ECSP003696A - SYNTHETIC COMBINATIONS OF AN NK1 RECEIVER ANTAGONIST AND A GABA STRUCTURAL ANALOG - Google Patents
SYNTHETIC COMBINATIONS OF AN NK1 RECEIVER ANTAGONIST AND A GABA STRUCTURAL ANALOGInfo
- Publication number
- ECSP003696A ECSP003696A ECSP003696A ECSP003696A EC SP003696 A ECSP003696 A EC SP003696A EC SP003696 A ECSP003696 A EC SP003696A EC SP003696 A ECSP003696 A EC SP003696A
- Authority
- EC
- Ecuador
- Prior art keywords
- structural analog
- synthetic combinations
- gaba
- antagonist
- receiver antagonist
- Prior art date
Links
- 239000005557 antagonist Substances 0.000 title 1
- 102000002002 Neurokinin-1 Receptors Human genes 0.000 abstract 3
- 108010040718 Neurokinin-1 Receptors Proteins 0.000 abstract 3
- BTCSSZJGUNDROE-UHFFFAOYSA-N gamma-aminobutyric acid Chemical class NCCCC(O)=O BTCSSZJGUNDROE-UHFFFAOYSA-N 0.000 abstract 3
- 239000002464 receptor antagonist Substances 0.000 abstract 2
- 229940044551 receptor antagonist Drugs 0.000 abstract 2
- 208000000094 Chronic Pain Diseases 0.000 abstract 1
- 208000002193 Pain Diseases 0.000 abstract 1
- 239000003814 drug Substances 0.000 abstract 1
- 238000004519 manufacturing process Methods 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 239000000825 pharmaceutical preparation Substances 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 239000011885 synergistic combination Substances 0.000 abstract 1
Landscapes
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La presente invención proporciona métodos de tratamiento usando combinaciones sinergísticas de un antagonista de receptor de NK1 y un análogo de GABA y composicioones farmacéuticas y productos que contienen al antagonista de receptor de NK1 y el análogo de GABA. La p resente invención también proporciona el uso de una natgonista de receptor de NK1 y un análogo de GABA para la fabricación de un medicamento para el tratamiento o la prevención del dolor crónico.The present invention provides methods of treatment using synergistic combinations of an NK1 receptor antagonist and a GABA analog and pharmaceutical compositions and products containing the NK1 receptor antagonist and the GABA analog. The present invention also provides the use of a NK1 receptor natgonist and a GABA analog for the manufacture of a medicament for the treatment or prevention of chronic pain.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003696 ECSP003696A (en) | 2000-10-06 | 2000-10-06 | SYNTHETIC COMBINATIONS OF AN NK1 RECEIVER ANTAGONIST AND A GABA STRUCTURAL ANALOG |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003696 ECSP003696A (en) | 2000-10-06 | 2000-10-06 | SYNTHETIC COMBINATIONS OF AN NK1 RECEIVER ANTAGONIST AND A GABA STRUCTURAL ANALOG |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP003696A true ECSP003696A (en) | 2001-03-22 |
Family
ID=42041285
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP003696 ECSP003696A (en) | 2000-10-06 | 2000-10-06 | SYNTHETIC COMBINATIONS OF AN NK1 RECEIVER ANTAGONIST AND A GABA STRUCTURAL ANALOG |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP003696A (en) |
-
2000
- 2000-10-06 EC ECSP003696 patent/ECSP003696A/en unknown
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