ECSP034715A - ERK2 HETEROCICLIC INHIBITORS AND THEIR USES OF THE SAME - Google Patents
ERK2 HETEROCICLIC INHIBITORS AND THEIR USES OF THE SAMEInfo
- Publication number
- ECSP034715A ECSP034715A ECSP034715A ECSP034715A EC SP034715 A ECSP034715 A EC SP034715A EC SP034715 A ECSP034715 A EC SP034715A EC SP034715 A ECSP034715 A EC SP034715A
- Authority
- EC
- Ecuador
- Prior art keywords
- inhibitors
- heterociclic
- erk2
- same
- compounds
- Prior art date
Links
- 101000876610 Dictyostelium discoideum Extracellular signal-regulated kinase 2 Proteins 0.000 title 1
- 101001052493 Homo sapiens Mitogen-activated protein kinase 1 Proteins 0.000 title 1
- 102100024193 Mitogen-activated protein kinase 1 Human genes 0.000 title 1
- 239000003112 inhibitor Substances 0.000 title 1
- 229940045988 antineoplastic drug protein kinase inhibitors Drugs 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 239000003909 protein kinase inhibitor Substances 0.000 abstract 2
- 239000012824 ERK inhibitor Substances 0.000 abstract 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
- 150000003217 pyrazoles Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
El invento se refiere a la química medicinal y se refiere a los compuestos de pirazol que son inhibidores de protein quinasa, especialmente inhibidores de ERK, composiciones que contienen dichos compuestos y métodos de uso. Los compuestos son útiles para tratar el cáncer y otras enfermedades que son aliviados por los inhibidores de protein quinasa.The invention relates to medicinal chemistry and refers to pyrazole compounds that are protein kinase inhibitors, especially ERK inhibitors, compositions containing said compounds and methods of use. The compounds are useful for treating cancer and other diseases that are relieved by protein kinase inhibitors.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US26781801P | 2001-02-09 | 2001-02-09 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP034715A true ECSP034715A (en) | 2003-10-28 |
Family
ID=34078830
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP034715 ECSP034715A (en) | 2001-02-09 | 2003-08-07 | ERK2 HETEROCICLIC INHIBITORS AND THEIR USES OF THE SAME |
Country Status (2)
| Country | Link |
|---|---|
| EC (1) | ECSP034715A (en) |
| ZA (1) | ZA200305799B (en) |
-
2003
- 2003-07-28 ZA ZA200305799A patent/ZA200305799B/en unknown
- 2003-08-07 EC ECSP034715 patent/ECSP034715A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| ZA200305799B (en) | 2004-07-28 |
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