ECSP003775A - Antagonistas del receptor integrina alfa v - Google Patents
Antagonistas del receptor integrina alfa vInfo
- Publication number
- ECSP003775A ECSP003775A ECSP003775A ECSP003775A EC SP003775 A ECSP003775 A EC SP003775A EC SP003775 A ECSP003775 A EC SP003775A EC SP003775 A ECSP003775 A EC SP003775A
- Authority
- EC
- Ecuador
- Prior art keywords
- alphav
- antagonists
- present
- integrin
- inhibiting
- Prior art date
Links
- 239000005557 antagonist Substances 0.000 title abstract 2
- 102000006495 integrins Human genes 0.000 title 1
- 108010044426 integrins Proteins 0.000 title 1
- 230000002401 inhibitory effect Effects 0.000 abstract 2
- 201000001320 Atherosclerosis Diseases 0.000 abstract 1
- 208000006386 Bone Resorption Diseases 0.000 abstract 1
- 206010012689 Diabetic retinopathy Diseases 0.000 abstract 1
- 206010061218 Inflammation Diseases 0.000 abstract 1
- 229940127449 Integrin Receptor Antagonists Drugs 0.000 abstract 1
- 108010040765 Integrin alphaV Proteins 0.000 abstract 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 208000001132 Osteoporosis Diseases 0.000 abstract 1
- 230000033115 angiogenesis Effects 0.000 abstract 1
- 206010003246 arthritis Diseases 0.000 abstract 1
- 230000015572 biosynthetic process Effects 0.000 abstract 1
- 230000024279 bone resorption Effects 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000002757 inflammatory effect Effects 0.000 abstract 1
- 230000004054 inflammatory process Effects 0.000 abstract 1
- 108010045077 integrin alphaVbeta5 Proteins 0.000 abstract 1
- 208000002780 macular degeneration Diseases 0.000 abstract 1
- 206010061289 metastatic neoplasm Diseases 0.000 abstract 1
- 150000002842 nonanoic acids Chemical class 0.000 abstract 1
- 208000037803 restenosis Diseases 0.000 abstract 1
- 238000003786 synthesis reaction Methods 0.000 abstract 1
- 230000004614 tumor growth Effects 0.000 abstract 1
- 230000002792 vascular Effects 0.000 abstract 1
- 230000003612 virological effect Effects 0.000 abstract 1
Landscapes
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención se refiere a derivados novedosos de ácido nonanoico, su síntesis, y su uso como antagonistas del receptor de integrina alfaV. Más particularmente, los compuestos de la presente invención son antagonistas de los receptores integrina alfaV beta3 y alfaV beta5 y son útiles para inhibir la resorción ósea, tratar y prevenir osteoporosis, e inhibir restenosis vascular, retinopatía diabética, degeneración macular, angiogenesis, ateroesclerosis, inflamación, artritis inflamatoria, enfermedad viral, cáncer y crecimiento de tumor metastásico.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003775 ECSP003775A (es) | 2000-11-17 | 2000-11-17 | Antagonistas del receptor integrina alfa v |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003775 ECSP003775A (es) | 2000-11-17 | 2000-11-17 | Antagonistas del receptor integrina alfa v |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP003775A true ECSP003775A (es) | 2001-08-27 |
Family
ID=42041343
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP003775 ECSP003775A (es) | 2000-11-17 | 2000-11-17 | Antagonistas del receptor integrina alfa v |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP003775A (es) |
-
2000
- 2000-11-17 EC ECSP003775 patent/ECSP003775A/es unknown
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