ECSP045288A - DERIVATIVES OF AZETIDINE AS ANTAGONISTS OF THE CCR-3 RECEIVER - Google Patents
DERIVATIVES OF AZETIDINE AS ANTAGONISTS OF THE CCR-3 RECEIVERInfo
- Publication number
- ECSP045288A ECSP045288A ECSP045288A ECSP045288A EC SP045288 A ECSP045288 A EC SP045288A EC SP045288 A ECSP045288 A EC SP045288A EC SP045288 A ECSP045288 A EC SP045288A
- Authority
- EC
- Ecuador
- Prior art keywords
- ccr
- azetidine
- antagonists
- derivatives
- receiver
- Prior art date
Links
- 102100024167 C-C chemokine receptor type 3 Human genes 0.000 title abstract 2
- 101710149862 C-C chemokine receptor type 3 Proteins 0.000 title abstract 2
- 239000005557 antagonist Substances 0.000 title 1
- HONIICLYMWZJFZ-UHFFFAOYSA-N azetidine Chemical class C1CNC1 HONIICLYMWZJFZ-UHFFFAOYSA-N 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 3
- 230000001404 mediated effect Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Los compuestos de la Fórmula I en forma de sal o libre, donde Ae, X, Y, R1, R2, R3, R5, m, n, p y q tienen los significados indicados en la especificación, son útiles para tratar condiciones mediadas por CCR3. También se describen las composiciones farmacéuticas que contienen los compuestos y procesos para preparar los compuestos.The compounds of Formula I in salt or free form, where Ae, X, Y, R1, R2, R3, R5, m, n, p and q have the meanings indicated in the specification, are useful for treating conditions mediated by CCR3. The pharmaceutical compositions containing the compounds and processes for preparing the compounds are also described.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB0206218A GB0206218D0 (en) | 2002-03-15 | 2002-03-15 | Organic compounds |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP045288A true ECSP045288A (en) | 2004-10-26 |
Family
ID=9933095
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP045288 ECSP045288A (en) | 2002-03-15 | 2004-09-10 | DERIVATIVES OF AZETIDINE AS ANTAGONISTS OF THE CCR-3 RECEIVER |
Country Status (3)
| Country | Link |
|---|---|
| EC (1) | ECSP045288A (en) |
| GB (1) | GB0206218D0 (en) |
| ZA (1) | ZA200406752B (en) |
-
2002
- 2002-03-15 GB GB0206218A patent/GB0206218D0/en not_active Ceased
-
2004
- 2004-08-25 ZA ZA200406752A patent/ZA200406752B/en unknown
- 2004-09-10 EC ECSP045288 patent/ECSP045288A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| GB0206218D0 (en) | 2002-05-01 |
| ZA200406752B (en) | 2006-05-31 |
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