ECSP034517A - NEW DERIVATIVES OF M-AMINO-PHENIL-IMINO-IMIDAZOLIDINE FOR THE TREATMENT OF URINE INCONTINENCE - Google Patents
NEW DERIVATIVES OF M-AMINO-PHENIL-IMINO-IMIDAZOLIDINE FOR THE TREATMENT OF URINE INCONTINENCEInfo
- Publication number
- ECSP034517A ECSP034517A EC2003004517A ECSP034517A ECSP034517A EC SP034517 A ECSP034517 A EC SP034517A EC 2003004517 A EC2003004517 A EC 2003004517A EC SP034517 A ECSP034517 A EC SP034517A EC SP034517 A ECSP034517 A EC SP034517A
- Authority
- EC
- Ecuador
- Prior art keywords
- amino
- treatment
- imidazolidine
- phenil
- imino
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
- A61K31/4164—1,3-Diazoles
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
- C07D233/04—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D233/28—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D233/44—Nitrogen atoms not forming part of a nitro radical
- C07D233/50—Nitrogen atoms not forming part of a nitro radical with carbocyclic radicals directly attached to said nitrogen atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Pharmacology & Pharmacy (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Urology & Nephrology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
La presente invención se refiere a derivados de m-amino-fenilimino-imidazolidina con un nuevo patrón de sustituyentes en el anillo de fenilo, a su uso para la preparación de medicamentos, en especial para el tratamiento de incontinencia de orina y a procedimientos de preparación de los mismos.The present invention relates to m-amino-phenylimino-imidazolidine derivatives with a new pattern of substituents on the phenyl ring, their use for the preparation of medicaments, especially for the treatment of urinary incontinence and preparation procedures for the same.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10051005 | 2000-10-14 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP034517A true ECSP034517A (en) | 2003-04-25 |
Family
ID=7659815
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2003004517A ECSP034517A (en) | 2000-10-14 | 2003-03-17 | NEW DERIVATIVES OF M-AMINO-PHENIL-IMINO-IMIDAZOLIDINE FOR THE TREATMENT OF URINE INCONTINENCE |
Country Status (23)
| Country | Link |
|---|---|
| EP (1) | EP1328517A2 (en) |
| JP (1) | JP2004511547A (en) |
| KR (1) | KR20030046503A (en) |
| CN (1) | CN1471514A (en) |
| AR (1) | AR035923A1 (en) |
| AU (1) | AU2002215943A1 (en) |
| BG (1) | BG107711A (en) |
| BR (1) | BR0114603A (en) |
| CA (1) | CA2425563A1 (en) |
| CZ (1) | CZ20031333A3 (en) |
| DE (1) | DE10150312A1 (en) |
| EA (1) | EA200300460A1 (en) |
| EC (1) | ECSP034517A (en) |
| EE (1) | EE200300177A (en) |
| HU (1) | HUP0302245A3 (en) |
| IL (1) | IL155338A0 (en) |
| MX (1) | MXPA03003162A (en) |
| NO (1) | NO20031697L (en) |
| PL (1) | PL361359A1 (en) |
| SK (1) | SK4342003A3 (en) |
| WO (1) | WO2002032876A2 (en) |
| YU (1) | YU28203A (en) |
| ZA (1) | ZA200302345B (en) |
