ECSP003786A - RANGE-HYDROXIL-2 (FLUOROALQUILOAMINOCARBONIL) -1-PIPERACINAPENTANAMIDAS AND USES OF THEM - Google Patents
RANGE-HYDROXIL-2 (FLUOROALQUILOAMINOCARBONIL) -1-PIPERACINAPENTANAMIDAS AND USES OF THEMInfo
- Publication number
- ECSP003786A ECSP003786A ECSP003786A ECSP003786A EC SP003786 A ECSP003786 A EC SP003786A EC SP003786 A ECSP003786 A EC SP003786A EC SP003786 A ECSP003786 A EC SP003786A
- Authority
- EC
- Ecuador
- Prior art keywords
- treatment
- compounds
- hiv
- aids
- inhibitors
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 4
- 208000030507 AIDS Diseases 0.000 abstract 3
- 208000031886 HIV Infections Diseases 0.000 abstract 3
- 208000037357 HIV infectious disease Diseases 0.000 abstract 3
- 208000033519 human immunodeficiency virus infectious disease Diseases 0.000 abstract 3
- 239000003112 inhibitor Substances 0.000 abstract 2
- 238000000034 method Methods 0.000 abstract 2
- 230000002265 prevention Effects 0.000 abstract 2
- 108010010369 HIV Protease Proteins 0.000 abstract 1
- 239000003443 antiviral agent Substances 0.000 abstract 1
- 229940121357 antivirals Drugs 0.000 abstract 1
- 230000003115 biocidal effect Effects 0.000 abstract 1
- 229940042399 direct acting antivirals protease inhibitors Drugs 0.000 abstract 1
- 230000002519 immonomodulatory effect Effects 0.000 abstract 1
- 239000004615 ingredient Substances 0.000 abstract 1
- 239000000137 peptide hydrolase inhibitor Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 230000010076 replication Effects 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 229960005486 vaccine Drugs 0.000 abstract 1
- 230000003612 virological effect Effects 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Los compuestos y Hidroxi-2-(fluoroalquiloaminocarbonil)-1-piperacinapentanamida son inhibidores de la proteasa VIH e inhibidores de la replicación VIH. Estos compuestos son útiles en la prevención o tratamiento de la infección por VIH y en el tratamiento del SIDA, sea como compuestos, sales farmacéuticamente aceptables, ingredientes de composiciones farmacéuticas, o bien en combinación con otros antivirales inmunomoduladores antibióticos o vacunas. Los métodos para el tratamiento del SIDA y métodos para la prevención o tratamiento de la infección por VIH son igualmente descritos. Estos compuestos son efectivos en contra de mutantes virales VIH que son resistentes a inhibidores de proteasa que, en la actualidad, se utilizan para el tratamiento del SIDA y la infección por VIH.The compounds and Hydroxy-2- (fluoroalkyloaminocarbonyl) -1-piperazinepentanamide are inhibitors of the HIV protease and inhibitors of HIV replication. These compounds are useful in the prevention or treatment of HIV infection and in the treatment of AIDS, whether as compounds, pharmaceutically acceptable salts, ingredients of pharmaceutical compositions, or in combination with other antibiotic immunomodulatory antivirals or vaccines. The methods for the treatment of AIDS and methods for the prevention or treatment of HIV infection are also described. These compounds are effective against HIV viral mutants that are resistant to protease inhibitors that are currently used for the treatment of AIDS and HIV infection.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US16747899P | 1999-11-24 | 1999-11-24 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP003786A true ECSP003786A (en) | 2002-03-25 |
Family
ID=40410317
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP003786 ECSP003786A (en) | 1999-11-24 | 2000-11-24 | RANGE-HYDROXIL-2 (FLUOROALQUILOAMINOCARBONIL) -1-PIPERACINAPENTANAMIDAS AND USES OF THEM |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP003786A (en) |
-
2000
- 2000-11-24 EC ECSP003786 patent/ECSP003786A/en unknown
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