ECSP088723A - New enantiomerically pure beta-agonists, procedures for their preparation and use as medicines - Google Patents
New enantiomerically pure beta-agonists, procedures for their preparation and use as medicinesInfo
- Publication number
- ECSP088723A ECSP088723A EC2008008723A ECSP088723A ECSP088723A EC SP088723 A ECSP088723 A EC SP088723A EC 2008008723 A EC2008008723 A EC 2008008723A EC SP088723 A ECSP088723 A EC SP088723A EC SP088723 A ECSP088723 A EC SP088723A
- Authority
- EC
- Ecuador
- Prior art keywords
- medicines
- preparation
- enantiomerically pure
- agonists
- procedures
- Prior art date
Links
- 229940079593 drug Drugs 0.000 title abstract 3
- 239000003814 drug Substances 0.000 title abstract 3
- 238000000034 method Methods 0.000 title abstract 2
- 229940125388 beta agonist Drugs 0.000 title 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 210000002345 respiratory system Anatomy 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/538—1,4-Oxazines, e.g. morpholine ortho- or peri-condensed with carbocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/02—Drugs for dermatological disorders for treating wounds, ulcers, burns, scars, keloids, or the like
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pulmonology (AREA)
- Immunology (AREA)
- Dermatology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
La presente invención se refiere a compuestos enantioméricamente puros de la fórmula 1 1en donde los radicales n, B, X, R1, m e Ym- pueden tener los significados mencionados en las reivindicaciones y en la descripción, a procedimientos para su preparación, así como a su preparación como medicamentos, en especial como medicamentos para el tratamiento de enfermedades de las vías respiratorias.The present invention relates to enantiomerically pure compounds of the formula 1 in which the radicals n, B, X, R1, I and Ym- can have the meanings mentioned in the claims and in the description, to processes for their preparation, as well as to its preparation as medicines, especially as medicines for the treatment of diseases of the respiratory tract.
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP06111191 | 2006-03-15 | ||
| EP06111342 | 2006-03-17 | ||
| EP06111338 | 2006-03-17 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ECSP088723A true ECSP088723A (en) | 2008-10-31 |
Family
ID=38006901
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EC2008008723A ECSP088723A (en) | 2006-03-15 | 2008-09-08 | New enantiomerically pure beta-agonists, procedures for their preparation and use as medicines |
Country Status (16)
| Country | Link |
|---|---|
| US (2) | US7534789B2 (en) |
| EP (1) | EP1996581A1 (en) |
| JP (1) | JP2009530245A (en) |
| KR (1) | KR20080106973A (en) |
| AR (1) | AR059836A1 (en) |
| AU (1) | AU2007224420A1 (en) |
| BR (1) | BRPI0709601A2 (en) |
| CA (1) | CA2643026A1 (en) |
| EA (1) | EA200801894A1 (en) |
| EC (1) | ECSP088723A (en) |
| MX (1) | MX2008011700A (en) |
| NO (1) | NO20083508L (en) |
| PE (1) | PE20080142A1 (en) |
| TW (1) | TW200804360A (en) |
| UY (1) | UY30207A1 (en) |
| WO (1) | WO2007104772A1 (en) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US7799336B2 (en) | 2004-04-30 | 2010-09-21 | Allergan, Inc. | Hypotensive lipid-containing biodegradable intraocular implants and related methods |
| PE20080142A1 (en) * | 2006-03-15 | 2008-04-14 | Boehringer Ingelheim Int | ENANTHOMERICALLY PURE BETA-AGONISTS AND THEIR PREPARATION PROCEDURES |
| SG11201603383VA (en) | 2013-10-31 | 2016-05-30 | Allergan Inc | Prostamide-containing intraocular implants and methods of use thereof |
Family Cites Families (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE2609645A1 (en) * | 1976-03-09 | 1977-09-15 | Boehringer Sohn Ingelheim | AMINOALKYLHETEROCYCLES |
