ECSP014089A - USEFUL TROPANO DERIVATIVES IN THERAPY - Google Patents
USEFUL TROPANO DERIVATIVES IN THERAPYInfo
- Publication number
- ECSP014089A ECSP014089A ECSP014089A ECSP014089A EC SP014089 A ECSP014089 A EC SP014089A EC SP014089 A ECSP014089 A EC SP014089A EC SP014089 A ECSP014089 A EC SP014089A
- Authority
- EC
- Ecuador
- Prior art keywords
- tropano
- therapy
- derivatives
- useful
- optionally substituted
- Prior art date
Links
- 238000002560 therapeutic procedure Methods 0.000 title 1
- 125000001153 fluoro group Chemical group F* 0.000 abstract 3
- 125000005913 (C3-C6) cycloalkyl group Chemical group 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 125000000217 alkyl group Chemical group 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 239000012453 solvate Substances 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
La presente invención proporciona compuestos de fórmula, cuyo gráfico consta indicado abajo, en la que R1 es un cicloalquilo C3-6 opcionalmente sustituido con uno o más átomos de flúor, o alquilo C1-6 opcionalmente sustituido con uno o más átomos de flúor, o cicloalquil (C3-6) metilo opcionalmente sustituido en el anillo con uno o más átomos de flúor; sales y solvatos farmacéuticamente aceptables de estos; y procedimientos para su preparación, intermedios utilizados en su preparación, composiciones que los contienen y usos de dichos compuestos.The present invention provides compounds of the formula, the graph of which is indicated below, in which R 1 is a C 3-6 cycloalkyl optionally substituted with one or more fluorine atoms, or C 1-6 alkyl optionally substituted with one or more fluorine atoms, or C3-6 cycloalkyl methyl optionally substituted on the ring with one or more fluorine atoms; pharmaceutically acceptable salts and solvates thereof; and procedures for its preparation, intermediates used in its preparation, compositions containing them and uses of said compounds.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0014046A GB0014046D0 (en) | 2000-05-26 | 2000-05-26 | Compounds useful in therapy |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP014089A true ECSP014089A (en) | 2003-01-13 |
Family
ID=9893283
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP014089 ECSP014089A (en) | 2000-05-26 | 2001-05-24 | USEFUL TROPANO DERIVATIVES IN THERAPY |
Country Status (6)
| Country | Link |
|---|---|
| CN (1) | CN1830445B (en) |
| EC (1) | ECSP014089A (en) |
| GB (1) | GB0014046D0 (en) |
| GT (1) | GT200100096A (en) |
| UA (1) | UA73170C2 (en) |
| ZA (1) | ZA200209516B (en) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CN102993197B (en) * | 2012-12-27 | 2015-09-02 | 蕾硕医药化工（长沙）有限公司 | Tropinone derivative and its preparation method and application |
| CN107304205B (en) * | 2016-04-22 | 2020-10-30 | 上海医药工业研究院 | A kind of maraviro intermediate and preparation method thereof |
-
2000
- 2000-05-26 GB GB0014046A patent/GB0014046D0/en not_active Ceased
-
2001
- 2001-05-09 CN CN2006100735840A patent/CN1830445B/en not_active Expired - Lifetime
- 2001-05-24 GT GT200100096A patent/GT200100096A/en unknown
- 2001-05-24 EC ECSP014089 patent/ECSP014089A/en unknown
- 2001-09-05 UA UA2002119374A patent/UA73170C2/en unknown
-
2002
- 2002-11-22 ZA ZA200209516A patent/ZA200209516B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN1830445B (en) | 2011-04-20 |
| UA73170C2 (en) | 2005-06-15 |
| GB0014046D0 (en) | 2000-08-02 |
| GT200100096A (en) | 2002-01-11 |
| ZA200209516B (en) | 2003-10-22 |
| CN1830445A (en) | 2006-09-13 |
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