Families Citing this family (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP4168086B1 (en) * | 2008-04-16 | 2008-10-22 | 国立大学法人福井大学 | Imidazoline derivatives |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2806811A1 (en) * | 1978-02-17 | 1979-08-23 | Boehringer Sohn Ingelheim | NEW SUBSTITUTED 2-PHENYLIMINO-IMIDAZOLIDINE, THEIR ACID-ADDITIONAL SALTS, THESE MEDICINAL PRODUCTS AND METHOD FOR MANUFACTURING THE SAME |
| CA1201066A (en) * | 1981-11-20 | 1986-02-25 | Alcon Laboratories, Inc. | N-¬3,5-dichloro-4-(2-imidazolidinylideneamino)- phenyl|-acetamide solutions for lowering intraocular pressure |
| DE19514579A1 (en) * | 1995-04-20 | 1996-10-24 | Boehringer Ingelheim Kg | Use of alpha-1-olone agonists for the treatment of urinary incontinence |
-
2001
- 2001-10-11 CA CA002425563A patent/CA2425563A1/en not_active Abandoned
- 2001-10-11 EP EP01987747A patent/EP1328517A2/en not_active Withdrawn
- 2001-10-11 PL PL01361359A patent/PL361359A1/en not_active Application Discontinuation
- 2001-10-11 EE EEP200300177A patent/EE200300177A/en unknown
- 2001-10-11 IL IL15533801A patent/IL155338A0/en unknown
- 2001-10-11 KR KR10-2003-7005143A patent/KR20030046503A/en not_active Withdrawn
- 2001-10-11 EA EA200300460A patent/EA200300460A1/en unknown
- 2001-10-11 JP JP2002536060A patent/JP2004511547A/en active Pending
- 2001-10-11 AU AU2002215943A patent/AU2002215943A1/en not_active Abandoned
- 2001-10-11 HU HU0302245A patent/HUP0302245A3/en unknown
- 2001-10-11 CZ CZ20031333A patent/CZ20031333A3/en unknown
- 2001-10-11 YU YU28203A patent/YU28203A/en unknown
- 2001-10-11 MX MXPA03003162A patent/MXPA03003162A/en unknown
- 2001-10-11 BR BR0114603-3A patent/BR0114603A/en not_active IP Right Cessation
- 2001-10-11 WO PCT/EP2001/011764 patent/WO2002032876A2/en not_active Ceased
- 2001-10-11 DE DE10150312A patent/DE10150312A1/en not_active Withdrawn
- 2001-10-11 CN CNA018170870A patent/CN1471514A/en active Pending
- 2001-10-11 SK SK434-2003A patent/SK4342003A3/en not_active Application Discontinuation
- 2001-10-12 AR ARP010104787A patent/AR035923A1/en not_active Application Discontinuation
-
2003
- 2003-03-17 EC EC2003004517A patent/ECSP034517A/en unknown
- 2003-03-26 ZA ZA200302345A patent/ZA200302345B/en unknown
- 2003-04-08 BG BG107711A patent/BG107711A/en unknown
- 2003-04-11 NO NO20031697A patent/NO20031697L/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| KR20030046503A (en) | 2003-06-12 |
| EP1328517A2 (en) | 2003-07-23 |
| IL155338A0 (en) | 2003-11-23 |
| AR035923A1 (en) | 2004-07-28 |
| SK4342003A3 (en) | 2003-10-07 |
| MXPA03003162A (en) | 2004-12-06 |
| AU2002215943A1 (en) | 2002-04-29 |
| YU28203A (en) | 2006-05-25 |
| BR0114603A (en) | 2003-10-14 |
| EE200300177A (en) | 2003-08-15 |
| WO2002032876A2 (en) | 2002-04-25 |
| CN1471514A (en) | 2004-01-28 |
| EA200300460A1 (en) | 2004-02-26 |
| HUP0302245A2 (en) | 2003-10-28 |
| PL361359A1 (en) | 2004-10-04 |
| CZ20031333A3 (en) | 2003-08-13 |
| NO20031697L (en) | 2003-05-26 |
| BG107711A (en) | 2004-02-27 |
| JP2004511547A (en) | 2004-04-15 |
| NO20031697D0 (en) | 2003-04-11 |
| DE10150312A1 (en) | 2002-07-04 |
| HUP0302245A3 (en) | 2004-01-28 |
| CA2425563A1 (en) | 2002-04-25 |
| ZA200302345B (en) | 2004-04-23 |
| WO2002032876A3 (en) | 2002-07-18 |
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