ECSP034606A - Uso de antiprogestinas para la induccion de apoptosis en una celula - Google Patents
Uso de antiprogestinas para la induccion de apoptosis en una celulaInfo
- Publication number
- ECSP034606A ECSP034606A EC2003004606A ECSP034606A ECSP034606A EC SP034606 A ECSP034606 A EC SP034606A EC 2003004606 A EC2003004606 A EC 2003004606A EC SP034606 A ECSP034606 A EC SP034606A EC SP034606 A ECSP034606 A EC SP034606A
- Authority
- EC
- Ecuador
- Prior art keywords
- cell
- antiprogestin
- apoptosis
- antiprogestines
- induction
- Prior art date
Links
- 230000006882 induction of apoptosis Effects 0.000 title 1
- 230000000708 anti-progestin effect Effects 0.000 abstract 4
- 239000003418 antiprogestin Substances 0.000 abstract 4
- -1 4-acetylphenyl Chemical group 0.000 abstract 2
- 210000004027 cell Anatomy 0.000 abstract 2
- 206010006187 Breast cancer Diseases 0.000 abstract 1
- 208000026310 Breast neoplasm Diseases 0.000 abstract 1
- IZGGUFACPUOLFX-RYRKJORJSA-N C1CCC=C2CC[C@@H]([C@H]3[C@@](C)(C(CC3)=O)CC3)C3=C21 Chemical compound C1CCC=C2CC[C@@H]([C@H]3[C@@](C)(C(CC3)=O)CC3)C3=C21 IZGGUFACPUOLFX-RYRKJORJSA-N 0.000 abstract 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 230000018199 S phase Effects 0.000 abstract 1
- 230000006907 apoptotic process Effects 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 230000022131 cell cycle Effects 0.000 abstract 1
- 230000001939 inductive effect Effects 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 210000004881 tumor cell Anatomy 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/57—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Epidemiology (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La presente invención se relaciona con métodos y usos para inducir apoptosis en una célula, en particular una célula de cáncer de mama, mediante la administración de antiprogestinas, en particular la antiprogestina 11b-(4-acetilfenil) -17b-hidroxi-17a-(1, 1 2, 2, 2-pentafluoroetil) estra-4, 9- dien-ona o un derivado o análogo de la misma aceptable para uso farmacéutico. La invención se relaciona además con un tratamiento para el cáncer, donde un indicador de alto riesgo es una cantidad incrementada de células tumorales en la fase S del ciclo celular, tratamiento que comprende una antiprogestina, en particular la antiprogestina 11b-(4-acetilfenil)-17b-hidroxi-17a-(1, 1 2, 2,2- pentafluoroetil)-extra-4, 9-dien-3-ona o un derivado o análogo de la misma aceptable para uso farmacéutico
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP00250342 | 2000-10-18 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP034606A true ECSP034606A (es) | 2003-06-25 |
Family
ID=32049951
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2003004606A ECSP034606A (es) | 2000-10-18 | 2003-05-14 | Uso de antiprogestinas para la induccion de apoptosis en una celula |
Country Status (7)
| Country | Link |
|---|---|
| US (1) | US20040072811A1 (es) |
| AR (1) | AR030998A1 (es) |
| EC (1) | ECSP034606A (es) |
| PE (1) | PE20020511A1 (es) |
| RS (1) | RS50350B (es) |
| UY (1) | UY26966A1 (es) |
| ZA (1) | ZA200303790B (es) |
Families Citing this family (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US20080261933A1 (en) * | 2007-04-23 | 2008-10-23 | Jens Hoffmann | Combination of progesterone-receptor antagonist together with a lutein-hormone-releasing hormone agonist and antagonist for use in brca mediated diseases |
| WO2013052652A1 (en) | 2011-10-04 | 2013-04-11 | Erard Gilles | Methods and systems for identifying and treating anti-progestin sensitive tumors |
| CN113559075A (zh) | 2014-11-17 | 2021-10-29 | 康泰科思特生物制药公司 | 奥那司酮延长释放组合物和方法 |
| CA2998924A1 (en) | 2015-09-25 | 2017-03-30 | Context Biopharma Inc. | Methods of making onapristone intermediates |
