ECSP003814A - INHIBITORS OF AMINOTRANSPHERASE DEPENDENT OF AMINO ACIDS OF RAMIFIED CHAIN AND ITS USE IN THE TREATMENT OF DIABETIC RETINOPATHY. - Google Patents
INHIBITORS OF AMINOTRANSPHERASE DEPENDENT OF AMINO ACIDS OF RAMIFIED CHAIN AND ITS USE IN THE TREATMENT OF DIABETIC RETINOPATHY.Info
- Publication number
- ECSP003814A ECSP003814A ECSP003814A ECSP003814A EC SP003814 A ECSP003814 A EC SP003814A EC SP003814 A ECSP003814 A EC SP003814A EC SP003814 A ECSP003814 A EC SP003814A
- Authority
- EC
- Ecuador
- Prior art keywords
- dependent
- inhibitors
- diabetic retinopathy
- aminotranspherase
- treatment
- Prior art date
Links
- 239000003112 inhibitor Substances 0.000 title abstract 3
- 206010012689 Diabetic retinopathy Diseases 0.000 title abstract 2
- 230000001419 dependent effect Effects 0.000 title abstract 2
- 150000001413 amino acids Chemical class 0.000 title 1
- 241000124008 Mammalia Species 0.000 abstract 1
- 241001465754 Metazoa Species 0.000 abstract 1
- 208000017442 Retinal disease Diseases 0.000 abstract 1
- 206010038923 Retinopathy Diseases 0.000 abstract 1
- 102000003929 Transaminases Human genes 0.000 abstract 1
- 108090000340 Transaminases Proteins 0.000 abstract 1
- 150000005693 branched-chain amino acids Chemical class 0.000 abstract 1
- 206010012601 diabetes mellitus Diseases 0.000 abstract 1
- 230000037361 pathway Effects 0.000 abstract 1
- 230000000069 prophylactic effect Effects 0.000 abstract 1
- 230000001225 therapeutic effect Effects 0.000 abstract 1
Landscapes
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
La presente invención se refiere a un método para el tratamiento profiláctico y terapéutico de la retinopatía diabética. El método consiste en la administración de un inhibidor de la vía de la aminotransferasa dependiente de aminoácido de cadena ramificada (BCAT), a un animal, tal como un mamífero, en particular un humano, en una cantidad suficiente para tratar profiláctica y terapéuticamente la retinopatía diabética. La presente invención también se refiere a varios inhibidores novedosos de la vía de la BCAT.The present invention relates to a method for the prophylactic and therapeutic treatment of diabetic retinopathy. The method consists in the administration of a branched-chain amino acid-dependent aminotransferase (BCAT) inhibitor to an animal, such as a mammal, in particular a human, in an amount sufficient to prophylactically and therapeutically treat retinopathy. diabetic The present invention also relates to several novel inhibitors of the BCAT pathway.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003814 ECSP003814A (en) | 2000-12-07 | 2000-12-07 | INHIBITORS OF AMINOTRANSPHERASE DEPENDENT OF AMINO ACIDS OF RAMIFIED CHAIN AND ITS USE IN THE TREATMENT OF DIABETIC RETINOPATHY. |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003814 ECSP003814A (en) | 2000-12-07 | 2000-12-07 | INHIBITORS OF AMINOTRANSPHERASE DEPENDENT OF AMINO ACIDS OF RAMIFIED CHAIN AND ITS USE IN THE TREATMENT OF DIABETIC RETINOPATHY. |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP003814A true ECSP003814A (en) | 2001-04-23 |
Family
ID=42041366
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP003814 ECSP003814A (en) | 2000-12-07 | 2000-12-07 | INHIBITORS OF AMINOTRANSPHERASE DEPENDENT OF AMINO ACIDS OF RAMIFIED CHAIN AND ITS USE IN THE TREATMENT OF DIABETIC RETINOPATHY. |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP003814A (en) |
-
2000
- 2000-12-07 EC ECSP003814 patent/ECSP003814A/en unknown
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