ECSP077207A - INDOLIL RENT AMINO SUBSTITUTED DERIVATIVES AS NEW INHIBITORS OF HISTONA DESACETILASA - Google Patents

INDOLIL RENT AMINO SUBSTITUTED DERIVATIVES AS NEW INHIBITORS OF HISTONA DESACETILASA

Info

Publication number
ECSP077207A
ECSP077207A ECSP077207A ECSP077207A EC SP077207 A ECSP077207 A EC SP077207A EC SP077207 A ECSP077207 A EC SP077207A EC SP077207 A ECSP077207 A EC SP077207A
Authority
EC
Ecuador
Prior art keywords
desacetilasa
histona
indolil
rent
substituted derivatives
Prior art date
Application number
Other languages
Spanish (es)
Inventor
Marc Gustaaf Celine Verdonck
Patrick Rene Angibaud
Bruno Roux
Isabelle Noelle Consta Pilatte
Holte Peter Ten
Janine Arts
Emelen Kristof Van
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of ECSP077207A publication Critical patent/ECSP077207A/en

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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

La invención comprende nuevos compuestos de fórmula (I) en la cual R1, R2, R3, X e Y tienen significados definidos, que tienen actividad inhibitoria de la enzima histona desacetilasa; su preparación, composiciones que los contienen y su uso como medicamento.The invention comprises new compounds of formula (I) in which R1, R2, R3, X and Y have defined meanings, which have histone deacetylase enzyme inhibitory activity; their preparation, compositions containing them and their use as a medicine.

ECSP077207 2004-07-29 2007-01-26 INDOLIL RENT AMINO SUBSTITUTED DERIVATIVES AS NEW INHIBITORS OF HISTONA DESACETILASA ECSP077207A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US59218204P 2004-07-29 2004-07-29

Publications (1)

Publication Number Publication Date
ECSP077207A true ECSP077207A (en) 2007-02-28

Family

ID=40433503

Family Applications (1)

Application Number Title Priority Date Filing Date
ECSP077207 ECSP077207A (en) 2004-07-29 2007-01-26 INDOLIL RENT AMINO SUBSTITUTED DERIVATIVES AS NEW INHIBITORS OF HISTONA DESACETILASA

Country Status (1)

Country Link
EC (1) ECSP077207A (en)

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