ECSP003783A - 2- (3,5-bis-trifluoromethyl-phenyl) -N-methyl-N- (6-morpholin-4-yl-4-o-totyl-pyridin-3-yl) -isobutyramide - Google Patents
2- (3,5-bis-trifluoromethyl-phenyl) -N-methyl-N- (6-morpholin-4-yl-4-o-totyl-pyridin-3-yl) -isobutyramideInfo
- Publication number
- ECSP003783A ECSP003783A ECSP003783A ECSP003783A EC SP003783 A ECSP003783 A EC SP003783A EC SP003783 A ECSP003783 A EC SP003783A EC SP003783 A ECSP003783 A EC SP003783A
- Authority
- EC
- Ecuador
- Prior art keywords
- isobutyramide
- morpholin
- pyridin
- trifluoromethyl
- bis
- Prior art date
Links
- -1 3,5-bis-trifluoromethyl-phenyl Chemical group 0.000 title abstract 2
- 229940047889 isobutyramide Drugs 0.000 title abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 102000002002 Neurokinin-1 Receptors Human genes 0.000 abstract 1
- 108010040718 Neurokinin-1 Receptors Proteins 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 102000005962 receptors Human genes 0.000 abstract 1
- 108020003175 receptors Proteins 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Este invento se refiere al compuesto de la fórmula que es la 2-(3,5-bis-trifluorometil-fenil)¿N-metil-N-(6-morfolin-4-il-4-o-tolil-piridin-3-il)-isobutiramida . Se ha encontrado que este compuesto tiene una alta afinidad al receptor NK-1 y es por tanto útil en el tratamiento de enfermedades relacionadas con este receptor.This invention relates to the compound of the formula which is 2- (3,5-bis-trifluoromethyl-phenyl) N-methyl-N- (6-morpholin-4-yl-4-o-tolyl-pyridin-3 -il) -isobutyramide. It has been found that this compound has a high affinity to the NK-1 receptor and is therefore useful in the treatment of diseases related to this receptor.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003783 ECSP003783A (en) | 2000-11-23 | 2000-11-23 | 2- (3,5-bis-trifluoromethyl-phenyl) -N-methyl-N- (6-morpholin-4-yl-4-o-totyl-pyridin-3-yl) -isobutyramide |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003783 ECSP003783A (en) | 2000-11-23 | 2000-11-23 | 2- (3,5-bis-trifluoromethyl-phenyl) -N-methyl-N- (6-morpholin-4-yl-4-o-totyl-pyridin-3-yl) -isobutyramide |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP003783A true ECSP003783A (en) | 2001-06-22 |
Family
ID=42041348
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP003783 ECSP003783A (en) | 2000-11-23 | 2000-11-23 | 2- (3,5-bis-trifluoromethyl-phenyl) -N-methyl-N- (6-morpholin-4-yl-4-o-totyl-pyridin-3-yl) -isobutyramide |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP003783A (en) |
-
2000
- 2000-11-23 EC ECSP003783 patent/ECSP003783A/en unknown
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