ECSP003556A - INDAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR THE INHIBITION OF PROTEIN KINASE AND METHODS FOR USE - Google Patents
INDAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR THE INHIBITION OF PROTEIN KINASE AND METHODS FOR USEInfo
- Publication number
- ECSP003556A ECSP003556A ECSP003556A ECSP003556A EC SP003556 A ECSP003556 A EC SP003556A EC SP003556 A ECSP003556 A EC SP003556A EC SP003556 A ECSP003556 A EC SP003556A
- Authority
- EC
- Ecuador
- Prior art keywords
- compounds
- pharmaceutical compositions
- methods
- inhibition
- protein kinase
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 3
- 102000001253 Protein Kinase Human genes 0.000 title abstract 2
- 238000000034 method Methods 0.000 title abstract 2
- 108060006633 protein kinase Proteins 0.000 title abstract 2
- BAXOFTOLAUCFNW-UHFFFAOYSA-N 1H-indazole Chemical class C1=CC=C2C=NNC2=C1 BAXOFTOLAUCFNW-UHFFFAOYSA-N 0.000 title 1
- 230000005764 inhibitory process Effects 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 206010012689 Diabetic retinopathy Diseases 0.000 abstract 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 102000004022 Protein-Tyrosine Kinases Human genes 0.000 abstract 1
- 108090000412 Protein-Tyrosine Kinases Proteins 0.000 abstract 1
- 201000004681 Psoriasis Diseases 0.000 abstract 1
- 230000033115 angiogenesis Effects 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 230000004663 cell proliferation Effects 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000000694 effects Effects 0.000 abstract 1
- 125000003453 indazolyl group Chemical class N1N=C(C2=C1C=CC=C2)* 0.000 abstract 1
- 230000035755 proliferation Effects 0.000 abstract 1
- 206010039073 rheumatoid arthritis Diseases 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
- 230000026683 transduction Effects 0.000 abstract 1
- 238000010361 transduction Methods 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Se describieron los compuestos de indazol que modulan y/o inhiben la actividad de ciertas quinasas de proteina. Estos compuestos y composiciones farmacéuticas que los contienen son capaces de mediar la transducción señalada de quinasa tirosina y asi modulan y/o inhiben la proliferación de células superfluas. El invento es dirigido también para el uso terapéutico y farmaco de las composiciones farmacéuticas que contienen tales compuestos y para los métodos de tratar el cáncer y otras enfermedades asociadas a angiogpénesis superfluo y/o la proliferación celular, como retinopatia diabética glucoma noevascular, artritis reumatoide y soriasis por administra cabntidades efectivas de tales compuestos.Indazole compounds that modulate and / or inhibit the activity of certain protein kinases were described. These compounds and pharmaceutical compositions containing them are capable of mediating the indicated transduction of tyrosine kinase and thus modulate and / or inhibit the proliferation of superfluous cells. The invention is also directed to the therapeutic and pharmaceutical use of pharmaceutical compositions containing such compounds and to methods of treating cancer and other diseases associated with superfluous angiogenesis and / or cell proliferation, such as diabetic retinopathy, noevascular glucoma, rheumatoid arthritis, and psoriasis by administering effective amounts of such compounds.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003556 ECSP003556A (en) | 2000-06-30 | 2000-06-30 | INDAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR THE INHIBITION OF PROTEIN KINASE AND METHODS FOR USE |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003556 ECSP003556A (en) | 2000-06-30 | 2000-06-30 | INDAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR THE INHIBITION OF PROTEIN KINASE AND METHODS FOR USE |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP003556A true ECSP003556A (en) | 2000-10-24 |
