ECSP045071A - CYCLLOXYGENASA-2 INHIBITOR COMBINATION / HISTONA DEACETILATE INHIBITOR - Google Patents
CYCLLOXYGENASA-2 INHIBITOR COMBINATION / HISTONA DEACETILATE INHIBITORInfo
- Publication number
- ECSP045071A ECSP045071A ECSP045071A ECSP045071A EC SP045071 A ECSP045071 A EC SP045071A EC SP045071 A ECSP045071 A EC SP045071A EC SP045071 A ECSP045071 A EC SP045071A
- Authority
- EC
- Ecuador
- Prior art keywords
- inhibitor
- combination
- deacetilate
- cyclloxygenasa
- histona
- Prior art date
Links
- 239000003112 inhibitor Substances 0.000 title 2
- 206010009944 Colon cancer Diseases 0.000 abstract 2
- 241000124008 Mammalia Species 0.000 abstract 2
- 206010028980 Neoplasm Diseases 0.000 abstract 2
- 210000001072 colon Anatomy 0.000 abstract 2
- 208000029742 colonic neoplasm Diseases 0.000 abstract 2
- 239000003255 cyclooxygenase 2 inhibitor Substances 0.000 abstract 2
- 230000003902 lesion Effects 0.000 abstract 2
- 230000036210 malignancy Effects 0.000 abstract 2
- 230000003211 malignant effect Effects 0.000 abstract 2
- 229940093444 Cyclooxygenase 2 inhibitor Drugs 0.000 abstract 1
- 229940111134 coxibs Drugs 0.000 abstract 1
- 229940121372 histone deacetylase inhibitor Drugs 0.000 abstract 1
- 239000003276 histone deacetylase inhibitor Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Landscapes
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
La invención se refiere a una combinación que comprende (a) un inhibidor de ciclooxigenasa-2 ("inhibidor de COX-2") y (b) un inhibidor de desacetilasa de histona ("HDAI") para uso simultáneo, concurrente, separado o secuencial, especialmente para utilizarse en el tratamiento de lesiones colon pre-malignas o un cáncer de colon u otras malignidades en un mamífero, particularmente un ser humano. La invención también se refiere a composiciones farmacéuticas que comprenden dicha combinación y a un método para tratar lesiones de colon pre-malignas (por ejemplo, pólipos) y cáncer de colon, así como otras malignidades, en un mamífero, particularmente un ser humano, con dicha combinación. La presente invención además también se refiere a un paquete o producto comercial que comprende dicha combinación.The invention relates to a combination comprising (a) a cyclooxygenase-2 inhibitor ("COX-2 inhibitor") and (b) a histone deacetylase inhibitor ("HDAI") for simultaneous, concurrent, separate or sequential, especially for use in the treatment of pre-malignant colon lesions or colon cancer or other malignancies in a mammal, particularly a human being. The invention also relates to pharmaceutical compositions comprising said combination and to a method for treating pre-malignant colon lesions (eg polyps) and colon cancer, as well as other malignancies, in a mammal, particularly a human being, with said combination. The present invention also further relates to a commercial package or product comprising said combination.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP045071 ECSP045071A (en) | 2004-04-21 | 2004-04-21 | CYCLLOXYGENASA-2 INHIBITOR COMBINATION / HISTONA DEACETILATE INHIBITOR |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP045071 ECSP045071A (en) | 2004-04-21 | 2004-04-21 | CYCLLOXYGENASA-2 INHIBITOR COMBINATION / HISTONA DEACETILATE INHIBITOR |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP045071A true ECSP045071A (en) | 2004-05-28 |
Family
ID=40435095
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP045071 ECSP045071A (en) | 2004-04-21 | 2004-04-21 | CYCLLOXYGENASA-2 INHIBITOR COMBINATION / HISTONA DEACETILATE INHIBITOR |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP045071A (en) |
-
2004
- 2004-04-21 EC ECSP045071 patent/ECSP045071A/en unknown
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