ECSP045322A - FORMULATIONS OF AN HID SUSPENSION WITH HFA - Google Patents
FORMULATIONS OF AN HID SUSPENSION WITH HFAInfo
- Publication number
- ECSP045322A ECSP045322A EC2004005322A ECSP045322A ECSP045322A EC SP045322 A ECSP045322 A EC SP045322A EC 2004005322 A EC2004005322 A EC 2004005322A EC SP045322 A ECSP045322 A EC SP045322A EC SP045322 A ECSP045322 A EC SP045322A
- Authority
- EC
- Ecuador
- Prior art keywords
- hfa
- hid
- formulations
- suspension
- hydroxidi
- Prior art date
Links
- 239000000203 mixture Substances 0.000 title abstract 2
- 239000000725 suspension Substances 0.000 title abstract 2
- BKIMMITUMNQMOS-UHFFFAOYSA-N nonane Chemical compound CCCCCCCCC BKIMMITUMNQMOS-UHFFFAOYSA-N 0.000 abstract 2
- CPELXLSAUQHCOX-UHFFFAOYSA-M Bromide Chemical compound [Br-] CPELXLSAUQHCOX-UHFFFAOYSA-M 0.000 abstract 1
- 239000012159 carrier gas Substances 0.000 abstract 1
- 238000009472 formulation Methods 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/007—Pulmonary tract; Aromatherapy
- A61K9/0073—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
- A61K9/008—Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy comprising drug dissolved or suspended in liquid propellant for inhalation via a pressurized metered dose inhaler [MDI]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/439—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom the ring forming part of a bridged ring system, e.g. quinuclidine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/10—Dispersions; Emulsions
- A61K9/12—Aerosols; Foams
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Epidemiology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Dispersion Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Otolaryngology (AREA)
- Medicinal Preparation (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
Abstract
La invención se refiere a formulaciones con gas portador que contienen suspensiones del anhidrato cristalino de bromuro de (1a,2b,4b,5a,7b)-7-[(hidroxidi-2- -tienilacetil)oxi]-9,9-dimetil-3-oxa-9-azonia-triciclo[3.3.1.02,4]nonano.The invention relates to carrier gas formulations containing suspensions of the crystalline bromide anhydrate of (1a, 2b, 4b, 5a, 7b) -7 - [(hydroxidi-2--thienylacetyl) oxy] -9,9-dimethyl- 3-oxa-9-azonia-tricycle [3.3.1.02.4] nonane.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE10214264A DE10214264A1 (en) | 2002-03-28 | 2002-03-28 | HFA suspension formulations of an anhydrate |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP045322A true ECSP045322A (en) | 2005-01-28 |
Family
ID=28050990
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2004005322A ECSP045322A (en) | 2002-03-28 | 2004-09-28 | FORMULATIONS OF AN HID SUSPENSION WITH HFA |
Country Status (21)
| Country | Link |
|---|---|
| EP (1) | EP1492498A2 (en) |
| JP (1) | JP5147158B2 (en) |
| KR (1) | KR101005717B1 (en) |
| CN (1) | CN1642525A (en) |
| AU (1) | AU2003221509B2 (en) |
| BR (1) | BR0308709A (en) |
| CA (1) | CA2479638C (en) |
| DE (1) | DE10214264A1 (en) |
| EA (1) | EA008610B1 (en) |
| EC (1) | ECSP045322A (en) |
| HR (1) | HRP20040890A2 (en) |
| IL (1) | IL163696A0 (en) |
| ME (1) | ME00246B (en) |
| MX (1) | MXPA04009338A (en) |
| NO (1) | NO20044004L (en) |
| NZ (1) | NZ536030A (en) |
| PL (1) | PL371295A1 (en) |
| RS (1) | RS52481B (en) |
| UA (1) | UA79776C2 (en) |
| WO (1) | WO2003082244A2 (en) |
| ZA (1) | ZA200405637B (en) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP2008540367A (en) * | 2005-05-02 | 2008-11-20 | ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング | New crystalline tiotropium bromide |
| WO2006117299A2 (en) * | 2005-05-02 | 2006-11-09 | Boehringer Ingelheim International Gmbh | Novel crystalline forms of tiotropium bromide |
| US8815258B2 (en) | 2009-05-29 | 2014-08-26 | Pearl Therapeutics, Inc. | Compositions, methods and systems for respiratory delivery of two or more active agents |
| AU2015201037C1 (en) * | 2009-05-29 | 2017-07-27 | Pearl Therapeutics, Inc. | Respiratory delivery of active agents |
| PL3111927T3 (en) | 2009-05-29 | 2020-06-29 | Pearl Therapeutics, Inc. | Compositions for respiratory delivery of active agents and associated methods and systems |