Family
ID=42041170
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP003556 ECSP003556A (en) | 2000-06-30 | 2000-06-30 | INDAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR THE INHIBITION OF PROTEIN KINASE AND METHODS FOR USE |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP003556A (en) |
-
2000
- 2000-06-30 EC ECSP003556 patent/ECSP003556A/en unknown
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| PA8498001A1 (en) | INDAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR THE INHIBITION OF PROTEIN KINASA, AND METHODS FOR USE | |
| DOP2001000120A (en) | COMPOUNDS, PHARMACEUTICAL COMPOSITIONS OF INDAZOL AND METHODS TO MEASURE AND INHIBIT THE CELL PROLIFERATION | |
| ECSP066335A (en) | INDAZOL 3,5-DISPOSED COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS TO INTERVENE IN OR INHIBIT THE CELL PROLIFERATION | |
| ECSP055858A (en) | 2- (1H-INDAZOL-6-ILAMINO) - BENZAMID COMPOUNDS AS INHIBITORS OF USEFUL PROTEINKINASES FOR THE TREATMENT OF OPHTHALMIC DISEASES | |
| UY26190A1 (en) | TIAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR INHIBITING PROTEINKINASES AND METHODS FOR THEIR USE | |
| CO5280047A1 (en) | AMIDA COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS TO INHIBIT PROTEINKINASES, AND THEIR INSTRUCTIONS FOR USE | |
| TWI262914B (en) | Compounds and pharmaceutical compositions for inhibiting protein kinases | |
| GT200400136A (en) | 3.5-DISPOSED INDAZOL COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS TO INTERVENE IN OR INHIBIT CELLULAR APPROVALIFERATION. | |
| GT200100061A (en) | PHARMACEUTICAL COMPOUNDS AND COMPOSITIONS AND METHODS TO INHIBIT PROTEIN KINASES. | |
| ES2191187T3 (en) | BICYCLE HETEROAROMATIC COMPOUNDS AS INHIBITORS OF PROTEIN TIROSIN-QUINASA. | |
| PA8489701A1 (en) | UREAS DIFENIL- (W-CARBOXIARIL SUBSTITUTED AS RAF QUINASA INHIBITORS | |
| PA8550101A1 (en) | DERIVATIVES OF BENZAMIDA TIAZOL AND PHARMACEUTICAL COMPOSITIONS TO INHIBIT THE PROLIFERATION OF CELLS, AND METHODS FOR USE | |
| BRPI0413565B8 (en) | Quinazoline analogues as erbb2 receptor inhibitors, their use and their pharmaceutical composition | |
| UY26877A1 (en) | PIRAZOL-TIAZOL COMPOUNDS, PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM, AND ITS INSTRUCTIONS FOR INHIBITING CYCLINE-DEPENDENT KINASES | |
| ECSP003556A (en) | INDAZOLE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR THE INHIBITION OF PROTEIN KINASE AND METHODS FOR USE | |
| PA8525701A1 (en) | COMPOUNDS WITH HETEROCICLIC-HYDROXIMINE-FLUORENE NUCLEES AND PHARMACEUTICAL COMPOSITIONS FOR THE INHIBITION OF KINASE PROTEINS AND METHODS FOR USE | |
| UY26543A1 (en) | INDAZOL COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS FOR MEASURING OR INHIBITING CELL PROLIFERATION. | |
| DOP2003000788A (en) | INDAZOL COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS TO INHIBIT PROTEINKINES, AND PROCEDURES FOR USE | |
| UY26888A1 (en) | COMPOUNDS WITH HETEROCYCLIC-HYDROXIMINE-FLUORENE NUCLEUS AND PHARMACEUTICAL COMPOSITIONS FOR THE INHIBITION OF KINASE PROTEINS AND METHODS FOR USE | |
| UY26547A1 (en) | AMIDE COMPOUNDS AND PHARMACEUTICAL COMPOSITIONS FOR INHIBITING PROTEINKINASES, AND THEIR METHOD OF USE | |
| DOP2004000953A (en) | INDAZOL COMPOUNDS 3,5-DISPOSED, PHARMACEUTICAL COMPOSITIONS AND METHODS TO INTERVENE IN OR INHIBIT THE CELL PROLIFERATION. | |
| UY26667A1 (en) | COMPOUNDS, PHARMACEUTICAL COMPOSITIONS AND METHODS FOR INHIBITING PROTEIN KINASES |