| US7056916B2 (en) | 2002-11-15 | 2006-06-06 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Medicaments for the treatment of chronic obstructive pulmonary disease |
| DE10253282A1 (en) * | 2002-11-15 | 2004-05-27 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Treatment of chronic obstructive pulmonary disease, using new or known N-substituted 2-amino-1-(benz-(1,4)-oxazin-3-on-8-yl)-ethanol derivative beta-mimetic agents, suitable for once-daily administration |
| DE102004003428A1 (en) | 2004-01-23 | 2005-08-11 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | New long-acting beta-2 agonists, and their use as pharmaceuticals |
| US7220742B2 (en) | 2004-05-14 | 2007-05-22 | Boehringer Ingelheim International Gmbh | Enantiomerically pure beta agonists, process for the manufacture thereof and use thereof as medicaments |
| DE102004024454A1 (en) * | 2004-05-14 | 2005-12-08 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | Novel enantiomerically pure beta agonists, process for their preparation and their use as pharmaceuticals |
| DE102004045648A1 (en) * | 2004-09-21 | 2006-03-23 | Boehringer Ingelheim Pharma Gmbh & Co. Kg | New betamimetics for the treatment of respiratory diseases |
| US20080176744A1 (en) | 2005-03-10 | 2008-07-24 | Basf Aktiengesellschaft | Use of 4-Aminopyrimidines for Controlling Harmful Fungi, Novel 4-Aminopyrimidines, Processes for Their Preparation and Compositions Comprising Them |
| CA2642239A1 (en) * | 2006-02-16 | 2007-08-23 | Boehringer Ingelheim International Gmbh | Drug combinations for the treatment of respiratory tract diseases |
| PE20080142A1 (en) * | 2006-03-15 | 2008-04-14 | Boehringer Ingelheim Int | ENANTHOMERICALLY PURE BETA-AGONISTS AND THEIR PREPARATION PROCEDURES |
-
2007
- 2007-03-13 PE PE2007000271A patent/PE20080142A1/en not_active Application Discontinuation
- 2007-03-14 AU AU2007224420A patent/AU2007224420A1/en not_active Abandoned
- 2007-03-14 CA CA002643026A patent/CA2643026A1/en not_active Abandoned
- 2007-03-14 KR KR1020087025108A patent/KR20080106973A/en not_active Withdrawn
- 2007-03-14 EA EA200801894A patent/EA200801894A1/en unknown
- 2007-03-14 MX MX2008011700A patent/MX2008011700A/en not_active Application Discontinuation
- 2007-03-14 TW TW096108791A patent/TW200804360A/en unknown
- 2007-03-14 BR BRPI0709601-1A patent/BRPI0709601A2/en not_active Application Discontinuation
- 2007-03-14 AR ARP070101031A patent/AR059836A1/en unknown
- 2007-03-14 EP EP07726883A patent/EP1996581A1/en not_active Withdrawn
- 2007-03-14 WO PCT/EP2007/052389 patent/WO2007104772A1/en not_active Ceased
- 2007-03-14 UY UY30207A patent/UY30207A1/en not_active Application Discontinuation
- 2007-03-14 JP JP2008558815A patent/JP2009530245A/en active Pending
- 2007-03-15 US US11/686,565 patent/US7534789B2/en not_active Expired - Fee Related
-
2008
- 2008-08-13 NO NO20083508A patent/NO20083508L/en not_active Application Discontinuation
- 2008-09-08 EC EC2008008723A patent/ECSP088723A/en unknown
-
2009
- 2009-04-07 US US12/419,505 patent/US7939658B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| CA2643026A1 (en) | 2007-09-20 |
| WO2007104772A1 (en) | 2007-09-20 |
| WO2007104772A9 (en) | 2007-11-22 |
| MX2008011700A (en) | 2008-09-24 |
| NO20083508L (en) | 2008-09-30 |
| EA200801894A1 (en) | 2009-02-27 |
| EP1996581A1 (en) | 2008-12-03 |
| PE20080142A1 (en) | 2008-04-14 |
| TW200804360A (en) | 2008-01-16 |
| JP2009530245A (en) | 2009-08-27 |
| AR059836A1 (en) | 2008-04-30 |
| UY30207A1 (en) | 2007-10-31 |
| US7534789B2 (en) | 2009-05-19 |
| AU2007224420A1 (en) | 2007-09-20 |
| US20070249595A1 (en) | 2007-10-25 |
| BRPI0709601A2 (en) | 2011-07-19 |
| US20090306068A1 (en) | 2009-12-10 |
| KR20080106973A (en) | 2008-12-09 |
| US7939658B2 (en) | 2011-05-10 |
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