 2000-06-09 EC ECSP003523 patent/ECSP003523A/en unknown
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