| JP2019503353A (ja) | 2015-12-15 | 2019-02-07 | コンテキスト・バイオファーマ・インコーポレイテッド | 非晶質オナプリストン組成物およびそれを作製する方法 |
| US20180148471A1 (en) | 2016-11-30 | 2018-05-31 | Arno Therapeutics, Inc. | Methods for onapristone synthesis dehydration and deprotection |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE19706061A1 (de) * | 1997-02-07 | 1998-08-13 | Schering Ag | Antigestagen wirksame Steroide mit fluorierter 17alpha-Alkylkette |
-
2001
- 2001-10-12 UY UY26966A patent/UY26966A1/es not_active Application Discontinuation
- 2001-10-17 RS YUP-299/03A patent/RS50350B/sr unknown
- 2001-10-17 PE PE2001001032A patent/PE20020511A1/es not_active Application Discontinuation
- 2001-10-17 US US10/399,319 patent/US20040072811A1/en not_active Abandoned
- 2001-10-17 AR ARP010104868A patent/AR030998A1/es unknown
-
2003
- 2003-05-14 EC EC2003004606A patent/ECSP034606A/es unknown
- 2003-05-15 ZA ZA200303790A patent/ZA200303790B/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ZA200303790B (en) | 2004-08-16 |
| US20040072811A1 (en) | 2004-04-15 |
| RS50350B (sr) | 2009-11-10 |
| PE20020511A1 (es) | 2002-06-15 |
| AR030998A1 (es) | 2003-09-03 |
| UY26966A1 (es) | 2002-06-20 |
| YU29903A (sh) | 2006-08-17 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| MX9700534A (es) | Uso de droloxifeno y sus sales farmaceuticamente aceptables en la preparacion de remedios para tratar las enfermedades de prostata, endometriosis y obesidad. | |
| AU4550801A (en) | Herbal composition phy906 and its use in chemotheraphy | |
| IS4073A (is) | Nýtt fjölvirknislyf gegn aukningu mótstöðu | |
| NO986104D0 (no) | Progesteron-anti-progesteron regimer | |
| AR043071A1 (es) | Uso de macrolidos para el tratamiento del cancer y degeneracion macular y una composicion farmaceutica | |
| BR0114665A (pt) | Uso de antiprogestinas para a profilaxia e tratamento de doenças dependentes de hormÈnio | |
| ECSP034606A (es) | Uso de antiprogestinas para la induccion de apoptosis en una celula | |
| EA200200943A1 (ru) | Гормональная терапия рака молочной железы | |
| BR0114696A (pt) | Uso de antiprogestinas para a indução de apoptose em uma célula | |
| CY1111406T1 (el) | Χρηση βαλερικης οιστραδιολης ή οιστραδιολης σε συνδυασμο με διενογεστη για την απο του στοματος θεραπεια της αιμορραγιας λογω δυσλειτουργιας της μητρας με τη μορφη απο του στοματος αντισυλληψης | |
| IT1093259B (it) | Composizione per il trattamento,in particolare,della cellulite | |
| AR032371A1 (es) | Uso de antiprogestinas para la profilaxis y el tratamiento de enfermedades dependientes de hormonas | |
| DK1161254T3 (da) | Behandling af autoimmune sygdomme med en ekstrakt af amerikansk ginseng | |
| AR109456A2 (es) | Uso de et743 para la preparación de un medicamento para el tratamiento de un paciente humano afectado por cáncer mediante terapia de combinación | |
| ES2086413T3 (es) | Utilizacion de agentes antigestagenos para la preparacion de medicamentos. | |
| IT8519041A1 (it) | Uso terapeutico del ciproterone acetato | |
| IT1224673B (it) | Composizione farmaceutica comprendente un analogo di somatostatina esuo impiego nel trattamento del cancro della mammella | |
| AR061949A1 (es) | Uso de nitro derivados de flavonas como agentes inductores de apoptosis para la preparacion de un medicamento | |
| DK1937274T3 (da) | Anvendelse af estradiolvalerat i kombination med dienogest til oral behandling af dysfunktionel uterin blødning i enhed med en oral kontraception | |
| MX145118A (es) | Mejoras en aparato medico auxiliar para el tratamiento de hemorroides | |
| GR21106B (el) | Βελτιωσεις εις και σχετικως προς μεθοδον παρασκευης φαρμακευτικων παρασκευασματων τεταρτογενων αμμωνιακων ενωσεων. | |
| AR023380A1 (es) | Compuestos para la terapia y el diagnostico de cancer de pulmon y metodos de uso de los mismos |