ECSP056252A - PIRAZOLOPIRIMIDINAS - Google Patents

PIRAZOLOPIRIMIDINAS

Info

Publication number
ECSP056252A
ECSP056252A ECSP056252A ECSP056252A EC SP056252 A ECSP056252 A EC SP056252A EC SP056252 A ECSP056252 A EC SP056252A EC SP056252 A ECSP056252 A EC SP056252A
Authority
EC
Ecuador
Prior art keywords
xii
products
obtaining
procedures
pirazolopirimidinas
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Hans Ludwig Elbe
Joerg Nico Greul
Ulrike Wachendorff-Neumann
Peter Dahmen
Kart-Heinz Kuck
Olaf Gebauer
Ulrich Heinemann
Herbert Gayer
Stefan Hillebrand
Ronald Ebbert
Oliver Guth
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from DE10339360A external-priority patent/DE10339360A1/en
Priority claimed from DE2003157570 external-priority patent/DE10357570A1/en
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of ECSP056252A publication Critical patent/ECSP056252A/en

Links

Landscapes

  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Nuevas pirazolopirimidinas de la fórmula (I) (I)en la queR1, R2, R3, R4, X y Hal tienen los significados anteriormente indicados,varios procedimientos para la obtención de estos productos y su empleo para la lucha contra los microorganismos indeseados. Nuevos productos intermedios de las fórmulas (II), (X), (XII-a) y (XII-b) (II) (X) (XII-a)y (XII-b)así como procedimientos para la obtención de estos productos.New pyrazolopyrimidines of the formula (I) (I) in which R1, R2, R3, R4, X and Hal have the meanings indicated above, various procedures for obtaining these products and their use for the fight against unwanted microorganisms. New intermediate products of the formulas (II), (X), (XII-a) and (XII-b) (II) (X) (XII-a) and (XII-b) as well as procedures for obtaining these products.

ECSP056252 2003-06-27 2005-12-26 PIRAZOLOPIRIMIDINAS ECSP056252A (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DE10328996 2003-06-27
DE10339360A DE10339360A1 (en) 2003-06-27 2003-08-27 New 7-amino-5-halo-pyrazolo-(1,5-a)-pyrimidine derivatives, useful as microbicides, especially fungicides or bactericides for protecting plants or materials such as wood
DE2003157570 DE10357570A1 (en) 2003-12-10 2003-12-10 New 7-amino-5-halo-pyrazolo-(1,5-a)-pyrimidine derivatives, useful as microbicides, especially fungicides or bactericides for protecting plants or materials such as wood

Publications (1)

Publication Number Publication Date
ECSP056252A true ECSP056252A (en) 2006-04-19

Family

ID=40506494

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP056252 ECSP056252A (en) 2003-06-27 2005-12-26 PIRAZOLOPIRIMIDINAS

Country Status (3)

Country Link
EA (1) EA009517B1 (en)
EC (1) ECSP056252A (en)
IL (1) IL172592A0 (en)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
SI2350075T1 (en) 2008-09-22 2014-06-30 Array Biopharma, Inc. Substituted imidazoš1,2bćpyridazine compounds as trk kinase inhibitors
CN102264736B (en) 2008-10-22 2013-08-14 阵列生物制药公司 Substituted pyrazolo[1,5-a]pyrimidine compounds as TRK kinase inhibitors
AR077468A1 (en) 2009-07-09 2011-08-31 Array Biopharma Inc PIRAZOLO COMPOUNDS (1,5-A) PYRIMIDINE SUBSTITUTED AS TRK-QUINASA INHIBITORS
HUE035248T2 (en) * 2011-08-17 2018-05-02 Adama Makhteshim Ltd 1-substituted-5-fluoro-3,6-dihydro-6-imino-2(1H)-pyrimidinone derivatives as fungicidal agents for use in plant protection
UA114490C2 (en) * 2011-10-06 2017-06-26 Байєр Інтеллектуал Проперті Гмбх Heterocyclylpyri(mi)dinylpyrazole as fungicidals
IN2014CN02475A (en) * 2011-10-06 2015-06-19 Bayer Ip Gmbh
HUE047711T2 (en) * 2012-12-28 2020-05-28 Adama Makhteshim Ltd N-(substituted)-5-fluoro-4-imino-3-methyl-2-oxo-3,4-dihydropyrimidine-1 (2h)-carboxylate derivatives
CA2894553C (en) * 2012-12-31 2021-03-02 Dow Agrosciences Llc 3-alkyl-5-fluoro-4-substituted-imino-3,4-dihydropyrimidin-2(1h)-one derivatives as fungicides
TWI746426B (en) 2014-11-16 2021-11-21 美商亞雷生物製藥股份有限公司 Crystalline form of (s)-n-(5-((r)-2-(2,5-difluorophenyl)-pyrrolidin-1-yl)-pyrazolo[1,5-a]pyrimidin-3-yl)-3-hydroxypyrrolidine-1-carboxamide hydrogen sulfate
EP3368039A1 (en) 2015-10-26 2018-09-05 The Regents of The University of Colorado, A Body Corporate Point mutations in trk inhibitor-resistant cancer and methods relating to the same
UA125025C2 (en) 2016-04-04 2021-12-29 Локсо Онколоджі, Інк. Methods of treating pediatric cancers
UA125026C2 (en) 2016-04-04 2021-12-29 Локсо Онколоджі, Інк. Liquid formulations of (s)-n-(5-(r)-2-(2,5-difluorophenyl)-pyrrolidin-1-yl)-pyrazolo[1,5-a]pyrimidin-3-yl)-3-hydroxypyrrolidine-1-carboxamide
ES2953467T3 (en) 2016-04-15 2023-11-13 Elanco Animal Health Gmbh Pyrazolopyrimidine derivatives
MX392604B (en) 2016-05-18 2025-03-24 Array Biopharma Inc Preparation of (s)-n-(5-((r)-2-(2,5-difluorophenyl)pyrrolidin-1-yl)pyrazolo[1,5-a]pyrimidin-3-y l)-3-hydroxypyrrolidine-1-carboxamide
JOP20190092A1 (en) 2016-10-26 2019-04-25 Array Biopharma Inc PROCESS FOR THE PREPARATION OF PYRAZOLO[1,5-a]PYRIMIDINES AND SALTS THEREOF
JOP20190213A1 (en) 2017-03-16 2019-09-16 Array Biopharma Inc Macrocyclic compounds as ros1 kinase inhibitors

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4908056A (en) * 1986-04-25 1990-03-13 E. I. Du Pont De Nemours And Company Heterocyclic acyl sulfonamides

Also Published As

Publication number Publication date
EA200600021A1 (en) 2006-06-30
EA009517B1 (en) 2008-02-28
IL172592A0 (en) 2006-04-10

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