ECSP055713A - NEW ANTIMICOBACTERIAL COMPOUNDS - Google Patents
NEW ANTIMICOBACTERIAL COMPOUNDSInfo
- Publication number
- ECSP055713A ECSP055713A ECSP055713A ECSP055713A EC SP055713 A ECSP055713 A EC SP055713A EC SP055713 A ECSP055713 A EC SP055713A EC SP055713 A ECSP055713 A EC SP055713A
- Authority
- EC
- Ecuador
- Prior art keywords
- compounds
- new
- formula
- antimicobacterial
- mdr
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title abstract 6
- 201000009671 multidrug-resistant tuberculosis Diseases 0.000 abstract 3
- 238000000034 method Methods 0.000 abstract 2
- 206010065048 Latent tuberculosis Diseases 0.000 abstract 1
- 241000187479 Mycobacterium tuberculosis Species 0.000 abstract 1
- 239000002253 acid Substances 0.000 abstract 1
- 208000015355 drug-resistant tuberculosis Diseases 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 150000003233 pyrroles Chemical class 0.000 abstract 1
- 150000003839 salts Chemical class 0.000 abstract 1
- 230000001988 toxicity Effects 0.000 abstract 1
- 231100000419 toxicity Toxicity 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
RESUMEN DE LA INVENCIÓN Nuevos derivados de pirrol de la fórmula (I) y sus sales por adición de ácido farmacéuticamente aceptables que tienen actividad antimicobacteriana superior contra cepas clínicamente sensibles así como resistentes de Mycobacterium tuberculosis que también tienen menor toxicidad en comparación a compuestos conocidos. El uso de los nuevos compuestos de la fórmula (I) para tratamiento de tuberculosis latente incluyendo Tuberculosis Resistente a Múltiples Fármacos (MDR TB). Los métodos para la preparación de los nuevos compuestos, composiciones farmacéuticas que contienen los nuevos compuestos y método de tratamiento de MDR TB mediante administración de compuestos de la fórmula (I).SUMMARY OF THE INVENTION New pyrrole derivatives of the formula (I) and their pharmaceutically acceptable acid addition salts having superior antimicobacterial activity against clinically sensitive as well as resistant Mycobacterium tuberculosis strains that also have lower toxicity compared to known compounds. The use of the new compounds of the formula (I) for the treatment of latent tuberculosis including Multiple Drug Resistant Tuberculosis (MDR TB). The methods for the preparation of the new compounds, pharmaceutical compositions containing the new compounds and method of treatment of MDR TB by administration of compounds of the formula (I).
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP055713 ECSP055713A (en) | 2005-03-31 | 2005-03-31 | NEW ANTIMICOBACTERIAL COMPOUNDS |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| ECSP055713 ECSP055713A (en) | 2005-03-31 | 2005-03-31 | NEW ANTIMICOBACTERIAL COMPOUNDS |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP055713A true ECSP055713A (en) | 2005-11-22 |
Family
ID=40202991
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ECSP055713 ECSP055713A (en) | 2005-03-31 | 2005-03-31 | NEW ANTIMICOBACTERIAL COMPOUNDS |
Country Status (1)
| Country | Link |
|---|---|
| EC (1) | ECSP055713A (en) |
-
2005
- 2005-03-31 EC ECSP055713 patent/ECSP055713A/en unknown
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