| SG11201507286QA (en) | 2013-03-15 | 2015-10-29 | Pearl Therapeutics Inc | Methods and systems for conditioning of particulate crystalline materials |
| CN114712337A (en) * | 2016-09-19 | 2022-07-08 | 墨西哥氟石股份公司 | Pharmaceutical composition |
Family Cites Families (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3931041C2 (en) * | 1989-09-16 | 2000-04-06 | Boehringer Ingelheim Kg | Esters of thienyl carboxylic acids with amino alcohols, their quaternization products, processes for their preparation and medicaments containing them |
| JP4672143B2 (en) * | 1998-08-04 | 2011-04-20 | ヤゴテック アーゲー | Pharmaceutical aerosol formulation |
| GB0009583D0 (en) * | 2000-04-18 | 2000-06-07 | Glaxo Group Ltd | Respiratory formulations |
| GB0009605D0 (en) * | 2000-04-18 | 2000-06-07 | Glaxo Group Ltd | Medicaments |
| GB0009592D0 (en) * | 2000-04-18 | 2000-06-07 | Glaxo Group Ltd | Respiratory combinations |
| GB0009606D0 (en) * | 2000-04-18 | 2000-06-07 | Glaxo Group Ltd | Therapeutic combinations |
| JP2004512379A (en) * | 2000-10-31 | 2004-04-22 | ベーリンガー インゲルハイム ファルマ ゲゼルシャフト ミット ベシュレンクテル ハフツング ウント コンパニー コマンディトゲゼルシャフト | New pharmaceutical composition |
| DE10113366A1 (en) * | 2001-03-20 | 2002-09-26 | Boehringer Ingelheim Pharma | Medicament for treating inflammatory or obstructive respiratory diseases, e.g. asthma or chronic obstructive pulmonary disease, containing synergistic combination of anticholinergic agent and endothelin antagonist |
| DE10111058A1 (en) * | 2001-03-08 | 2002-09-12 | Boehringer Ingelheim Pharma | New drug compositions based on anticholinergics and NK¶1¶ receptor antagonists |
-
2002
- 2002-03-28 DE DE10214264A patent/DE10214264A1/en not_active Withdrawn
-
2003
- 2003-03-20 EP EP03717219A patent/EP1492498A2/en not_active Withdrawn
- 2003-03-20 CN CNA038072475A patent/CN1642525A/en active Pending
- 2003-03-20 IL IL16369603A patent/IL163696A0/en unknown
- 2003-03-20 EA EA200401159A patent/EA008610B1/en unknown
- 2003-03-20 WO PCT/EP2003/002899 patent/WO2003082244A2/en not_active Ceased
- 2003-03-20 HR HR20040890A patent/HRP20040890A2/en not_active Application Discontinuation
- 2003-03-20 JP JP2003579782A patent/JP5147158B2/en not_active Expired - Lifetime
- 2003-03-20 UA UA20041008758A patent/UA79776C2/en unknown
- 2003-03-20 ME MEP-2008-473A patent/ME00246B/en unknown
- 2003-03-20 CA CA2479638A patent/CA2479638C/en not_active Expired - Fee Related
- 2003-03-20 BR BR0308709-3A patent/BR0308709A/en not_active Application Discontinuation
- 2003-03-20 NZ NZ536030A patent/NZ536030A/en not_active IP Right Cessation
- 2003-03-20 MX MXPA04009338A patent/MXPA04009338A/en active IP Right Grant
- 2003-03-20 RS YU86004A patent/RS52481B/en unknown
- 2003-03-20 PL PL03371295A patent/PL371295A1/en not_active Application Discontinuation
- 2003-03-20 KR KR1020047015174A patent/KR101005717B1/en not_active Expired - Lifetime
- 2003-03-20 AU AU2003221509A patent/AU2003221509B2/en not_active Expired
-
2004
- 2004-07-15 ZA ZA2004/05637A patent/ZA200405637B/en unknown
- 2004-09-23 NO NO20044004A patent/NO20044004L/en not_active Application Discontinuation
- 2004-09-28 EC EC2004005322A patent/ECSP045322A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| UA79776C2 (en) | 2007-07-25 |
| WO2003082244A2 (en) | 2003-10-09 |
| MXPA04009338A (en) | 2005-01-25 |
| EP1492498A2 (en) | 2005-01-05 |
| DE10214264A1 (en) | 2003-10-16 |
| AU2003221509A1 (en) | 2003-10-13 |
| NZ536030A (en) | 2006-07-28 |
| CN1642525A (en) | 2005-07-20 |
| ME00246B (en) | 2011-05-10 |
| BR0308709A (en) | 2005-01-04 |
| NO20044004L (en) | 2004-10-05 |
| EA008610B1 (en) | 2007-06-29 |
| WO2003082244A3 (en) | 2004-02-05 |
| CA2479638A1 (en) | 2003-10-09 |
| CA2479638C (en) | 2011-01-04 |
| YU86004A (en) | 2006-08-17 |
| HRP20040890A2 (en) | 2005-06-30 |
| IL163696A0 (en) | 2005-12-18 |
| PL371295A1 (en) | 2005-06-13 |
| MEP47308A (en) | 2011-02-10 |
| AU2003221509B2 (en) | 2008-01-24 |
| JP2005527550A (en) | 2005-09-15 |
| KR101005717B1 (en) | 2011-01-05 |
| ZA200405637B (en) | 2005-07-27 |
| JP5147158B2 (en) | 2013-02-20 |
| EA200401159A1 (en) | 2005-04-28 |
| RS52481B (en) | 2013-02-28 |
| KR20040098022A (en) | 2004-11-18 |
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