ECSP003818A - ACTIVE COMPOUNDS IN THE GLUCOCORTICOID RECEIVER - Google Patents
ACTIVE COMPOUNDS IN THE GLUCOCORTICOID RECEIVERInfo
- Publication number
- ECSP003818A ECSP003818A ECSP003818A ECSP003818A EC SP003818 A ECSP003818 A EC SP003818A EC SP003818 A ECSP003818 A EC SP003818A EC SP003818 A ECSP003818 A EC SP003818A
- Authority
- EC
- Ecuador
- Prior art keywords
- compounds
- glucocorticoid
- receiver
- active compounds
- methods
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 6
- 239000003862 glucocorticoid Substances 0.000 title 1
- 238000000034 method Methods 0.000 abstract 2
- WQZGKKKJIJFFOK-GASJEMHNSA-N Glucose Natural products OC[C@H]1OC(O)[C@H](O)[C@@H](O)[C@@H]1O WQZGKKKJIJFFOK-GASJEMHNSA-N 0.000 abstract 1
- 239000008280 blood Substances 0.000 abstract 1
- 210000004369 blood Anatomy 0.000 abstract 1
- 239000003850 glucocorticoid receptor antagonist Substances 0.000 abstract 1
- 239000008103 glucose Substances 0.000 abstract 1
- 210000004185 liver Anatomy 0.000 abstract 1
- 230000018406 regulation of metabolic process Effects 0.000 abstract 1
- 238000002560 therapeutic procedure Methods 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Esta invención se relaciona con compuestos novedosos que son antagonistas del receptor glucocorticoide selectivo para el hígado, con métodos para preparar tales compuestos y con métodos para usar tales compuestos en terapia y en la regulación del metabolismo, especialmente bajando los niveles de glucosa en la sangre. Los compuestos mencionados son los compuestos de acuerdo a la fórmula I: (gráfico)This invention relates to novel compounds that are selective glucocorticoid receptor antagonists for the liver, with methods for preparing such compounds and with methods for using such compounds in therapy and in the regulation of metabolism, especially by lowering blood glucose levels. The compounds mentioned are the compounds according to formula I: (graph)
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003818 ECSP003818A (en) | 2000-12-07 | 2000-12-07 | ACTIVE COMPOUNDS IN THE GLUCOCORTICOID RECEIVER |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP003818 ECSP003818A (en) | 2000-12-07 | 2000-12-07 | ACTIVE COMPOUNDS IN THE GLUCOCORTICOID RECEIVER |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP003818A true ECSP003818A (en) | 2001-06-22 |
Family
ID=42041370
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP003818 ECSP003818A (en) | 2000-12-07 | 2000-12-07 | ACTIVE COMPOUNDS IN THE GLUCOCORTICOID RECEIVER |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP003818A (en) |
-
2000
- 2000-12-07 EC ECSP003818 patent/ECSP003818A/en unknown
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