ECSP066649A - EFFECTIVE PREPARATION OF A PHARMACEUTICALLY ACTIVE BASIC SUBSTANCE - Google Patents

EFFECTIVE PREPARATION OF A PHARMACEUTICALLY ACTIVE BASIC SUBSTANCE

Info

Publication number
ECSP066649A
ECSP066649A EC2006006649A ECSP066649A ECSP066649A EC SP066649 A ECSP066649 A EC SP066649A EC 2006006649 A EC2006006649 A EC 2006006649A EC SP066649 A ECSP066649 A EC SP066649A EC SP066649 A ECSP066649 A EC SP066649A
Authority
EC
Ecuador
Prior art keywords
pharmaceutically active
basic substance
effective preparation
active basic
preparation
Prior art date
Application number
EC2006006649A
Other languages
Spanish (es)
Inventor
Wolfgang Wiehl
Irene Loose
Ralf Buellesbach
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Publication of ECSP066649A publication Critical patent/ECSP066649A/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0007Effervescent
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/16Amides, e.g. hydroxamic acids
    • A61K31/165Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide
    • A61K31/167Amides, e.g. hydroxamic acids having aromatic rings, e.g. colchicine, atenolol, progabide having the nitrogen of a carboxamide group directly attached to the aromatic ring, e.g. lidocaine, paracetamol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/02Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Emergency Medicine (AREA)
  • Biomedical Technology (AREA)
  • Urology & Nephrology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)

Abstract

El objeto de la presente invención es una preparación efervescente que contiene una sal efervescente, al menos una sustancia básica farmacéuticamente activa y opcionalmente uno o más principios activos adicionales, caracterizada porque evita la alcalinización de la orina y con ello una acumulación aumentada de la sustancia básica farmacéuticamente activa, un fármaco que contiene esta preparación efervescente, procedimientos para su preparación y su uso.The object of the present invention is an effervescent preparation containing an effervescent salt, at least one pharmaceutically active basic substance and optionally one or more additional active ingredients, characterized in that it prevents the alkalization of the urine and thereby an increased accumulation of the basic substance pharmaceutically active, a drug that contains this effervescent preparation, procedures for its preparation and its use.

EC2006006649A 2003-12-19 2006-06-16 EFFECTIVE PREPARATION OF A PHARMACEUTICALLY ACTIVE BASIC SUBSTANCE ECSP066649A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE10359790A DE10359790A1 (en) 2003-12-19 2003-12-19 Effervescent preparation of a basic pharmaceutically active substance

Publications (1)

Publication Number Publication Date
ECSP066649A true ECSP066649A (en) 2006-10-25

Family

ID=34683574

Family Applications (1)

Application Number Title Priority Date Filing Date
EC2006006649A ECSP066649A (en) 2003-12-19 2006-06-16 EFFECTIVE PREPARATION OF A PHARMACEUTICALLY ACTIVE BASIC SUBSTANCE

Country Status (16)

Country Link
EP (1) EP1696874A1 (en)
JP (1) JP2007515418A (en)
KR (1) KR20060109492A (en)
CN (1) CN1893920A (en)
AR (1) AR046955A1 (en)
AU (1) AU2004308590A1 (en)
BR (1) BRPI0417796A (en)
CA (1) CA2550342A1 (en)
DE (1) DE10359790A1 (en)
EC (1) ECSP066649A (en)
IL (1) IL176356A0 (en)
MA (1) MA28276A1 (en)
MX (1) MXPA06006658A (en)
NO (1) NO20063327L (en)
WO (1) WO2005063199A1 (en)
ZA (1) ZA200604946B (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US9078824B2 (en) 2007-09-24 2015-07-14 The Procter & Gamble Company Composition and method of stabilized sensitive ingredient
TR201107202T1 (en) * 2008-11-11 2012-02-21 Berko �La� Ve K�Mya Sanay� A.�. A pharmaceutical composition comprising ibuprofen, pseudoephedrine and chlorpheniramine.
KR101057640B1 (en) * 2009-05-27 2011-08-18 (주)다산메디켐 Multi-layer tablet comprising an effervescent layer
WO2013109224A1 (en) * 2012-01-18 2013-07-25 Mahmut Bilgic Pharmaceutical compositions comprising diclofenac
CN104622831B (en) * 2013-11-06 2018-06-22 江苏豪森药业集团有限公司 A kind of oral tablet and preparation method thereof
CN107951034B (en) * 2017-12-01 2021-03-23 郑州拓洋生物工程有限公司 Vitamin effervescent preparation and preparation method thereof

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4613497A (en) * 1984-02-29 1986-09-23 Health Products Development, Inc. Dry, water-foamable pharmaceutical compositions
CA2021548A1 (en) * 1989-09-01 1991-03-02 Ronald Nash Duvall Effervescent cold or sinus allergy medicine composition having reduced sodium content
CA2084028A1 (en) * 1991-11-27 1993-05-28 Harish B. Pandya Hot flu composition
AU7407194A (en) * 1993-08-03 1995-02-28 Warner-Lambert Company Pleasant tasting effervescent cold/allergy medications
JP2000063269A (en) * 1998-08-20 2000-02-29 Taiho Yakuhin Kogyo Kk Solid preparation

Also Published As

Publication number Publication date
CA2550342A1 (en) 2005-07-14
CN1893920A (en) 2007-01-10
WO2005063199A1 (en) 2005-07-14
BRPI0417796A (en) 2007-03-20
MA28276A1 (en) 2006-11-01
JP2007515418A (en) 2007-06-14
AU2004308590A1 (en) 2005-07-14
EP1696874A1 (en) 2006-09-06
DE10359790A1 (en) 2005-07-21
KR20060109492A (en) 2006-10-20
IL176356A0 (en) 2006-10-05
AR046955A1 (en) 2006-01-04
NO20063327L (en) 2006-07-18
MXPA06006658A (en) 2006-08-31
ZA200604946B (en) 2007-09-26

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