ECSP045481A - EXCITING AMINO ACID PROPHARMS - Google Patents
EXCITING AMINO ACID PROPHARMSInfo
- Publication number
- ECSP045481A ECSP045481A ECSP045481A ECSP045481A EC SP045481 A ECSP045481 A EC SP045481A EC SP045481 A ECSP045481 A EC SP045481A EC SP045481 A ECSP045481 A EC SP045481A
- Authority
- EC
- Ecuador
- Prior art keywords
- amino acid
- propharms
- exciting amino
- exciting
- methods
- Prior art date
Links
- 150000001413 amino acids Chemical class 0.000 title 1
- 238000000034 method Methods 0.000 abstract 2
- 208000012902 Nervous system disease Diseases 0.000 abstract 1
- 208000025966 Neurological disease Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000002461 excitatory amino acid Effects 0.000 abstract 1
- 239000003257 excitatory amino acid Substances 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 239000000651 prodrug Substances 0.000 abstract 1
- 229940002612 prodrug Drugs 0.000 abstract 1
- 208000020016 psychiatric disease Diseases 0.000 abstract 1
Landscapes
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Abstract
Esta invención se refiere a profármacos de aminoácidos excitadores sintéticos y a procedimientos para su preparación. La invención se refiere además a procedimientos de uso y a composiciones farmacéuticas que comprenden compuestos para el tratamiento de trastornos neurológicos y trastornos psiquiátricos.This invention relates to synthetic excitatory amino acid prodrugs and methods for their preparation. The invention further relates to methods of use and pharmaceutical compositions comprising compounds for the treatment of neurological disorders and psychiatric disorders.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP02380120 | 2002-06-11 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP045481A true ECSP045481A (en) | 2005-01-28 |
Family
ID=38691951
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP045481 ECSP045481A (en) | 2002-06-11 | 2004-12-09 | EXCITING AMINO ACID PROPHARMS |
Country Status (2)
| Country | Link |
|---|---|
| CN (2) | CN100482680C (en) |
| EC (1) | ECSP045481A (en) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP5945592B2 (en) * | 2011-06-17 | 2016-07-05 | イーライ リリー アンド カンパニー | Bicyclo (3.1.0) hexane-2,6-dicarboxylic acid derivative as MGLU2 receptor agonist |
| RS56328B1 (en) * | 2012-06-01 | 2017-12-29 | Taisho Pharmaceutical Co Ltd | Prodrug of fluorine-containing amino acid |
Family Cites Families (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5688826A (en) * | 1995-11-16 | 1997-11-18 | Eli Lilly And Company | Excitatory amino acid derivatives |
-
2003
- 2003-06-06 CN CNB038135116A patent/CN100482680C/en not_active Expired - Lifetime
- 2003-06-06 CN CNA2008100962167A patent/CN101362793A/en active Pending
-
2004
- 2004-12-09 EC ECSP045481 patent/ECSP045481A/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| CN101084236A (en) | 2007-12-05 |
| CN100482680C (en) | 2009-04-29 |
| CN101362793A (en) | 2009-02-11 |
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